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Found 8 with Last Name = 'fortin' and Initial = 's'
TargetCytochrome P450 1A1(Homo sapiens (Human))
H�Pital Saint-Fran�Ois D'Assise

Curated by ChEMBL
LigandPNGBDBM50239593(CHEMBL4096550)
Affinity DataKi:  240nMAssay Description:Inhibition of human supersomes CYP1A1-mediated 7-ethoxyresorufin conversion to fluorescent resorufin preincubated with 7-ethoxyresorufin for 5 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Homo sapiens (Human))
H�Pital Saint-Fran�Ois D'Assise

Curated by ChEMBL
LigandPNGBDBM50585332(CHEMBL5077719)
Affinity DataKi:  300nMAssay Description:Binding affinity to recombinant CYP1A1 in human liver microsomes assessed as inhibition constant measured for 15 mins in the presence of NADPH regene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Homo sapiens (Human))
H�Pital Saint-Fran�Ois D'Assise

Curated by ChEMBL
LigandPNGBDBM50239591(CHEMBL4104764)
Affinity DataKi:  490nMAssay Description:Inhibition of human supersomes CYP1A1-mediated 7-ethoxyresorufin conversion to fluorescent resorufin preincubated with 7-ethoxyresorufin for 5 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Homo sapiens (Human))
H�Pital Saint-Fran�Ois D'Assise

Curated by ChEMBL
LigandPNGBDBM50585331(CHEMBL5073496)
Affinity DataKi:  500nMAssay Description:Binding affinity to recombinant CYP1A1 in human liver microsomes assessed as inhibition constant measured for 15 mins in the presence of NADPH regene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Homo sapiens (Human))
H�Pital Saint-Fran�Ois D'Assise

Curated by ChEMBL
LigandPNGBDBM50239592(CHEMBL4078072)
Affinity DataKi:  540nMAssay Description:Inhibition of human supersomes CYP1A1-mediated 7-ethoxyresorufin conversion to fluorescent resorufin preincubated with 7-ethoxyresorufin for 5 mins f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A1(Homo sapiens (Human))
H�Pital Saint-Fran�Ois D'Assise

Curated by ChEMBL
LigandPNGBDBM50585333(CHEMBL5084275)
Affinity DataKi:  1.70E+3nMAssay Description:Binding affinity to recombinant CYP1A1 in human liver microsomes assessed as inhibition constant measured for 15 mins in the presence of NADPH regene...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM15339(6-fluoro-2-[4-(2-fluorophenyl)phenyl]-3-methyl-qui...)
Affinity DataIC50:  12nMAssay Description:Inhibition of recombinant N-terminal His-tagged human DHODH (31 to 395 residues) expressed in Escherichia coli using L-DHO as substrate measured ever...More data for this Ligand-Target Pair
TargetDihydroorotate dehydrogenase (quinone), mitochondrial(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50559136(CHEMBL2165736)
Affinity DataIC50:  72nMAssay Description:Inhibition of recombinant N-terminal His-tagged human DHODH (31 to 395 residues) expressed in Escherichia coli using L-DHO as substrate measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed