Compile Data Set for Download or QSAR
maximum 50k data
Found 111 with Last Name = 'fenton' and Initial = 'rj'
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50165355((2R,4S)-3-(acetylamino)-4-{[(E)-amino(imino)methyl...)
Affinity DataIC50:  0.770nMAssay Description:Inhibitory concentration against neuraminidase of influenza A/Mem/Bel/71 (H3N1) virus starin; (n=5)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4942((2R,3R,4S)-4-carbamimidamido-2-(diethylcarbamoyl)-...)
Affinity DataIC50:  1nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4972((2R,3R,4S)-4-amino-3-acetamido-2-{[2-(3-phenylphen...)
Affinity DataIC50:  2nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4945((2R,3R,4S)-4-amino-3-acetamido-2-[(2-phenylethyl)(...)
Affinity DataIC50:  2nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4940((2R,3R,4S)-4-carbamimidamido-2-(dipropylcarbamoyl)...)
Affinity DataIC50:  2nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4967((2R,3R,4S)-4-amino-3-acetamido-2-{[2-(4-phenylphen...)
Affinity DataIC50:  2nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50165355((2R,4S)-3-(acetylamino)-4-{[(E)-amino(imino)methyl...)
Affinity DataIC50:  2.48nMAssay Description:Inhibitory concentration against neuraminidase of influenza A/PR/8/34 (H1N1) virus starin; (n=5)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4937((2R,3R,4S)-4-amino-2-(diethylcarbamoyl)-3-acetamid...)
Affinity DataIC50:  3nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4966((2R,3R,4S)-4-amino-3-acetamido-2-{[2-(3-hydroxyphe...)
Affinity DataIC50:  3nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4941((2R,3R,4S)-4-amino-3-acetamido-2-[ethyl(propyl)car...)
Affinity DataIC50:  3nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50165355((2R,4S)-3-(acetylamino)-4-{[(E)-amino(imino)methyl...)
Affinity DataIC50:  3.25nMAssay Description:Inhibitory concentration against neuraminidase of influenza A/Chicken/Vietnam/8/2004(H5N1) virus starin; (n=5)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza B virus)
Glaxo Wellcome Research And Development

LigandPNGBDBM4934((2R,3R,4S)-4-carbamimidamido-3-acetamido-2-[(1R,2R...)
Affinity DataIC50:  4nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4933((2R,3R,4S)-4-carbamimidamido-3-acetamido-2-[methyl...)
Affinity DataIC50:  4nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4943((2R,3R,4S)-4-amino-2-[butyl(propyl)carbamoyl]-3-ac...)
Affinity DataIC50:  4nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4946((2R,3R,4S)-4-carbamimidamido-3-acetamido-2-[(2-phe...)
Affinity DataIC50:  5nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4952((2R,3R,4S)-4-amino-3-acetamido-2-[ethyl(2-phenylet...)
Affinity DataIC50:  5nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4965((2R,3R,4S)-4-amino-3-acetamido-2-{[2-(3-methoxyphe...)
Affinity DataIC50:  5nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4934((2R,3R,4S)-4-carbamimidamido-3-acetamido-2-[(1R,2R...)
Affinity DataIC50:  5nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4935((2R,3R,4S)-4-amino-2-[(2,5-dimethylpyrrolidin-1-yl...)
Affinity DataIC50:  6nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4968((2R,3R,4S)-4-amino-2-{[2-(2,4-dichlorophenyl)ethyl...)
Affinity DataIC50:  6nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4949((2R,3R,4S)-4-carbamimidamido-3-acetamido-2-[nonyl(...)
Affinity DataIC50:  7nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50165356((2R,4S)-4-carbamimidamido-2-[(1R)-1-({[12-({[(1R)-...)
Affinity DataIC50:  7.86nMAssay Description:Inhibitory concentration against neuraminidase of influenza A/Mem/Bel/71 (H3N1) virus starin; (n=5)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4963((2R,3R,4S)-4-amino-3-acetamido-2-{[2-(4-methoxyphe...)
Affinity DataIC50:  8nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4959((2R,3R,4S)-4-amino-3-acetamido-2-[(2-phenylethyl)(...)
Affinity DataIC50:  8nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4956((2R,3R,4S)-4-amino-2-[(2-azidoethyl)(2-phenylethyl...)
Affinity DataIC50:  9nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4971((2R,3R,4S)-4-amino-3-acetamido-2-{[2-(2-methoxyphe...)
Affinity DataIC50:  9nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4964((2R,3R,4S)-4-amino-3-acetamido-2-{[2-(4-hydroxyphe...)
Affinity DataIC50:  9nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4957((2R,3R,4S)-4-amino-3-acetamido-2-[(2-hydroxyethyl)...)
Affinity DataIC50:  12nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4929((2R,3R,4S)-4-amino-2-(dipropylcarbamoyl)-3-acetami...)
Affinity DataIC50:  12nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4969((2R,3R,4S)-4-amino-3-acetamido-2-({2-[4-(propan-2-...)
Affinity DataIC50:  12nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4958((2R,3R,4S)-4-amino-3-acetamido-2-[(2-methylpropyl)...)
Affinity DataIC50:  14nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4947((2R,3R,4S)-4-amino-3-acetamido-2-[(3-phenylpropyl)...)
Affinity DataIC50:  18nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50165356((2R,4S)-4-carbamimidamido-2-[(1R)-1-({[12-({[(1R)-...)
Affinity DataIC50:  21.7nMAssay Description:Inhibitory concentration against neuraminidase of influenza A/PR/8/34 (H1N1) virus starin; (n=5)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4948((2R,3R,4S)-4-amino-3-acetamido-2-[nonyl(propyl)car...)
Affinity DataIC50:  23nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4932((2R,3R,4S)-4-carbamimidamido-2-(dimethylcarbamoyl)...)
Affinity DataIC50:  25nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4938((2R,3R,4S)-4-amino-2-[bis(prop-2-en-1-yl)carbamoyl...)
Affinity DataIC50:  40nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4961((2R,3R,4S)-4-amino-2-[cyclopropyl(2-phenylethyl)ca...)
Affinity DataIC50:  46nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Puerto Rico/8/34/Mount Sinai(...)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50165356((2R,4S)-4-carbamimidamido-2-[(1R)-1-({[12-({[(1R)-...)
Affinity DataIC50:  61nMAssay Description:Inhibitory concentration against neuraminidase of influenza A/Chicken/Vietnam/8/2004(H5N1) virus starin; (n=5)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4976((2R,3R,4S)-4-amino-2-{[(2R,5R)-2,5-dimethylpyrroli...)
Affinity DataIC50:  110nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4977((2R,3R,4S)-4-amino-2-{[(2S,5S)-2,5-dimethylpyrroli...)
Affinity DataIC50:  110nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4928((2R,3R,4S)-4-amino-3-acetamido-2-[methyl(propyl)ca...)
Affinity DataIC50:  180nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4970((2R,3R,4S)-4-amino-2-{[2-(4-benzylphenyl)ethyl](pr...)
Affinity DataIC50:  270nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4978((2R,3R,4S)-4-amino-2-{[(2R,5S)-2,5-diethylpyrrolid...)
Affinity DataIC50:  290nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4974((2R,3R,4S)-4-amino-3-acetamido-2-[(2-methylpyrroli...)
Affinity DataIC50:  310nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4951((2R,3R,4S)-4-amino-3-acetamido-2-[methyl(2-phenyle...)
Affinity DataIC50:  320nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza B virus)
Glaxo Wellcome Research And Development

LigandPNGBDBM4937((2R,3R,4S)-4-amino-2-(diethylcarbamoyl)-3-acetamid...)
Affinity DataIC50:  360nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza B virus)
Glaxo Wellcome Research And Development

LigandPNGBDBM4941((2R,3R,4S)-4-amino-3-acetamido-2-[ethyl(propyl)car...)
Affinity DataIC50:  410nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4936((2R,3R,4S)-4-amino-2-(dibutylcarbamoyl)-3-acetamid...)
Affinity DataIC50:  450nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza B virus)
Glaxo Wellcome Research And Development

LigandPNGBDBM4942((2R,3R,4S)-4-carbamimidamido-2-(diethylcarbamoyl)-...)
Affinity DataIC50:  490nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuraminidase(Influenza A virus (A/Singapore/1/57(H2N2)))
Glaxo Wellcome Research And Development

LigandPNGBDBM4931((2R,3R,4S)-4-carbamimidamido-3-acetamido-2-(propyl...)
Affinity DataIC50:  500nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 111 total ) | Next | Last >>
Jump to: