Compile Data Set for Download or QSAR
maximum 50k data
Found 60 with Last Name = 'erker' and Initial = 't'
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50217120(1,2-dihydro-7-methoxy-3-(2,3,4-trimethoxyphenyl)-n...)
Affinity DataIC50:  15nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50217117(2-(2,3,4-trimethoxyphenyl)-1H-indene | CHEMBL22856...)
Affinity DataIC50:  30nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50217121(1,2-dihydro-3-(3,4-dimethoxyphenyl)-7-methoxynapht...)
Affinity DataIC50:  30nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009280(CHEMBL3233494)
Affinity DataIC50:  40nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009293(CHEMBL3233505)
Affinity DataIC50:  60nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009290(CHEMBL3233503)
Affinity DataIC50:  120nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009279(CHEMBL2220507)
Affinity DataIC50:  130nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009289(CHEMBL3233502)
Affinity DataIC50:  140nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009282(CHEMBL3233496)
Affinity DataIC50:  140nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009292(CHEMBL3233504)
Affinity DataIC50:  140nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50217121(1,2-dihydro-3-(3,4-dimethoxyphenyl)-7-methoxynapht...)
Affinity DataIC50:  380nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50217115(2-(2-methoxyphenyl)-1H-indene | CHEMBL376583)
Affinity DataIC50:  460nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50217119(1,2-dihydro-3-(2,3,4-trimethoxyphenyl)naphthalene ...)
Affinity DataIC50:  480nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM23926((E)-resveratrol | 5-[(E)-2-(4-hydroxyphenyl)etheny...)
Affinity DataIC50:  535nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009277(CHEMBL3233492)
Affinity DataIC50:  650nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50217119(1,2-dihydro-3-(2,3,4-trimethoxyphenyl)naphthalene ...)
Affinity DataIC50:  660nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009278(CHEMBL3233493)
Affinity DataIC50:  870nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM23926((E)-resveratrol | 5-[(E)-2-(4-hydroxyphenyl)etheny...)
Affinity DataIC50:  996nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009284(CHEMBL3233497)
Affinity DataIC50:  1.15E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50217117(2-(2,3,4-trimethoxyphenyl)-1H-indene | CHEMBL22856...)
Affinity DataIC50:  1.33E+3nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009275(CHEMBL3233220)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009283(CHEMBL3233017)
Affinity DataIC50:  1.74E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009286(CHEMBL3233499)
Affinity DataIC50:  2.33E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009285(CHEMBL3233498)
Affinity DataIC50:  2.63E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009274(CHEMBL3233219)
Affinity DataIC50:  2.75E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009281(CHEMBL3233495)
Affinity DataIC50:  3.55E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009287(CHEMBL3233500)
Affinity DataIC50:  3.89E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009273(CHEMBL3233218)
Affinity DataIC50:  8.51E+3nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009276(CHEMBL3233491)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50217118(5-(2-1H-indenyl)-1,3-benzodioxole | CHEMBL229139)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009294(CHEMBL3233506)
Affinity DataIC50:  2.04E+4nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50217116(1,2-dihydro-3-(3,4-dimethoxyphenyl)naphthalene | C...)
Affinity DataIC50:  6.11E+4nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50217115(2-(2-methoxyphenyl)-1H-indene | CHEMBL376583)
Affinity DataIC50:  6.23E+4nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM22360(2-(acetyloxy)benzoate | 2-(acetyloxy)benzoic acid ...)
Affinity DataIC50:  9.00E+4nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50217122(5-(1,2-dihydro-3-naphthalenyl)-1,3-benzodioxole | ...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50217118(5-(2-1H-indenyl)-1,3-benzodioxole | CHEMBL229139)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM22360(2-(acetyloxy)benzoate | 2-(acetyloxy)benzoic acid ...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50217116(1,2-dihydro-3-(3,4-dimethoxyphenyl)naphthalene | C...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50217120(1,2-dihydro-7-methoxy-3-(2,3,4-trimethoxyphenyl)-n...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human recombinant COX2 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50217122(5-(1,2-dihydro-3-naphthalenyl)-1,3-benzodioxole | ...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ovine COX1 by measuring PGE2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetATP-dependent translocase ABCB1(Homo sapiens (Human))
Medical University Vienna

Curated by ChEMBL
LigandPNGBDBM50009288(CHEMBL3233501)
Affinity DataIC50:  1.41E+5nMAssay Description:Inhibition of P-gp-mediated daunorubicin efflux in human CCRF-CEM/VCR1000 cells measured within 1 hr by FACS flow cytometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50497215(CHEMBL3289482)
Affinity DataEC50:  5.53E+4nMAssay Description:Modulation of GABAA alpha1beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chlorid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50497207(CHEMBL3289501)
Affinity DataEC50:  1.02E+5nMAssay Description:Modulation of GABAA alpha1beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chlorid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-2/gamma-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50497208(CHEMBL3289196)
Affinity DataEC50:  1.60E+4nMAssay Description:Modulation of GABAA alpha3beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as modulation of GABA-induced chloride ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50497209(CHEMBL3289485)
Affinity DataEC50:  3.68E+4nMAssay Description:Modulation of GABAA alpha1beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chlorid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50497210(CHEMBL3289204)
Affinity DataEC50:  6.77E+4nMAssay Description:Modulation of GABAA alpha1beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chlorid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50497211(CHEMBL3289476)
Affinity DataEC50:  7.08E+4nMAssay Description:Modulation of GABAA alpha1beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chlorid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Homo sapiens (Human))
University Of Vienna

Curated by ChEMBL
LigandPNGBDBM50497208(CHEMBL3289196)
Affinity DataEC50:  1.38E+4nMAssay Description:Modulation of GABAA alpha1beta2gamma2S receptor (unknown origin) expressed in Xenopus laevis oocytes assessed as potentiation of GABA-induced chlorid...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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