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Found 5061 with Last Name = 'fernandes' and Initial = 's'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321606((3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazo...)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321606((3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazo...)
Affinity DataKi:  0.130nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321607((3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazo...)
Affinity DataKi:  0.690nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Universidade Federal De S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50121205(CHEBI:18295 | Histamine)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]-Histamine from human histamine 4 receptor transfected in HEK293T cells incubated for 16 hrs by liquid scintillation counter anal...More data for this Ligand-Target Pair
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321604((3S,6S,9S,12S,15R,18S,21S,24R,27S)-18-((1H-imidazo...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK1 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321604((3S,6S,9S,12S,15R,18S,21S,24R,27S)-18-((1H-imidazo...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK1 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universidade Federal De S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50121205(CHEBI:18295 | Histamine)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]-Histamine from human histamine 3 receptor transfected in HEK293T cells incubated for 16 hrs by liquid scintillation counter anal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM21123((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM21123((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321605((6R,9S,12S,15R,18S,21S,24S,27S)-12-((1H-imidazol-5...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universidade Federal De S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50552436(CHEMBL4749654)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-Histamine from human histamine 3 receptor transfected in HEK293T cells incubated for 16 hrs by liquid scintillation counter anal...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321605((6R,9S,12S,15R,18S,21S,24S,27S)-12-((1H-imidazol-5...)
Affinity DataKi:  4.90nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321598((S)-3-((4R,7S,10S,13R,16S,22S)-16-((1H-imidazol-5-...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321608((3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazo...)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universidade Federal De S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50552434(CHEMBL4747180)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]-Histamine from human histamine 3 receptor transfected in HEK293T cells incubated for 16 hrs by liquid scintillation counter anal...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321601((2S,5R,11S,18S,21S)-2-amino-21-((S)-1-amino-1-oxo-...)
Affinity DataKi:  7.40nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321599((S)-3-((4R,7S,10S,13R,16S,22S)-16-((1H-imidazol-5-...)
Affinity DataKi:  8.60nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321607((3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazo...)
Affinity DataKi:  9nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK1 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321607((3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazo...)
Affinity DataKi:  9nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK1 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321608((3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazo...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321608((3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazo...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321596((3S,6R,9S,12S,15S,18S)-3-((1H-imidazol-5-yl)methyl...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK1 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321596((3S,6R,9S,12S,15S,18S)-3-((1H-imidazol-5-yl)methyl...)
Affinity DataKi:  15nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK1 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universidade Federal De S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50552435(CHEMBL4756432)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]-Histamine from human histamine 3 receptor transfected in HEK293T cells incubated for 16 hrs by liquid scintillation counter anal...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
S£O Paulo State University

Curated by ChEMBL
LigandPNGBDBM50516759(CHEMBL4458610)
Affinity DataKi:  17nMAssay Description:Inhibition of human chymotrypsin-like activity of 20S proteasome (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321608((3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazo...)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK2 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321606((3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazo...)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK1 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321597((3S,6R,9S,12S,15S,18S)-3-((1H-imidazol-5-yl)methyl...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321606((3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazo...)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK1 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321608((3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazo...)
Affinity DataKi:  18nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK2 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321597((3S,6R,9S,12S,15S,18S)-3-((1H-imidazol-5-yl)methyl...)
Affinity DataKi:  32nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK1 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universidade Federal De S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50552430(CHEMBL4798369)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-Histamine from human histamine 3 receptor transfected in HEK293T cells incubated for 16 hrs by liquid scintillation counter anal...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-lactamase TEM(Escherichia coli)
S£O Paulo State University

Curated by ChEMBL
LigandPNGBDBM50516761(CHEMBL3286879)
Affinity DataKi:  40nMAssay Description:Inhibition of bacterial beta lactamase TEM-1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321604((3S,6S,9S,12S,15R,18S,21S,24R,27S)-18-((1H-imidazo...)
Affinity DataKi:  42nMAssay Description:Displacement of [3H]DPDPE from human delta opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321596((3S,6R,9S,12S,15S,18S)-3-((1H-imidazol-5-yl)methyl...)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]DAMGO from rat mu opioid receptor expressed in mouse HN9.10 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321609((S)-4-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)...)
Affinity DataKi:  61nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK2 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321609((S)-4-((S)-1-amino-1-oxo-3-phenylpropan-2-ylamino)...)
Affinity DataKi:  61nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK2 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Universidade Federal De S£O Paulo

Curated by ChEMBL
LigandPNGBDBM50552439(CHEMBL4568949)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]-Histamine from human histamine 4 receptor transfected in HEK293T cells incubated for 16 hrs by liquid scintillation counter anal...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321597((3S,6R,9S,12S,15S,18S)-3-((1H-imidazol-5-yl)methyl...)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK2 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321606((3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazo...)
Affinity DataKi:  110nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK2 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321606((3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazo...)
Affinity DataKi:  110nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK2 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321607((3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazo...)
Affinity DataKi:  120nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK2 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321607((3S,6S,9S,12S,15R,18S,21S,27R,30S)-18-((1H-imidazo...)
Affinity DataKi:  120nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK2 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321602((3S,6S,9S,12S,15R,18S)-18-((1H-imidazol-5-yl)methy...)
Affinity DataKi:  160nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK2 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321605((6R,9S,12S,15R,18S,21S,24S,27S)-12-((1H-imidazol-5...)
Affinity DataKi:  180nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK2 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321605((6R,9S,12S,15R,18S,21S,24S,27S)-12-((1H-imidazol-5...)
Affinity DataKi:  180nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK2 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321604((3S,6S,9S,12S,15R,18S,21S,24R,27S)-18-((1H-imidazo...)
Affinity DataKi:  190nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK2 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321604((3S,6S,9S,12S,15R,18S,21S,24R,27S)-18-((1H-imidazo...)
Affinity DataKi:  190nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK2 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321596((3S,6R,9S,12S,15S,18S)-3-((1H-imidazol-5-yl)methyl...)
Affinity DataKi:  200nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK2 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50321596((3S,6R,9S,12S,15S,18S)-3-((1H-imidazol-5-yl)methyl...)
Affinity DataKi:  200nMAssay Description:Displacement of [125I]CCK-8(SO3) from human CCK2 receptor expressed in human HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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