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Found 33 with Last Name = 'fenical' and Initial = 'w'
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347488(CHEMBL1802205)
Affinity DataIC50:  160nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347486(CHEMBL1802199)
Affinity DataIC50:  186nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347476(CHEMBL1802264)
Affinity DataIC50:  320nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347471(CHEMBL1802260)
Affinity DataIC50:  450nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347482(CHEMBL1802271)
Affinity DataIC50:  480nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347468(CHEMBL1802203)
Affinity DataIC50:  690nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347469(CHEMBL1802258)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347484(CHEMBL1802277)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347472(CHEMBL1802261)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347483(CHEMBL1802272)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347481(CHEMBL1802270)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347479(CHEMBL1802267)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrnithine decarboxylase(Homo sapiens (Human))
University Of California - San Diego

Curated by ChEMBL
LigandPNGBDBM50476063(SALINIKETAL A)
Affinity DataIC50:  5.05E+3nMAssay Description:Inhibition of TPA-induced ornithine decarboxylase expressed in T24 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347478(CHEMBL1802266)
Affinity DataIC50:  1.05E+4nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347489(CHEMBL1802273)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347480(CHEMBL1802269)
Affinity DataIC50:  1.13E+4nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50316814(CHEMBL1097104 | cryptosphaerolide)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of Mcl1 protein by Mcl1/Bak fluorescence resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM81111(1-methoxy-7,8-dimethyl-phenazine | 1-methoxy-7,8-d...)
Affinity DataIC50:  1.17E+4nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50316815((1R,3S,4R,8S,10R,11S,14R)-4-methoxy-10,11-dimethyl...)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of Mcl1 protein by Mcl1/Bak fluorescence resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347470(CHEMBL1802259)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347474(CHEMBL1420181)
Affinity DataIC50:  1.53E+4nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347475(CHEMBL1802263)
Affinity DataIC50:  1.82E+4nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347487(CHEMBL1802200)
Affinity DataIC50:  1.85E+4nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrnithine decarboxylase(Homo sapiens (Human))
University Of California - San Diego

Curated by ChEMBL
LigandPNGBDBM50476064(SALINIKETAL B)
Affinity DataIC50:  1.89E+4nMAssay Description:Inhibition of TPA-induced ornithine decarboxylase expressed in T24 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347467(CHEMBL1802202)
Affinity DataIC50:  2.69E+4nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347485(CHEMBL1802197)
Affinity DataIC50:  3.11E+4nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347477(CHEMBL1802265)
Affinity DataIC50:  3.55E+4nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347466(CHEMBL1802201)
Affinity DataIC50:  3.68E+4nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Ewha Womans University

Curated by ChEMBL
LigandPNGBDBM50042944((E)-1-(2,4-Dihydroxy-phenyl)-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50:  5.15E+4nMAssay Description:Ability to displace [3H]quipazine binding to 5-hydroxytryptamine 3 receptor sites in NG 108-15.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosyldihydronicotinamide dehydrogenase [quinone](Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50347473(CHEMBL1802262)
Affinity DataIC50:  6.08E+4nMAssay Description:Inhibition of human QR2 expressed in Escherichia coli BL21 (DE3) using MTT and NMeH as substrate assessed as formazan formationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxiredoxin-1(Homo sapiens)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50411905(CHEMBL272733)
Affinity DataKd:  2.61E+3nMAssay Description:Binding affinity to full-length human PRDX1 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxiredoxin-1(Homo sapiens)
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50504090(CHEMBL4092369)
Affinity DataKd:  1.83E+3nMAssay Description:Binding affinity to full-length human PRDX1 by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholine receptor subunit alpha/beta/delta/gamma(Torpedo californica)
University Of California San Diego

Curated by ChEMBL
LigandPNGBDBM50000690(10,25-dimethoxy-15,15,30-trimethyl-(1S,16R)-7,23-d...)
Affinity DataEC50:  3.20E+6nMAssay Description:In vitro ability of the compound to inhibit the binding of [125I]-alpha-bungarotoxin to nicotinic acetylcholine receptor on membranes prepared from t...More data for this Ligand-Target Pair