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Found 147 with Last Name = 'escher' and Initial = 'e'
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Universite De Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50313242(CHEMBL1076603 | [Sar1,Bpa3]AngII)
Affinity DataKi:  0.700nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Universite De Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50313247(CHEMBL1076632 | [Sar1,Bpa8]AngII)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Universite De Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50313240(CHEMBL1076633 | [Sar1,Tdf8]AngII)
Affinity DataKi:  0.900nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Universite De Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50313241(CHEMBL1076604 | [Sar1,Tdf3]AngII)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50406623(CHEMBL2115369)
Affinity DataKi:  1.40nMAssay Description:Negative log of Kd for Vasopressin V1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V1a receptor(RAT)
University Of Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50406622(CHEMBL2115364)
Affinity DataKi:  1.90nMAssay Description:Inhibition of the 3 nM VP stimulation of phospholipase-C in cultured WRK cells was used as a V1-mediated assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Universite De Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50313244(CHEMBL1076601 | [Sar1,Bpa2]AngII)
Affinity DataKi:  18.3nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Universite De Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50313246(CHEMBL1076612 | [Bpa1]AngII)
Affinity DataKi:  19.4nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Universite De Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50313243(CHEMBL1076602 | [Sar1,Tdf2]AngII)
Affinity DataKi:  24.7nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Universite De Sherbrooke

Curated by ChEMBL
LigandPNGBDBM50313245(CHEMBL1076613 | [Tdf1]AngII)
Affinity DataKi:  26.4nMAssay Description:Displacement of [125I][Sar1,Ile8]Ang2 from wild-type human AT1 receptor expressed in CHO cells by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379090(CHEMBL2012527)
Affinity DataIC50:  1.36nMAssay Description:Displacement of [125I]-SDF-1alpha from human CXCR4 receptor expressed in HEK293 cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379088(CHEMBL2012525)
Affinity DataIC50:  1.56nMAssay Description:Displacement of [125I]-SDF-1alpha from human CXCR4 receptor expressed in HEK293 cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379089(CHEMBL2012526)
Affinity DataIC50:  2.22nMAssay Description:Displacement of [125I]-SDF-1alpha from human CXCR4 receptor expressed in HEK293 cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379097(CHEMBL2012524)
Affinity DataIC50:  5.67nMAssay Description:Displacement of [125I]-SDF-1alpha from human CXCR4 receptor expressed in HEK293 cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379098(CHEMBL2012523)
Affinity DataIC50:  9.57nMAssay Description:Displacement of [125I]-SDF-1alpha from human CXCR4 receptor expressed in HEK293 cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379096(CHEMBL2012652)
Affinity DataIC50:  16.5nMAssay Description:Displacement of [125I]-SDF-1alpha from human CXCR4 receptor expressed in HEK293 cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196251(CHEMBL3912312)
Affinity DataIC50:  18nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379093(CHEMBL2012531)
Affinity DataIC50:  21.2nMAssay Description:Displacement of [125I]-SDF-1alpha from human CXCR4 receptor expressed in HEK293 cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379092(CHEMBL2012530)
Affinity DataIC50:  21.7nMAssay Description:Displacement of [125I]-SDF-1alpha from human CXCR4 receptor expressed in HEK293 cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379099(CHEMBL2012653)
Affinity DataIC50:  24.9nMAssay Description:Displacement of [125I]-SDF-1alpha from human CXCR4 receptor expressed in HEK293 cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196240(CHEMBL3896146)
Affinity DataIC50:  25nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379094(CHEMBL2012532)
Affinity DataIC50:  28.3nMAssay Description:Displacement of [125I]-SDF-1alpha from human CXCR4 receptor expressed in HEK293 cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196275(CHEMBL3930215)
Affinity DataIC50:  31nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196255(CHEMBL3955461)
Affinity DataIC50:  34nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379095(CHEMBL2012651)
Affinity DataIC50:  38.6nMAssay Description:Displacement of [125I]-SDF-1alpha from human CXCR4 receptor expressed in HEK293 cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196241(CHEMBL3902240)
Affinity DataIC50:  48nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196239(CHEMBL3924163)
Affinity DataIC50:  56nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196257(CHEMBL3903301)
Affinity DataIC50:  59nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379091(CHEMBL2012528)
Affinity DataIC50:  62.0nMAssay Description:Displacement of [125I]-SDF-1alpha from human CXCR4 receptor expressed in HEK293 cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196263(CHEMBL3974242)
Affinity DataIC50:  64nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196262(CHEMBL3978794)
Affinity DataIC50:  69nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196256(CHEMBL3970509)
Affinity DataIC50:  73nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196242(CHEMBL3940962)
Affinity DataIC50:  78nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196276(CHEMBL3982241)
Affinity DataIC50:  84nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196269(CHEMBL3976727)
Affinity DataIC50:  84nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196261(CHEMBL3959440)
Affinity DataIC50:  90nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196278(CHEMBL3949729)
Affinity DataIC50:  94nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196254(CHEMBL3954553)
Affinity DataIC50:  95nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196258(CHEMBL3924080)
Affinity DataIC50:  102nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196244(CHEMBL3896065)
Affinity DataIC50:  109nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196243(CHEMBL3923006)
Affinity DataIC50:  112nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196264(CHEMBL3983197)
Affinity DataIC50:  127nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196277(CHEMBL3963508)
Affinity DataIC50:  137nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196274(CHEMBL3912645)
Affinity DataIC50:  137nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196252(CHEMBL3932032)
Affinity DataIC50:  151nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50379100(CHEMBL2012529)
Affinity DataIC50:  170nMAssay Description:Displacement of [125I]-SDF-1alpha from human CXCR4 receptor expressed in HEK293 cells after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196271(CHEMBL3933112)
Affinity DataIC50:  171nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196265(CHEMBL3894327)
Affinity DataIC50:  222nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196272(CHEMBL3942093)
Affinity DataIC50:  230nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50196267(CHEMBL3923084)
Affinity DataIC50:  267nMAssay Description:Displacement of [125I]-CXCL12 from HA-tagged human recombinant CXCR4 expressed in HEK293 cells incubated for 1 hr by gamma-radiation counting analysi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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