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Found 86 with Last Name = 'fejzo' and Initial = 'j'
TargetEstrogen receptor beta(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50154137(3-(6-HYDROXY-NAPHTHALEN-2-YL)-BENZO[D]ISOOXAZOL-6-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of estrogen receptor betaMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50154078(7-Bromo-2-(4-hydroxy-2-methyl-phenyl)-benzooxazol-...)
Affinity DataIC50:  1nMAssay Description:Inhibition of estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314628((E)-N-Hydroxy-3-{4-[3-(2-methyl-1H-indol-3-yl)pyrr...)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314637((E)-3-{4-[3-(2-tert-Butyl-1H-indol-3-yl)piperidin-...)
Affinity DataIC50:  3nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314630((E)-N-Hydroxy-3-(4-{1-[2-(2-methyl-1H-indol-3-yl)e...)
Affinity DataIC50:  3nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50154062(2-(5-HYDROXY-NAPHTHALEN-1-YL)-1,3-BENZOOXAZOL-6-OL...)
Affinity DataIC50:  5nMAssay Description:Inhibition of estrogen receptor betaMore data for this Ligand-Target Pair
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314627((E)-N-Hydroxy-3-{4-[3-(2-methyl-1H-indol-3-yl)pipe...)
Affinity DataIC50:  5nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314642((E)-3-{4-[(R)-3-(2-tert-Butyl-1H-indol-3-yl)piperi...)
Affinity DataIC50:  7.5nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314642((E)-3-{4-[(R)-3-(2-tert-Butyl-1H-indol-3-yl)piperi...)
Affinity DataIC50:  9nMAssay Description:Inhibition of FLAG-tagged HDAC3 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM19428((2E)-N-hydroxy-3-(4-{[(2-hydroxyethyl)[2-(1H-indol...)
Affinity DataIC50:  9nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314640((E)-3-{4-[3-(2-tert-Butyl-1H-indol-3-yl)piperidin-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314635((E)-N-Hydroxy-3-{4-[3-(1H-indol-3-yl)piperidin-1-y...)
Affinity DataIC50:  11nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314636((E)-N-Hydroxy-3-{4-[3-(2-phenyl-1H-indol-3-yl)pipe...)
Affinity DataIC50:  11nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314633(CHEMBL1093362 | N-hydroxy-3-(2-(2-(2-methyl-1H-ind...)
Affinity DataIC50:  13nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314643((E)-3-{4-[(S)-3-(2-tert-Butyl-1H-indol-3-yl)piperi...)
Affinity DataIC50:  15nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314639((E)-3-{3-Fluoro-4-[3-(2-phenyl-1H-indol-3-yl)piper...)
Affinity DataIC50:  16nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314641((E)-3-{4-[3-(2-tert-Butyl-1H-indol-3-yl)piperidin-...)
Affinity DataIC50:  19nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314643((E)-3-{4-[(S)-3-(2-tert-Butyl-1H-indol-3-yl)piperi...)
Affinity DataIC50:  21nMAssay Description:Inhibition of FLAG-tagged HDAC3 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314629((E)-N-Hydroxy-3-{4-[2-(2-methyl-1H-indol-3-ylmethy...)
Affinity DataIC50:  24nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314631(CHEMBL1088949 | N-hydroxy-3-(2-(2-(2-methyl-1H-ind...)
Affinity DataIC50:  27nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314642((E)-3-{4-[(R)-3-(2-tert-Butyl-1H-indol-3-yl)piperi...)
Affinity DataIC50:  28nMAssay Description:Inhibition of HDAC4 expressed in baculovirus system by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314642((E)-3-{4-[(R)-3-(2-tert-Butyl-1H-indol-3-yl)piperi...)
Affinity DataIC50:  31nMAssay Description:Inhibition of HDAC2 expressed in baculovirus system by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314643((E)-3-{4-[(S)-3-(2-tert-Butyl-1H-indol-3-yl)piperi...)
Affinity DataIC50:  38nMAssay Description:Inhibition of HDAC4 expressed in baculovirus system by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314632(CHEMBL1089701 | N-hydroxy-3-(2-(2-(2-methyl-1H-ind...)
Affinity DataIC50:  41nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314643((E)-3-{4-[(S)-3-(2-tert-Butyl-1H-indol-3-yl)piperi...)
Affinity DataIC50:  48nMAssay Description:Inhibition of HDAC2 expressed in baculovirus system by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50148169((4-Chloro-phenyl)-[4-(4-methoxy-pyridin-2-ylamino)...)
Affinity DataIC50:  53nMAssay Description:Inhibition of iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50124525(4'-amino-5'-fluorospiro[hexahydropyridine-4,2'-(1'...)
Affinity DataIC50:  67nMAssay Description:Inhibition of iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50035206(4-(5-Methoxy-1a,2,3,7b-tetrahydro-1H-cyclopropa[a]...)
Affinity DataIC50:  69nMAssay Description:Inhibition of aromataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314634(CHEMBL1089301 | N-hydroxy-3-(3-(2-(2-methyl-1H-ind...)
Affinity DataIC50:  76nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM19956(3-arylquinazolinethione, 1bd | 7-hydroxy-3-(4-hydr...)
Affinity DataIC50:  79nMAssay Description:Inhibition of estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50148164(4-(4-Methoxy-pyridin-2-ylamino)-piperidine-1-carbo...)
Affinity DataIC50:  89nMAssay Description:Inhibition of iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM10009(1-[(6-Methoxybenzofuran-2-yl)-p-tolylmethyl]-1H-1,...)
Affinity DataIC50:  100nMAssay Description:Inhibition of aromataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314643((E)-3-{4-[(S)-3-(2-tert-Butyl-1H-indol-3-yl)piperi...)
Affinity DataIC50:  110nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314642((E)-3-{4-[(R)-3-(2-tert-Butyl-1H-indol-3-yl)piperi...)
Affinity DataIC50:  118nMAssay Description:Inhibition of FLAG-tagged HDAC6 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314638((E)-3-{3-Fluoro-4-[3-(1H-indol-3-yl)piperidin-1-yl...)
Affinity DataIC50:  136nMAssay Description:Inhibition of FLAG-tagged HDAC1 expressed in HEK293 cells by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM10002((6-Methoxybenzofuran-2-yl)-(4-methoxyphenyl)-3-pyr...)
Affinity DataIC50:  160nMAssay Description:Inhibition of aromataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314642((E)-3-{4-[(R)-3-(2-tert-Butyl-1H-indol-3-yl)piperi...)
Affinity DataIC50:  217nMAssay Description:Inhibition of HDAC8 expressed in baculovirus system by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM9471(4-(1H-Imidazol-1-ylmethyl)-7-methoxy-2H-chromen-2-...)
Affinity DataIC50:  280nMAssay Description:Inhibition of aromataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50124528(CHEMBL170176 | ethyl 4'-amino-1H,1'H-spiro[piperid...)
Affinity DataIC50:  300nMAssay Description:Inhibition of iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50314643((E)-3-{4-[(S)-3-(2-tert-Butyl-1H-indol-3-yl)piperi...)
Affinity DataIC50:  364nMAssay Description:Inhibition of HDAC8 expressed in baculovirus system by fluorescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50376217(CHEMBL362476)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50091813(4-Ethyl-pyridin-2-ylamine | 4-ethylpyridin-2-amine...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50237936(4-Ethyl-5,6-dihydro-1H-pyridin-(2Z)-ylideneamine |...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50376215(CHEMBL409050)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50376221(CHEMBL261781)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNitric oxide synthase, inducible(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50117550((3aR,9bS)-7-methoxy-2,3,3a,9b-tetrahydro-1H-cyclop...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of iNOSMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM10025(5-(1H-imidazol-1-ylmethyl)-7,8-dihydroquinoline | ...)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of aromataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50376223(CHEMBL438549)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of aromataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50376225(CHEMBL258553)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50168378(2-methyl-6-o-tolylnaphthalene | 6-(2-Hydroxy-pheny...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of estrogen receptor betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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