Compile Data Set for Download or QSAR
maximum 50k data
Found 479 with Last Name = 'gaudette' and Initial = 'f'
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303276(CHEMBL565807 | N-(4-(2-(1-ethyl-1H-imidazole-4-car...)
Affinity DataIC50:  1nMAssay Description:Inhibition of VEGFR2 assessed as inhibition of ERK phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM93149(2-oxoimidazolidine-1-carboxamide, 16)
Affinity DataIC50:  2nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM93147(2-oxoimidazolidine-1-carboxamide, 14)
Affinity DataIC50:  3nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248054(CHEMBL508395 | N-(3-fluoro-4-(2-(4-((methyl(2-(4-m...)
Affinity DataIC50:  3nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248089(CHEMBL517469 | N-(4-(2-(1-ethyl-1H-imidazol-4-yl)t...)
Affinity DataIC50:  3nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM93145(2-oxoimidazolidine-1-carboxamide, 5)
Affinity DataIC50:  4nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM93150(2-oxoimidazolidine-1-carboxamide, 17)
Affinity DataIC50:  4nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303262(CHEMBL566010 | N1-(3-fluoro-4-(2-(pyrrolidine-1-ca...)
Affinity DataIC50:  4nMAssay Description:Inhibition of GST-fused recombinant VEGFR2 expressed in baculovirus infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303276(CHEMBL565807 | N-(4-(2-(1-ethyl-1H-imidazole-4-car...)
Affinity DataIC50:  4nMAssay Description:Inhibition of TPR-met autophosphorylation expressed in HEK293T cells after 150 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM93148(2-oxoimidazolidine-1-carboxamide, 15)
Affinity DataIC50:  5nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303266(CHEMBL565990 | N1-(4-(2-(1-ethyl-1H-imidazole-4-ca...)
Affinity DataIC50:  5nMAssay Description:Inhibition of GST-fused recombinant VEGFR2 expressed in baculovirus infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303272(CHEMBL567475 | N1-(4-(2-(1-ethyl-1H-imidazole-4-ca...)
Affinity DataIC50:  5nMAssay Description:Inhibition of GST-fused recombinant VEGFR2 expressed in baculovirus infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303267(CHEMBL576504 | N1-(4-(2-(1-(2-(dimethylamino)ethyl...)
Affinity DataIC50:  6nMAssay Description:Inhibition of GST-fused recombinant VEGFR2 expressed in baculovirus infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303273(CHEMBL566844 | N1-(4-(2-(1-ethyl-1H-imidazole-4-ca...)
Affinity DataIC50:  6nMAssay Description:Inhibition of GST-fused recombinant VEGFR2 expressed in baculovirus infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303277(CHEMBL565782 | N1-(4-(2-(1-ethyl-1H-imidazole-4-ca...)
Affinity DataIC50:  6nMAssay Description:Inhibition of GST-fused recombinant VEGFR2 expressed in baculovirus infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248088(CHEMBL464211 | N-(4-(2-(1-ethyl-1H-imidazol-4-yl)t...)
Affinity DataIC50:  7nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248510(CHEMBL489326 | N-(4-(6,7-dimethoxyquinolin-4-yloxy...)
Affinity DataIC50:  7nMAssay Description:Inhibition of VEGFR2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303275(CHEMBL584701 | N1-(4-(2-(1-ethyl-1H-imidazole-4-ca...)
Affinity DataIC50:  7nMAssay Description:Inhibition of GST-fused recombinant VEGFR2 expressed in baculovirus infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50247962(CHEMBL462232 | N-(3-fluoro-4-(2-(1-methyl-1H-imida...)
Affinity DataIC50:  8nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248048(CHEMBL449757 | N-(3-fluoro-4-(2-(1-(3-(pyrrolidin-...)
Affinity DataIC50:  8nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248053(4-(4-(7-(2-fluoro-4-(2-oxo-3-phenylimidazolidine-1...)
Affinity DataIC50:  8nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303276(CHEMBL565807 | N-(4-(2-(1-ethyl-1H-imidazole-4-car...)
Affinity DataIC50:  8nMAssay Description:Inhibition of GST-fused recombinant VEGFR2 expressed in baculovirus infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248558(CHEMBL465131 | N-(3-fluoro-4-(2-(1-methyl-1H-imida...)
Affinity DataIC50:  9nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50247984(CHEMBL453613 | N-(4-(2-(1-ethyl-1H-imidazol-4-yl)t...)
Affinity DataIC50:  10nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50299777(CHEMBL573761 | N-(4-(6,7-dimethoxyquinolin-4-yloxy...)
Affinity DataIC50:  10nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248557(CHEMBL465130 | N1-(3-fluoro-4-(2-(1-methyl-1H-imid...)
Affinity DataIC50:  10nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248557(CHEMBL465130 | N1-(3-fluoro-4-(2-(1-methyl-1H-imid...)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant GST-fused VEGFR2 expressed in baculovirus infected Sf9 cells by DELFIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50306503(4,4,4-trifluoro-3-(3-fluoro-4-(2-(1-methyl-1H-imid...)
Affinity DataIC50:  10nMAssay Description:Inhibition of recombinant GST-fused VEGFR2 expressed in baculovirus infected Sf9 cells by DELFIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303269(CHEMBL585205 | N1-cyclohexyl-N3-(4-(2-(1-ethyl-1H-...)
Affinity DataIC50:  10nMAssay Description:Inhibition of GST-fused recombinant VEGFR2 expressed in baculovirus infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303271(CHEMBL565603 | N1-(4-(2-(1-ethyl-1H-imidazole-4-ca...)
Affinity DataIC50:  10nMAssay Description:Inhibition of GST-fused recombinant VEGFR2 expressed in baculovirus infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50247962(CHEMBL462232 | N-(3-fluoro-4-(2-(1-methyl-1H-imida...)
Affinity DataIC50:  10nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50306503(4,4,4-trifluoro-3-(3-fluoro-4-(2-(1-methyl-1H-imid...)
Affinity DataIC50:  10nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248051(CHEMBL448276 | N-(3-fluoro-4-(2-(4-(piperazin-1-yl...)
Affinity DataIC50:  11nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50247984(CHEMBL453613 | N-(4-(2-(1-ethyl-1H-imidazol-4-yl)t...)
Affinity DataIC50:  12nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248052(CHEMBL447616 | N-(3-fluoro-4-(2-(4-((4-methylpiper...)
Affinity DataIC50:  12nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248091(CHEMBL518676 | N-(3-fluoro-4-(2-(1-methyl-1H-imida...)
Affinity DataIC50:  12nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303274(CHEMBL577742 | N1-(4-(2-(1-ethyl-1H-imidazole-4-ca...)
Affinity DataIC50:  13nMAssay Description:Inhibition of GST-fused recombinant VEGFR2 expressed in baculovirus infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248046(CHEMBL445871 | N-(4-(2-(1-(2-(dimethylamino)ethyl)...)
Affinity DataIC50:  14nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248090(CHEMBL462835 | N-(4-(2-(1-ethyl-1H-imidazol-4-yl)t...)
Affinity DataIC50:  14nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248556(CHEMBL464510 | N1-(3-fluoro-4-(2-(1-methyl-1H-imid...)
Affinity DataIC50:  15nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303278(CHEMBL566836 | N-(4-(2-(1-ethyl-1H-imidazole-4-car...)
Affinity DataIC50:  15nMAssay Description:Inhibition of GST-fused recombinant VEGFR2 expressed in baculovirus infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248053(4-(4-(7-(2-fluoro-4-(2-oxo-3-phenylimidazolidine-1...)
Affinity DataIC50:  16nMAssay Description:Inhibition of GST-fused recombinant c-Met (unknown origin) catalytic domain expressed in baculovirus-infected Trichoplusia ni Hi5 cells after 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248602(CHEMBL459478 | N-(3-fluoro-4-(2-(1-isopropyl-1H-im...)
Affinity DataIC50:  16nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303270(CHEMBL566215 | N1-(4-(2-(1-ethyl-1H-imidazole-4-ca...)
Affinity DataIC50:  18nMAssay Description:Inhibition of GST-fused recombinant VEGFR2 expressed in baculovirus infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303268(2-(4-(7-(2-fluoro-4-(3-oxo-3-(phenylamino)propanam...)
Affinity DataIC50:  19nMAssay Description:Inhibition of GST-fused recombinant VEGFR2 expressed in baculovirus infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50303266(CHEMBL565990 | N1-(4-(2-(1-ethyl-1H-imidazole-4-ca...)
Affinity DataIC50:  19nMAssay Description:Inhibition of GST-fused recombinant C-met expressed in baculovirus infected high five cells after 30 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50247984(CHEMBL453613 | N-(4-(2-(1-ethyl-1H-imidazol-4-yl)t...)
Affinity DataIC50:  20nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Methylgene

LigandPNGBDBM93146(2-oxoimidazolidine-1-carboxamide, 13)
Affinity DataIC50:  20nMAssay Description:Inhibition assay using kinase inhibitors.More data for this Ligand-Target Pair
In DepthDetails
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50247962(CHEMBL462232 | N-(3-fluoro-4-(2-(1-methyl-1H-imida...)
Affinity DataIC50:  20nMAssay Description:Inhibition of c-MetMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Methylgene

Curated by ChEMBL
LigandPNGBDBM50248047(CHEMBL503524 | N-(3-fluoro-4-(2-(1-(2-(pyrrolidin-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of GST-fused recombinant VGFR2 (unknown origin) catalytic domain expressed in baculovirus-infected Sf9 cells after 10 mins by DELFIA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 479 total ) | Next | Last >>
Jump to: