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Found 649 with Last Name = 'el-gamal' and Initial = 'm'
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525467(CHEMBL4450307)
Affinity DataKi:  18nMAssay Description:Inhibition of human carbonic anhydrase 9More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525475(CHEMBL4471122)
Affinity DataKi:  18nMAssay Description:Inhibition of human carbonic anhydrase 9More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525476(CHEMBL4581749)
Affinity DataKi:  18nMAssay Description:Inhibition of human carbonic anhydrase 9More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525479(CHEMBL4531097)
Affinity DataKi:  18nMAssay Description:Inhibition of human carbonic anhydrase 9More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525477(CHEMBL4554643)
Affinity DataKi:  18nMAssay Description:Inhibition of human carbonic anhydrase 9More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525478(CHEMBL4533212)
Affinity DataKi:  18nMAssay Description:Inhibition of human carbonic anhydrase 9More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525466(CHEMBL4440045)
Affinity DataKi:  18nMAssay Description:Inhibition of human carbonic anhydrase 9More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525474(CHEMBL4457432)
Affinity DataKi:  18nMAssay Description:Inhibition of human carbonic anhydrase 9More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 9(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525483(CHEMBL4546356)
Affinity DataKi:  18nMAssay Description:Inhibition of human carbonic anhydrase 9More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525479(CHEMBL4531097)
Affinity DataKi:  29nMAssay Description:Inhibition of human carbonic anhydrase 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525476(CHEMBL4581749)
Affinity DataKi:  29nMAssay Description:Inhibition of human carbonic anhydrase 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525483(CHEMBL4546356)
Affinity DataKi:  29nMAssay Description:Inhibition of human carbonic anhydrase 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525478(CHEMBL4533212)
Affinity DataKi:  29nMAssay Description:Inhibition of human carbonic anhydrase 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525477(CHEMBL4554643)
Affinity DataKi:  29nMAssay Description:Inhibition of human carbonic anhydrase 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525466(CHEMBL4440045)
Affinity DataKi:  29nMAssay Description:Inhibition of human carbonic anhydrase 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525475(CHEMBL4471122)
Affinity DataKi:  29nMAssay Description:Inhibition of human carbonic anhydrase 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525467(CHEMBL4450307)
Affinity DataKi:  29nMAssay Description:Inhibition of human carbonic anhydrase 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525474(CHEMBL4457432)
Affinity DataKi:  29nMAssay Description:Inhibition of human carbonic anhydrase 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525477(CHEMBL4554643)
Affinity DataKi:  42nMAssay Description:Inhibition of human carbonic anhydrase 4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 4(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525474(CHEMBL4457432)
Affinity DataKi:  76nMAssay Description:Inhibition of human carbonic anhydrase 4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585092(CHEMBL5087577)
Affinity DataIC50:  0.0700nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50136297(CHEMBL136112 | Sulfamic acid 2-adamantan-2-ylidene...)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of steroid sulfatase (unknown origin) expressed in human MCF7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50136297(CHEMBL136112 | Sulfamic acid 2-adamantan-2-ylidene...)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of steroid sulfatase (unknown origin) expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50121079(CHEMBL3622064)
Affinity DataIC50:  0.25nMAssay Description:Inhibition of aromatase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50118560(CHEMBL262050 | Sulfamic acid 2-adamantan-1-yl-4-ox...)
Affinity DataIC50:  0.340nMAssay Description:Inhibition of human steroid sulfatase by fluorimetric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525470(CHEMBL4456330)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of human placental steroid sulfatase expressed in HEK293 cells using [3H] E1S as substrate after 2 hrs by liquid scintillation counting me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525473(CHEMBL4520442)
Affinity DataIC50:  0.680nMAssay Description:Inhibition of steroid sulfatase in human MCF7 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50428286(DABRAFENIB | GSK2118436A)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin)More data for this Ligand-Target Pair
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50134329(CHEMBL122708 | Sulfamic acid (11R,12S,15S,16S)-13-...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of human placental steroid sulfatase expressed in HEK293 cells using [3H] E1S as substrate after 2 hrs by liquid scintillation counting me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50587662(CHEMBL1915474)
Affinity DataIC50:  0.978nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin) incubated for 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585081(CHEMBL5086749)
Affinity DataIC50:  0.980nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525469(CHEMBL4517286)
Affinity DataIC50:  1nMAssay Description:Inhibition of steroid sulfatase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50121063(CHEMBL3622010)
Affinity DataIC50:  1nMAssay Description:Inhibition of steroid sulfatase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525472(CHEMBL4459312)
Affinity DataIC50:  1nMAssay Description:Inhibition of steroid sulfatase in human MCF7 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525481(CHEMBL4436186)
Affinity DataIC50:  1nMAssay Description:Inhibition of steroid sulfatase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM435721(US10570155, Compound 25III | US11332479, Compound ...)
Affinity DataIC50:  1nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585092(CHEMBL5087577)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of human wild type CRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50460035(CHEMBL4227505)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of CSF1R (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585085(CHEMBL5080553)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of human BRAF V600E mutant using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation co...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50167323(CHEMBL3797224)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of steroid sulfatase in human JEG-3 cells assessed as [14C]-Estrone formation using [3H]E1S as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM5447(CHEMBL939 | GEFITINIB | Iressa | N-(3-Chloro-4-flu...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of EGFR (unknown origin) incubated for 40 mins by intrinsic ATPase activity luminescence assayMore data for this Ligand-Target Pair
TargetCytochrome P450 2D6(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM8610(1-[4-(4-{[(2R,4S)-2-(2,4-dichlorophenyl)-2-(1H-imi...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of CYP2D6 (unknown origin) using EOMCC as a substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585095(CHEMBL5079413)
Affinity DataIC50:  2nMAssay Description:Inhibition of human wild type CRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585092(CHEMBL5087577)
Affinity DataIC50:  2nMAssay Description:Inhibition of human wild type BRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM13058(6-oxo-6,7,8,9,10,11-hexahydrocyclohepta[c]chromen-...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of steroid sulfatase in human JEG3 cells using [3H] E1S as substrate incubated for 20 hrs by scintillation spectrometry analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585088(CHEMBL5073246)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of human wild type CRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSteryl-sulfatase(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50525471(CHEMBL4442535)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of steroid sulfatase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM8610(1-[4-(4-{[(2R,4S)-2-(2,4-dichlorophenyl)-2-(1H-imi...)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of CYP3A4 (unknown origin) using BOMCC as a substrate incubated for 20 mins by fluorescence based analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase B-raf(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50563431(CHEMBL4793723)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of BRAF V600E mutant (unknown origin) using Ser/Thr 03 as substrate after 1 hr in presence of ATP by Z'-LYTE assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRAF proto-oncogene serine/threonine-protein kinase(Homo sapiens (Human))
National Research Centre (Nrc)

Curated by ChEMBL
LigandPNGBDBM50585085(CHEMBL5080553)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of human wild type CRAF using myelin basic protein as substrate in presence of [gamma-33P]ATP incubated for 40 mins by scintillation count...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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