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Found 160 with Last Name = 'farrell' and Initial = 'tm'
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274627(CHEMBL483581 | N-[1-(2-carbamoylethyl)-2-[(4-cyano...)
Affinity DataIC50:  2nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM26811(CHEMBL485202 | N-[2-benzamido-1-(2-carbamoylethyl)...)
Affinity DataIC50:  3nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50275692(CHEMBL528989 | N-(1-(3-methoxypropyl)-5-((phenylam...)
Affinity DataIC50:  3nMAssay Description:Inhibition of ITK (unknown origin) by DELPHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196941(CHEMBL246365 | N2-(2-chlorobenzyl)-N4-((3-(aminome...)
Affinity DataIC50:  3nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM26813(CHEMBL460824 | N-[(2E)-5-[benzene(methyl)amido]-1-...)
Affinity DataIC50:  3nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274471(CHEMBL485556 | N-(1-(3-amino-3-oxopropyl)-5-(N-met...)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274471(CHEMBL485556 | N-(1-(3-amino-3-oxopropyl)-5-(N-met...)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274668(CHEMBL485030 | N-(1-(3-amino-3-oxopropyl)-2-(4-cya...)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196932(CHEMBL392642 | N2-(2-(methylthio)benzyl)-N4-((4-(a...)
Affinity DataIC50:  5nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196957(CHEMBL246175 | N2-(2-bromobenzyl)-N4-((4-(aminomet...)
Affinity DataIC50:  5nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM26812(CHEMBL485203 | N-[(2E)-5-[benzene(methyl)amido]-1-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50275651(CHEMBL487357 | N-(5-((cyclohexyl(methyl)amino)meth...)
Affinity DataIC50:  6nMAssay Description:Inhibition of ITK (unknown origin) by DELPHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196961(CHEMBL246174 | N2-(2-(trifluoromethylthio)benzyl)-...)
Affinity DataIC50:  6nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196936(CHEMBL246386 | N2-(2,5-dichlorobenzyl)-N4-((4-(ami...)
Affinity DataIC50:  7nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274666(CHEMBL485626 | N-[1-(2-carbamoylethyl)-2-[(4-cyano...)
Affinity DataIC50:  7nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274001(CHEMBL462301 | N-[5-(Benzoyl-ethyl-amino)-1-(2-car...)
Affinity DataIC50:  7nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196978(CHEMBL246183 | N2-(2,3-dichlorobenzyl)-N4-((4-(ami...)
Affinity DataIC50:  8nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM26830(CHEMBL457706 | N-[(2E)-5-[benzene(methyl)amido]-1-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274154(CHEMBL519033 | N-(1-(3-amino-3-oxopropyl)-5-(4,4-d...)
Affinity DataIC50:  8nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274000(CHEMBL460389 | N-(1-(3-amino-3-oxopropyl)-5-(N-met...)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274665(CHEMBL484945 | N-[1-(2-carbamoylethyl)-2-[(4-cyano...)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM26827(CHEMBL458796 | N-[(2E)-5-[benzene(methyl)amido]-1-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196959(CHEMBL396929 | N2-(2-nitrobenzyl)-N4-((4-(aminomet...)
Affinity DataIC50:  11nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274628(CHEMBL484766 | N-[1-(2-carbamoylethyl)-2-[(4-cyano...)
Affinity DataIC50:  12nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM26813(CHEMBL460824 | N-[(2E)-5-[benzene(methyl)amido]-1-...)
Affinity DataIC50:  12nMAssay Description:Inhibition of ITK (unknown origin) by DELPHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196951(CHEMBL247979 | N2-(2-(trifluoromethyl)benzyl)-N4-(...)
Affinity DataIC50:  12nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196987(CHEMBL245912 | N2-(2,3-dimethylbenzyl)-N4-((4-(ami...)
Affinity DataIC50:  13nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM26820(BMCL186218 Compound 1 | CHEMBL457886 | N-[(2E)-5-[...)
Affinity DataIC50:  14nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196991(CHEMBL245977 | N2-(2-(difluoromethyl)benzyl)-N4-((...)
Affinity DataIC50:  15nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196952(CHEMBL395690 | N2-(2-methoxybenzyl)-N4-((4-(aminom...)
Affinity DataIC50:  17nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196972(CHEMBL248183 | N2-(2-(trifluoromethoxy)benzyl)-N4-...)
Affinity DataIC50:  18nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196958(CHEMBL246159 | N2-(2-chlorobenzyl)-N4-(((1s,4s)-4-...)
Affinity DataIC50:  18nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274003(CHEMBL462514 | N-[5-(Benzoyl-propyl-amino)-1-(2-ca...)
Affinity DataIC50:  18nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50275615(3-cyano-N-(5-((cyclohexyl(methyl)amino)methyl)-1-(...)
Affinity DataIC50:  20nMAssay Description:Inhibition of ITK (unknown origin) by DELPHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196975(CHEMBL245783 | N2-(2,3-difluorobenzyl)-N4-((4-(ami...)
Affinity DataIC50:  22nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274747(CHEMBL457705 | N-(1-(3-amino-3-oxopropyl)-5-(N-met...)
Affinity DataIC50:  23nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274002(CHEMBL517901 | N-(1-(3-amino-3-oxopropyl)-5-(N-eth...)
Affinity DataIC50:  27nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196990(CHEMBL246184 | N2-(2,4-dichlorobenzyl)-N4-((4-(ami...)
Affinity DataIC50:  27nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274701(CHEMBL485201 | N-(1-(3-amino-3-oxopropyl)-2-(4-cya...)
Affinity DataIC50:  27nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50275654(4-cyano-N-(5-((cyclohexyl(methyl)amino)methyl)-1-(...)
Affinity DataIC50:  27nMAssay Description:Inhibition of ITK (unknown origin) by DELPHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196982(CHEMBL395691 | N2-(2-chlorobenzyl)-N4-(((1r,4r)-4-...)
Affinity DataIC50:  29nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50275653(CHEMBL487563 | N-(1-(3-(1H-imidazol-1-yl)propyl)-5...)
Affinity DataIC50:  30nMAssay Description:Inhibition of ITK (unknown origin) by DELPHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196980(CHEMBL247572 | N4-((4-(aminomethyl)cyclohexyl)meth...)
Affinity DataIC50:  31nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196948(CHEMBL428751 | N*4*-(4-aminomethyl-cyclohexylmethy...)
Affinity DataIC50:  34nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50275556(4-cyano-N-(5-(((cyclopentylmethyl)(methyl)amino)me...)
Affinity DataIC50:  34nMAssay Description:Inhibition of ITK (unknown origin) by DELPHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196956(CHEMBL396370 | N2-(2,5-difluorobenzyl)-N4-((4-(ami...)
Affinity DataIC50:  35nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50274667(CHEMBL490269 | N-[1-(2-carbamoylethyl)-2-[(4-cyano...)
Affinity DataIC50:  35nMAssay Description:Inhibition of recombinant ITK (unknown origin) by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Johnson & Johnson

Curated by ChEMBL
LigandPNGBDBM50275618(CHEMBL488170 | N-(5-((cyclohexyl(methyl)amino)meth...)
Affinity DataIC50:  36nMAssay Description:Inhibition of ITK (unknown origin) by DELPHIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196973(CHEMBL438669 | N*4*-(4-aminomethyl-cyclohexylmethy...)
Affinity DataIC50:  39nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50196954(CHEMBL246177 | N*4*-(4-aminomethyl-cyclohexylmethy...)
Affinity DataIC50:  39nMAssay Description:Inhibition of PKCtheta by FP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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