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Found 21 with Last Name = 'garada' and Initial = 'b'
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50058293(3-(4-Fluoro-phenyl)-8-(3-phenyl-propyl)-8-aza-bicy...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of [3H]WIN35,428 binding to dopamine transporter using of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50058287(3-(4-Fluoro-phenyl)-8-(5-phenyl-pentyl)-8-aza-bicy...)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of [3H]WIN35,428 binding to dopamine transporter using of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50058286((1R,12R) | (1R,12S) | CHEMBL119561 | Diastereiosom...)
Affinity DataIC50:  7.38nMAssay Description:Inhibition of [3H]WIN35,428 binding to dopamine transporter using of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50058294((2R,3S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-(3-phe...)
Affinity DataIC50:  19.7nMAssay Description:Inhibition of [3H]- citalopram binding to serotonin transporter of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50058294((2R,3S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-(3-phe...)
Affinity DataIC50:  22nMAssay Description:Inhibition of [3H]WIN35,428 binding to dopamine transporter using of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50058292(CHEMBL118075 | O-1196 | O-863 | [N-[2-[(3'-N'-Prop...)
Affinity DataIC50:  37.2nMAssay Description:Inhibition of [3H]WIN35,428 binding to dopamine transporter using of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50058287(3-(4-Fluoro-phenyl)-8-(5-phenyl-pentyl)-8-aza-bicy...)
Affinity DataIC50:  49.9nMAssay Description:Inhibition of [3H]- citalopram binding to serotonin transporter of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50058295(8-Benzyl-3-(4-fluoro-phenyl)-8-aza-bicyclo[3.2.1]o...)
Affinity DataIC50:  58.9nMAssay Description:Inhibition of [3H]WIN35,428 binding to dopamine transporter using of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50058289((2R,3S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-(5-phe...)
Affinity DataIC50:  99nMAssay Description:Inhibition of [3H]WIN35,428 binding to dopamine transporter using of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50058286((1R,12R) | (1R,12S) | CHEMBL119561 | Diastereiosom...)
Affinity DataIC50:  124nMAssay Description:Inhibition of [3H]- citalopram binding to serotonin transporter of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50058293(3-(4-Fluoro-phenyl)-8-(3-phenyl-propyl)-8-aza-bicy...)
Affinity DataIC50:  133nMAssay Description:Inhibition of [3H]- citalopram binding to serotonin transporter of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50058290((2R,3S)-8-Benzyl-3-[bis-(4-fluoro-phenyl)-methoxy]...)
Affinity DataIC50:  223nMAssay Description:Inhibition of [3H]WIN35,428 binding to dopamine transporter using of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50058292(CHEMBL118075 | O-1196 | O-863 | [N-[2-[(3'-N'-Prop...)
Affinity DataIC50:  264nMAssay Description:Inhibition of [3H]- citalopram binding to serotonin transporter of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50279764(CHEMBL55730 | Diastereiosomer of[N-[2-[(3'-N'-Prop...)
Affinity DataIC50:  343nMAssay Description:Inhibition of [3H]WIN35,428 binding to dopamine transporter using of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50279764(CHEMBL55730 | Diastereiosomer of[N-[2-[(3'-N'-Prop...)
Affinity DataIC50:  343nMAssay Description:Inhibition of [3H]WIN35,428 binding to dopamine transporter using of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50058289((2R,3S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-(5-phe...)
Affinity DataIC50:  550nMAssay Description:Inhibition of [3H]- citalopram binding to serotonin transporter of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50058295(8-Benzyl-3-(4-fluoro-phenyl)-8-aza-bicyclo[3.2.1]o...)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of [3H]- citalopram binding to serotonin transporter of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Macaca fascicularis)
Organix

Curated by ChEMBL
LigandPNGBDBM50058286((1R,12R) | (1R,12S) | CHEMBL119561 | Diastereiosom...)
Affinity DataIC50:  2.96E+3nMAssay Description:Inhibition of [3H]WIN35,428 binding to dopamine transporter using of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50058290((2R,3S)-8-Benzyl-3-[bis-(4-fluoro-phenyl)-methoxy]...)
Affinity DataIC50:  4.97E+3nMAssay Description:Inhibition of [3H]- citalopram binding to serotonin transporter of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50058286((1R,12R) | (1R,12S) | CHEMBL119561 | Diastereiosom...)
Affinity DataIC50:  5.02E+3nMAssay Description:Inhibition of [3H]- citalopram binding to serotonin transporter of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Organix

Curated by ChEMBL
LigandPNGBDBM50279764(CHEMBL55730 | Diastereiosomer of[N-[2-[(3'-N'-Prop...)
Affinity DataIC50:  5.52E+4nMAssay Description:Inhibition of [3H]- citalopram binding to serotonin transporter of Cynomolgus monkey caudate-putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed