Affinity DataKi: 1.10nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D3 in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D3 in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D3 in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D3 in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D3 in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D3 in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D2L in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 8.80nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D2L in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D3 in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 27nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D2L in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D3 in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D3 in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 68nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D2L in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 114nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D2L in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 213nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D2L in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 245nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D2L in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 354nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D2L in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 622nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D2L in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 756nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D3 in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 782nMAssay Description:Tested for the binding constant against cloned human Dopamine receptor D2L in HEK cells by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 0.960nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 2.96nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 3.67nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 4.10nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 4.5nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 8.23nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 9.37nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 10.1nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 10.6nMAssay Description:Inhibition of binding of 3[H] WIN-35 428 to Dopamine transporter (DAT) of rat striatum.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 10.6nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 11.6nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 14.3nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 17.2nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 19.6nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 19.7nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 23.4nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 26.6nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 26.9nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 32.1nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 34.4nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 63.1nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 65.1nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 65.3nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:In vitro binding affinity at dopamine transporter in rat striatum by [3H]WIN-35428 displacement.More data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 113nMAssay Description:Inhibition of 3[H] WIN-35 428 binding to Dopamine transporter (DAT)More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 132nMAssay Description:In vitro binding affinity at serotonin transporter in rat striatum by [3H]- citalopram displacement.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 132nMAssay Description:Inhibition of binding of [3H]- citalopram to Serotonin transporter (SERT) of rat cerebral cortex.More data for this Ligand-Target Pair
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Wayne State University
Curated by ChEMBL
Wayne State University
Curated by ChEMBL
Affinity DataIC50: 137nMAssay Description:In vitro binding affinity at serotonin transporter in rat striatum by [3H]- citalopram displacement.More data for this Ligand-Target Pair