Compile Data Set for Download or QSAR
maximum 50k data
Found 89 with Last Name = 'elias' and Initial = 'r'
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92800(Bisanilinopyrimidine, 3o | US9249124, 16)
Affinity DataIC50:  0.800nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92810(Bisanilinopyrimidine, 6c | US9249124, 26)
Affinity DataIC50:  2nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM87054(Bisanilinopyrimidine inhibitor, 8 | Bisanilinopyri...)
Affinity DataIC50:  2.10nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM87053(Bisanilinopyrimidine inhibitor, 7 | Bisanilinopyri...)
Affinity DataIC50:  2.5nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92844(Bisanilinopyrimidine, 12b | US9249124, 60)
Affinity DataIC50:  2.90nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92846(Bisanilinopyrimidine, 12d | US9249124, 62)
Affinity DataIC50:  3nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92843(Bisanilinopyrimidine, 12a | US9249124, 59)
Affinity DataIC50:  3.10nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92805(Bisanilinopyrimidine, 4d | US9249124, 21)
Affinity DataIC50:  3.17nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92817(Bisanilinopyrimidine, 6j | US9249124, 33)
Affinity DataIC50:  3.30nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM87052(Bisanilinopyrimidine inhibitor, 6 | Bisanilinopyri...)
Affinity DataIC50:  3.70nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92799(Bisanilinopyrimidine, 3n | US9249124, 15)
Affinity DataIC50:  3.90nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92812(Bisanilinopyrimidine, 6e | US9249124, 28)
Affinity DataIC50:  4nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92827(Bisanilinopyrimidine, 6t)
Affinity DataIC50:  4.5nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92803(Bisanilinopyrimidine, 3r | US9249124, 19)
Affinity DataIC50:  5.10nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM87048(Bisanilinopyrimidine inhibitor, 2 | Bisanilinopyri...)
Affinity DataIC50:  6.10nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92818(Bisanilinopyrimidine, 6k)
Affinity DataIC50:  6.60nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92825(Bisanilinopyrimidine, 6r | US9249124, 41)
Affinity DataIC50:  8.5nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM87047(Bisanilinopyrimidine inhibitor, 1 | Bisanilinopyri...)
Affinity DataIC50:  10nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
TargetAurora kinase B(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92841(Bisanilinopyrimidine, 9m | US9249124, 57)
Affinity DataIC50:  10.7nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM16011(2-{[5-fluoro-2-(phenylamino)pyrimidin-4-yl]amino}b...)
Affinity DataIC50:  11.3nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92840(Bisanilinopyrimidine, 9l | US9249124, 56)
Affinity DataIC50:  12.3nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92841(Bisanilinopyrimidine, 9m | US9249124, 57)
Affinity DataIC50:  14.4nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92845(Bisanilinopyrimidine, 12c | US9249124, 61)
Affinity DataIC50:  17.3nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92830(Bisanilinopyrimidine, 9c | US9249124, 46)
Affinity DataIC50:  18nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92802(Bisanilinopyrimidine, 3q | US9249124, 18)
Affinity DataIC50:  18.3nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92822(Bisanilinopyrimidine, 6o)
Affinity DataIC50:  18.7nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92801(Bisanilinopyrimidine, 3p | US9249124, 17)
Affinity DataIC50:  19.9nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92842(Bisanilinopyrimidine, 9n | US9249124, 58)
Affinity DataIC50:  21.2nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92838(Bisanilinopyrimidine, 9j | US9249124, 54)
Affinity DataIC50:  21.4nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92839(Bisanilinopyrimidine, 9k | US9249124, 55)
Affinity DataIC50:  23.2nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92838(Bisanilinopyrimidine, 9j | US9249124, 54)
Affinity DataIC50:  25.6nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92835(Bisanilinopyrimidine, 9h | US9249124, 51)
Affinity DataIC50:  27nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM87051(Bisanilinopyrimidine inhibitor, 5 | Bisanilinopyri...)
Affinity DataIC50:  28nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92829(Bisanilinopyrimidine, 9b | US9249124, 44)
Affinity DataIC50:  28.1nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92839(Bisanilinopyrimidine, 9k | US9249124, 55)
Affinity DataIC50:  30nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92836(Bisanilinopyrimidine, 6p | US9249124, 52)
Affinity DataIC50:  30.2nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92820(Bisanilinopyrimidine, 6m | US9249124, 36)
Affinity DataIC50:  35nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM87050(Bisanilinopyrimidine inhibitor, 4 | Bisanilinopyri...)
Affinity DataIC50:  35.1nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92793(Bisanilinopyrimidine, 3g)
Affinity DataIC50:  38.2nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
TargetAurora kinase B(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92840(Bisanilinopyrimidine, 9l | US9249124, 56)
Affinity DataIC50:  40.4nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM87055(Bisanilinopyrimidine inhibitor, 9 | Bisanilinopyri...)
Affinity DataIC50:  43nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
TargetAurora kinase B(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92837(Bisanilinopyrimidine, 9i | US9249124, 53)
Affinity DataIC50:  43.3nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92831(Bisanilinopyrimidine, 9d | US9249124, 47)
Affinity DataIC50:  44.9nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92813(Bisanilinopyrimidine, 6f | US9249124, 29)
Affinity DataIC50:  46.6nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92836(Bisanilinopyrimidine, 6p | US9249124, 52)
Affinity DataIC50:  50.2nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92826(Bisanilinopyrimidine, 6s | US9249124, 42)
Affinity DataIC50:  50.2nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase B(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92842(Bisanilinopyrimidine, 9n | US9249124, 58)
Affinity DataIC50:  56.6nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM16005(2-[(2-{[4-(morpholin-4-yl)phenyl]amino}pyrimidin-4...)
Affinity DataIC50:  57.6nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Tel Aviv University

Curated by ChEMBL
LigandPNGBDBM31774(CHEMBL104 | Canesten | Clotrimazole | Lotrimin | M...)
Affinity DataIC50:  67nMAssay Description:Inhibition of recombinant human CYP3A4 using Luciferin-PPXE as substrate preincubated for 10 mins followed by NADPH addition measured after 15 mins b...More data for this Ligand-Target Pair
TargetAurora kinase A(Homo sapiens (Human))
Moffitt Cancer Center

LigandPNGBDBM92832(Bisanilinopyrimidine, 9e)
Affinity DataIC50:  71.2nMAssay Description:In vitro enzyme activity assay using Aurora Kinase A. More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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