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Found 32 with Last Name = 'folmer' and Initial = 'bj'
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233026(CHEMBL403138 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233007(CHEMBL403139 | N-((1S,13bR)-6-chloro-1,2,3,4,9,13b...)
Affinity DataIC50:  26nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233014((rac)-N-(6-chloro-1,3,4,13b-tetrahydro-2H-9-oxa-4a...)
Affinity DataIC50:  43nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233013(CHEMBL253944 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataIC50:  133nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233009(CHEMBL253734 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataIC50:  193nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233028(1-((1S,13bR)-6-chloro-1,3,4,13b-tetrahydro-2H-9-ox...)
Affinity DataIC50:  314nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233020(CHEMBL252451 | N-((1S,13bR)-6,7-dichloro-1,3,4,13b...)
Affinity DataIC50:  318nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233022(2,2,2-trifluoro-N-((1S,13bR)-6-fluoro-1,3,4,13b-te...)
Affinity DataIC50:  730nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233015(CHEMBL252646 | N-((1S,13bR)-7-chloro-1,3,4,13b-tet...)
Affinity DataIC50:  2.22E+3nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233014((rac)-N-(6-chloro-1,3,4,13b-tetrahydro-2H-9-oxa-4a...)
Affinity DataEC50:  10.6nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233017(CHEMBL252850 | N-((1S,13bR)-5-acetyl-1,3,4,13b-tet...)
Affinity DataEC50:  0.960nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233016(CHEMBL253735 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233018(CHEMBL401627 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataEC50:  450nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233013(CHEMBL253944 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataEC50:  10.3nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233027(2,2,2-trifluoro-N-(1S,13bR)-1,3,4,13b-tetrahydro-2...)
Affinity DataEC50:  222nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233019(CHEMBL402526 | N-((1S,13bR)-5-chloro-1,3,4,13b-tet...)
Affinity DataEC50:  19nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233021(CHEMBL252648 | N-((1S,13bR)-6-acetyl-1,3,4,13b-tet...)
Affinity DataEC50:  258nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233023(CHEMBL404432 | N-((1S,13bR)-6-chloro-9-methyl-1,2,...)
Affinity DataEC50:  9.80nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233025(CHEMBL404433 | N-((1S,13bR)-5,6-dichloro-1,3,4,13b...)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233022(2,2,2-trifluoro-N-((1S,13bR)-6-fluoro-1,3,4,13b-te...)
Affinity DataEC50:  198nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233009(CHEMBL253734 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataEC50:  4.45E+3nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233024((1S,13bR)-6-chloro-1,3,4,13b-tetrahydro-2H-9-oxa-4...)
Affinity DataEC50:  513nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233020(CHEMBL252451 | N-((1S,13bR)-6,7-dichloro-1,3,4,13b...)
Affinity DataEC50:  38nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233015(CHEMBL252646 | N-((1S,13bR)-7-chloro-1,3,4,13b-tet...)
Affinity DataEC50:  993nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233008(2,2,2-trifluoro-N-((1S,13bR)-5-vinyl-1,3,4,13b-tet...)
Affinity DataEC50:  0.810nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233007(CHEMBL403139 | N-((1S,13bR)-6-chloro-1,2,3,4,9,13b...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233006(((1S,13bR)-6-chloro-1,3,4,13b-tetrahydro-2H-9-oxa-...)
Affinity DataEC50:  598nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233026(CHEMBL403138 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataEC50:  3nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233029(2,2,2-trifluoro-N-((1S,13bR)-6-vinyl-1,3,4,13b-tet...)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233010(CHEMBL252253 | N-((1R,13bS)-6-chloro-1,3,4,13b-tet...)
Affinity DataEC50:  54nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233011(((1S,13bR)-6-chloro-1,3,4,13b-tetrahydro-2H-9-oxa-...)
Affinity DataEC50:  1.34E+3nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233012(CHEMBL252449 | N-((1S,13bR)-6-chloro-1,3,4,13b-tet...)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed