Affinity DataIC50: 15nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
Affinity DataIC50: 380nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
Affinity DataIC50: 460nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
Affinity DataIC50: 480nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
Affinity DataIC50: 535nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
Affinity DataIC50: 660nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 870nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
Affinity DataIC50: 996nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.33E+3nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 2.33E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 2.63E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 3.55E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 3.89E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 8.51E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
Affinity DataIC50: 1.28E+4nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 2.04E+4nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
Affinity DataIC50: 6.11E+4nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
Affinity DataIC50: 6.23E+4nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
Affinity DataIC50: 9.00E+4nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna
Curated by ChEMBL
Medical University Vienna
Curated by ChEMBL
Affinity DataIC50: 1.41E+5nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataEC50: 5.53E+4nMAssay Description:Modulation of GABAA alpha1beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chlorid...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataEC50: 1.02E+5nMAssay Description:Modulation of GABAA alpha1beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chlorid...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataEC50: 1.60E+4nMAssay Description:Modulation of GABAA alpha3beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as modulation of GABA-induced chloride ...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataEC50: 3.68E+4nMAssay Description:Modulation of GABAA alpha1beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chlorid...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataEC50: 6.77E+4nMAssay Description:Modulation of GABAA alpha1beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chlorid...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataEC50: 7.08E+4nMAssay Description:Modulation of GABAA alpha1beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chlorid...More data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Vienna
Curated by ChEMBL
University Of Vienna
Curated by ChEMBL
Affinity DataEC50: 1.38E+4nMAssay Description:Modulation of GABAA alpha1beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chlorid...More data for this Ligand-Target Pair