Affinity DataIC50: 0.200nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.290nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.290nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated guinea pig brain membranesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(RAT)
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated guinea pig brain membranesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 2.30nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(RAT)
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 5nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(RAT)
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
Affinity DataIC50: 14nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(RAT)
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 20nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(RAT)
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 30nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(RAT)
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(RAT)
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 32nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated guinea pig brain membranesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(RAT)
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 53nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 57nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Tested in vitro for amylase release from rat pancreatic acini (% of amylase secretion at 1 mM)More data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(RAT)
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 70nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 72nMAssay Description:In vitro binding affinity against Cholecystokinin type B receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Inhibition of [125I]-BH-CCK- binding to peripheral cholecystokinin type B receptor from rat pancreatic aciniMore data for this Ligand-Target Pair