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Found 60 with Last Name = 'esteva-font' and Initial = 'c'
TargetUrea transporter 1(Homo sapiens (Human))
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394962(CHEMBL1394231)
Affinity DataIC50:  11nMAssay Description:Inhibition of UT-B in human erythrocytes assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394962(CHEMBL1394231)
Affinity DataIC50:  11nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50394961(CHEMBL2165788)
Affinity DataIC50:  14nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50435308(CHEMBL2391344)
Affinity DataIC50:  38nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50435309(CHEMBL2391345)
Affinity DataIC50:  43nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50435310(CHEMBL2391346)
Affinity DataIC50:  353nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50435307(CHEMBL2391349)
Affinity DataIC50: >800nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50435305(CHEMBL2391347)
Affinity DataIC50: >800nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Mus musculus)
San Francisco State University

Curated by ChEMBL
LigandPNGBDBM50435306(CHEMBL2391348)
Affinity DataIC50: >800nMAssay Description:Inhibition of UT-B in mouse acetamide-loaded erythrocyte assessed as increase of hypotonic lysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50134204(CHEMBL3740772)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50135099(CHEMBL3739636)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50135098(CHEMBL3741585)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115198(10‐(4‐bromobenzenesulfonyl)‐N...)
Affinity DataIC50:  2.80E+3nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115182(N‐(4‐ethoxyphenyl)‐8‐metho...)
Affinity DataIC50:  3.30E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115184(8‐methoxy‐N‐(4‐methoxyphen...)
Affinity DataIC50:  3.50E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115190(2‐(2‐{[(5E)‐2‐imino‐...)
Affinity DataIC50:  3.70E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115185(8‐methoxy‐N‐[3‐(methylsulf...)
Affinity DataIC50:  3.80E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50322180(3-(2,5-dimethylphenylsulfonyl)-N-isopropylthieno[2...)
Affinity DataIC50:  3.80E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115194(4‐(4,5‐dihydro‐1,3‐thiazol...)
Affinity DataIC50:  4.20E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115191((5E)‐5‐[(2‐hydroxy‐3‐...)
Affinity DataIC50:  4.60E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115190(2‐(2‐{[(5E)‐2‐imino‐...)
Affinity DataIC50:  4.80E+3nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115183(8‐hydroxy‐N‐[(3‐methoxyphe...)
Affinity DataIC50:  5.30E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115193((5E)‐5‐[(4‐hydroxy‐3‐...)
Affinity DataIC50:  6.20E+3nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115184(8‐methoxy‐N‐(4‐methoxyphen...)
Affinity DataIC50:  6.20E+3nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115191((5E)‐5‐[(2‐hydroxy‐3‐...)
Affinity DataIC50:  6.30E+3nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115192((5E)‐5‐[(2,3‐dimethoxyphenyl)met...)
Affinity DataIC50:  7.00E+3nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50134208(CHEMBL3742039)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM50322180(3-(2,5-dimethylphenylsulfonyl)-N-isopropylthieno[2...)
Affinity DataIC50:  1.50E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50134205(CHEMBL3741102)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115182(N‐(4‐ethoxyphenyl)‐8‐metho...)
Affinity DataIC50:  1.60E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50135104(CHEMBL3741981)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM50134206(CHEMBL3742032)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK-UT-A1-AQP1-YFP cells after 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115187(N‐(3‐chloro‐4‐methoxypheny...)
Affinity DataIC50:  1.90E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115185(8‐methoxy‐N‐[3‐(methylsulf...)
Affinity DataIC50:  2.00E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115186(N‐(4‐ethoxyphenyl)‐8‐metho...)
Affinity DataIC50:  2.40E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115188(N‐(3‐chloro‐4‐methylphenyl...)
Affinity DataIC50:  2.40E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115193((5E)‐5‐[(4‐hydroxy‐3‐...)
Affinity DataIC50:  2.50E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115189(N‐(3‐fluoro‐4‐methylphenyl...)
Affinity DataIC50:  2.50E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115187(N‐(3‐chloro‐4‐methoxypheny...)
Affinity DataIC50:  2.70E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM50322183(3-(4-ethylphenylsulfonyl)-N-(3-methoxypropyl)thien...)
Affinity DataIC50:  2.80E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM50135101(CHEMBL3739701)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibition of UT-B in rat whole blood after 15 mins by RBC lysis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115186(N‐(4‐ethoxyphenyl)‐8‐metho...)
Affinity DataIC50:  3.40E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115197(10‐(benzenesulfonyl)‐N‐methyl...)
Affinity DataIC50:  3.50E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115196(2‐N‐(3‐methoxyphenyl)‐4...)
Affinity DataIC50:  4.20E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM115192((5E)‐5‐[(2,3‐dimethoxyphenyl)met...)
Affinity DataIC50:  4.30E+4nMAssay Description:Erythrocyte suspension (100 µL) was added to each well of a 96-well microplate to which test compounds were added. After 15 min incubation, 20 &...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115195(1‐N‐[bis(methylsulfanyl)‐1,3,5&#...)
Affinity DataIC50:  4.50E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115198(10‐(4‐bromobenzenesulfonyl)‐N...)
Affinity DataIC50: >5.00E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 1(Rattus norvegicus (Rat))
University Of California San Francisco

LigandPNGBDBM50135106(CHEMBL3739646)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of UT-B in rat whole blood after 15 mins by RBC lysis assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115197(10‐(benzenesulfonyl)‐N‐methyl...)
Affinity DataIC50: >5.00E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrea transporter 2(Rattus norvegicus (Rat))
University Of California

Curated by ChEMBL
LigandPNGBDBM115196(2‐N‐(3‐methoxyphenyl)‐4...)
Affinity DataIC50: >5.00E+4nMAssay Description:The urea concentration dependence of UT-A1 inhibition was studied from inhibitor concentration response data (0.3 - 60 µM) using different of ur...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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