Affinity DataKi: 0.100nMAssay Description:Compound was tested for inhibition of Sunflower beta-trypsinMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C delta C1b domainMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain (Wild type)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.150nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (F13G)More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity at recombinant Hsp90alpha incubated for 16 hrs by fluorescence polarization competition assayMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.351nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain (Wild type)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.720nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (T12G)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.820nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (F13G)More data for this Ligand-Target Pair
TargetRAS guanyl-releasing protein 1(Rattus norvegicus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.850nMAssay Description:Binding affinity against RAS guanyl releasing protein using [3H]- PDBu as the labeled ligandMore data for this Ligand-Target Pair
TargetSuppressor of tumorigenicity 14 protein(Homo sapiens (Human))
National Cancer Institute-Frederick
Curated by ChEMBL
National Cancer Institute-Frederick
Curated by ChEMBL
Affinity DataKi: 0.920nMAssay Description:Compound was tested for inhibition of Matriptase from human breast cancer cellsMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.08nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (L20G)More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Compound was tested for inhibition of bovine beta trypsinMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.24nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (T12G)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.41nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (Q27V)More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Binding affinity at recombinant Hsp90alpha incubated for 16 hrs by fluorescence polarization competition assayMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.01nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C delta C1b domainMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.01nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain (Wild type)More data for this Ligand-Target Pair
TargetRAS guanyl-releasing protein 1(Rattus norvegicus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.54nMAssay Description:Binding affinity against RAS guanyl releasing protein using [3H]- PDBu as the labeled ligandMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 2.71nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain (Wild type)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 3.14nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (T8G)More data for this Ligand-Target Pair
TargetRAS guanyl-releasing protein 1(Rattus norvegicus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 6.15nMAssay Description:Binding affinity against RAS guanyl releasing protein using [3H]- PDBu as the labeled ligandMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 6.59nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (L20G)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 7.80nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (F13G)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 10.7nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C delta C1b domainMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 10.8nMAssay Description:Displacement of [3H]-PDBu from protein kinase C delta C1b domain mutant (P11G)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 10.9nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (F13G)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 10.9nMAssay Description:Binding Affinity to cocaine site of dopamine transporter in caudate nuclei which was homogenized and incubated with [3H]-mazindol .More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 11.3nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (L20G)More data for this Ligand-Target Pair
TargetRAS guanyl-releasing protein 1(Rattus norvegicus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 13.9nMAssay Description:Binding affinity against RAS guanyl releasing protein using [3H]- PDBu as the labeled ligandMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 14.2nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (Q27V)More data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
University Of Michigan Cancer Center
Curated by ChEMBL
University Of Michigan Cancer Center
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Binding affinity for RasGPR3, guanine nucleotide exchange factorMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 18.4nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (T8G)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 19.1nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (T12G)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 25nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (W22G)More data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 25.3nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (T12G)More data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Compound was tested for the inhibition of norepinephrine [3H]NE reuptake into rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Inhibition of [3H]NE uptake at Norepinephrine transporter in rat parietal/occipital cortex was determinedMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 35.1nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C delta C1b domainMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Compound was tested for the inhibition of norepinephrine [3H]NE reuptake into rat cortical membranesMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Inhibition of [3H]DA binding to dopamine transporter of rat brain synaptosomesMore data for this Ligand-Target Pair
TargetRas guanyl-releasing protein 3(Homo sapiens (Human))
University Of Michigan Cancer Center
Curated by ChEMBL
University Of Michigan Cancer Center
Curated by ChEMBL
Affinity DataKi: 42nMAssay Description:Binding affinity for RasGPR3, guanine nucleotide exchange factorMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Inhibition of [3H]NE uptake at Norepinephrine transporter in rat parietal/occipital cortex was determinedMore data for this Ligand-Target Pair
TargetProtein kinase C delta type(Mus musculus)
Georgetown University Medical Center
Curated by ChEMBL
Georgetown University Medical Center
Curated by ChEMBL
Affinity DataKi: 47.1nMAssay Description:Displacement of [3H]PDBu from protein kinase C delta C1b domain mutant (Q27V)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKi: 48nMAssay Description:Tested for the ability to displace [3H]WIN-35 428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKi: 51nMAssay Description:Inhibition of [3H]-DA Uptake at dopamine transporter in rat cortex was measured by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKi: 52nMAssay Description:Inhibition of [3H]- Mazindol binding to dopamine transporter of rat striatal membrane.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
University Of Michigan
Curated by ChEMBL
University Of Michigan
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:Inhibition of [3H]DA binding to dopamine transporter of rat brain synaptosomesMore data for this Ligand-Target Pair