TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 0.130nMAssay Description:Displacement of [3H]prazosin from rat salivary gland adrenergic alpha 1A receptor after 45 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Rattus norvegicus (Rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Displacement of [3H]prazosin from rat salivary gland adrenergic alpha 1A receptor after 45 mins by liquid scintillation counterMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidade Federal Do Rio Grande Do Sul
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]-8-OH-DPAT from 5HT1A receptor in Wistar rat hippocampus homogenateMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 0.420nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 0.490nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 0.550nMAssay Description:Displacement of [3H]prazosin from rat liver adrenergic alpha1B receptor after 45 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 0.619nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 0.650nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 0.690nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 0.690nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 0.729nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul
Curated by ChEMBL
Affinity DataKi: 2.20nMAssay Description:Agonist activity at dopamine D2 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 2.90nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul
Curated by ChEMBL
Affinity DataKi: 3.60nMAssay Description:Antagonist activity at dopamine D4 receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 4.51nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
TargetAlpha-1B adrenergic receptor(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 5.55nMAssay Description:Displacement of [3H]prazosin from rat liver adrenergic alpha1B receptor after 45 mins by liquid scintillation counterMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 5.60nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 6.10nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 6.61nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 6.90nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidade Federal Do Rio Grande Do Sul
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul
Curated by ChEMBL
Affinity DataKi: 7nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in Wistar rat cortex homogenateMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 7.01nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 7.19nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 7.19nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 8.02nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 8.41nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 8.41nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 9.02nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universidade Federal Do Rio Grande Do Sul
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Agonist activity at 5HT1A receptorMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 9.51nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 9.59nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 10.4nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 10.5nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 10.7nMAssay Description:Displacement of [3H]CP-55940 from CB1 receptor in rat brain by filtration assayMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Universidade Federal Do Rio De Janeiro
Curated by ChEMBL
Affinity DataKi: 11.0nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptor by filtration assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universidade Federal Do Rio Grande Do Sul
Curated by ChEMBL
Universidade Federal Do Rio Grande Do Sul
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]ketanserin from 5HT2A receptor in rat cortex membraneMore data for this Ligand-Target Pair