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Found 38 with Last Name = 'garlapati' and Initial = 'a'
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50278495(4-chloro-1-(4-(3-(piperidin-1-yl)propoxy)benzyl)pi...)
Affinity DataKi:  0.0680nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50278350(4-fluoro-1-(4-(3-(piperidin-1-yl)propoxy)benzyl)pi...)
Affinity DataKi:  0.0940nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50278449(4-bromo-1-(4-(3-(piperidin-1-yl)propoxy)benzyl)pip...)
Affinity DataKi:  0.200nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50278448(4,4-difluoro-1-(4-(3-(piperidin-1-yl)propoxy)benzy...)
Affinity DataKi:  0.240nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50278445(4-fluoro-1-(4-(3-(pyrrolidin-1-yl)propoxy)benzyl)p...)
Affinity DataKi:  0.260nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50278444((R)-1-(3-(4-((3-fluoropyrrolidin-1-yl)methyl)pheno...)
Affinity DataKi:  0.280nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50278400((S)-1-(3-(4-((3-fluoropyrrolidin-1-yl)methyl)pheno...)
Affinity DataKi:  0.280nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50278446((R)-3-fluoro-1-(4-(3-(pyrrolidin-1-yl)propoxy)benz...)
Affinity DataKi:  0.310nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50159110(1-(3-(4-(piperidin-1-ylmethyl)phenoxy)propyl)piper...)
Affinity DataKi:  0.580nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50278496(1-(4-(3-(piperidin-1-yl)propoxy)benzyl)piperidin-4...)
Affinity DataKi:  0.840nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50278447(4-fluoro-1-(3-(4-(pyrrolidin-1-ylmethyl)phenoxy)pr...)
Affinity DataKi:  0.990nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50247053(1-(3-(3-(4-chlorophenyl)propoxy)propyl)piperidine ...)
Affinity DataKi:  2.70nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50126888(1-[4-(4-Piperidin-1-ylmethyl-benzyloxy)-benzyl]-pi...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50133003(4-(3-(piperidin-1-yl)propoxy)benzonitrile | 4-(3-P...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50278398(1-(3-(4-(fluoromethyl)phenoxy)propyl)piperidine | ...)
Affinity DataKi:  17.3nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50278399(1-(3-(4-(2-fluoroethyl)phenoxy)propyl)piperidine |...)
Affinity DataKi:  43nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Johann Wolfgang Goethe-UniversitäT

Curated by ChEMBL
LigandPNGBDBM50278397(4-(3-(4,4-difluoropiperidin-1-yl)propoxy)benzonitr...)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in HEL293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidylate synthase(Homo sapiens (Human))
University College Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50316412(2-amino-4-oxo-5-thiopyridyl-6-methyl pyrrolo(2,3-d...)
Affinity DataIC50:  340nMAssay Description:Inhibition of thymidylate synthaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10/8/9(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102624(CHEMBL1234032)
Affinity DataIC50:  1.59E+3nMAssay Description:Inhibition of JNK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102618(CHEMBL3342921)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102620(CHEMBL3342924)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102615(CHEMBL3342918)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102632(CHEMBL3342913)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102619(CHEMBL3342922)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102617(CHEMBL3342920)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102613(CHEMBL3342917)
Affinity DataIC50:  5.80E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102629(CHEMBL3342912)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102616(CHEMBL3342919)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102626(CHEMBL3342908)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102622(CHEMBL3342926)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102621(CHEMBL3342925)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102611(CHEMBL3342915)
Affinity DataIC50:  6.90E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102628(CHEMBL3342910)
Affinity DataIC50:  8.10E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102623(CHEMBL3342928)
Affinity DataIC50:  8.90E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102612(CHEMBL3342916)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102625(CHEMBL3342907)
Affinity DataIC50:  9.60E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102627(CHEMBL3342909)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Kakatiya University

Curated by ChEMBL
LigandPNGBDBM50102607(CHEMBL3342914)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of FLAG-tagged JNK-1 (unknown origin) transfected in African green monkey COS cells by SDS-PAGE analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed