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Found 40 with Last Name = 'gaudy' and Initial = 'f'
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataKi:  0.270nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1C(Gallus gallus)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.460nMAssay Description:In vitro binding affinity against melatonin receptor using 2-[125I]iodomelatonin (0.05 nM) and chicken brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50470867(CHEMBL318179)
Affinity DataKi:  0.700nMAssay Description:In vitro binding affinity against melatonin receptor using 2-[125I]iodomelatonin (0.05 nM) and chicken brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataKi:  1.09nMAssay Description:The compound was evaluated for binding affinity against 5-hydroxytryptamine 1A receptor in rat hippocampal membranes using [3H]-8-OH-DPAT as radiolig...More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataKi:  2.30nMAssay Description:The compound was evaluated for binding affinity against 5-hydroxytryptamine 1A receptor in rat hippocampal membranes using [3H]-8-OH-DPAT as radiolig...More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50016737((8-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-dip...)
Affinity DataKi:  3.10nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1C(Gallus gallus)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50470869(CHEMBL12477)
Affinity DataKi:  6nMAssay Description:In vitro binding affinity against melatonin receptor using 2-[125I]iodomelatonin (0.05 nM) and chicken brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280934(1-tert-Butylamino-3-(thiochroman-8-yloxy)-propan-2...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280934(1-tert-Butylamino-3-(thiochroman-8-yloxy)-propan-2...)
Affinity DataKi:  18nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280931(7-Dipropylamino-4-methyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKi:  18nMAssay Description:The compound was evaluated for binding affinity against 5-hydroxytryptamine 1A receptor in rat hippocampal membranes using [3H]-8-OH-DPAT as radiolig...More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280931(7-Dipropylamino-4-methyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKi:  18.4nMAssay Description:The compound was evaluated for binding affinity against 5-hydroxytryptamine 1A receptor in rat hippocampal membranes using [3H]-8-OH-DPAT as radiolig...More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280932(9-Methoxy-1,2,3,4-tetrahydro-anthracen-2-ylamine |...)
Affinity DataKi:  23nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in rat striatal membranes using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1C(Gallus gallus)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50470866(CHEMBL320810)
Affinity DataKi:  29nMAssay Description:Binding affinity towards melatonin receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50470868(CHEMBL12795)
Affinity DataKi:  29nMAssay Description:In vitro binding affinity against melatonin receptor using 2-[125I]iodomelatonin (0.05 nM) and chicken brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50470871(CHEMBL106276)
Affinity DataKi:  32nMAssay Description:In vitro binding affinity against melatonin receptor using 2-[125I]iodomelatonin (0.05 nM) and chicken brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280934(1-tert-Butylamino-3-(thiochroman-8-yloxy)-propan-2...)
Affinity DataKi:  38nMAssay Description:The compound was evaluated for binding affinity against 5-hydroxytryptamine 1A receptor in rat hippocampal membranes using [3H]8-OH-DPAT as radioliga...More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280931(7-Dipropylamino-4-methyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKi:  47nMAssay Description:The compound was evaluated for binding affinity against 5-hydroxytryptamine 1A receptor in rat hippocampal membranes using [3H]-8-OH-DPAT as radiolig...More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280935(10-Methoxy-1,2,3,4-tetrahydro-phenanthren-2-ylamin...)
Affinity DataKi:  76nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in rat striatal membranes using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280931(7-Dipropylamino-4-methyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKi:  81nMAssay Description:The compound was evaluated for binding affinity against 5-hydroxytryptamine 1A receptor in rat hippocampal membranes using [3H]-8-OH-DPAT as radiolig...More data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280936((8-Methoxy-5-methyl-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  115nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50016733(8-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-ylamine ...)
Affinity DataKi:  158nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1C(Gallus gallus)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50035176(8-M-ADOT | CHEMBL53015 | N-(8-Methoxy-1,2,3,4-tetr...)
Affinity DataKi:  161nMAssay Description:In vitro binding affinity against melatonin receptor using 2-[125I]iodomelatonin (0.05 nM) and chicken brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50470870(CHEMBL104997)
Affinity DataKi:  168nMAssay Description:In vitro binding affinity against melatonin receptor using 2-[125I]iodomelatonin (0.05 nM) and chicken brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50470866(CHEMBL320810)
Affinity DataKi:  195nMAssay Description:In vitro binding affinity against melatonin receptor using 2-[125I]iodomelatonin (0.05 nM) and chicken brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1C(Gallus gallus)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM50470865(CHEMBL317669)
Affinity DataKi:  273nMAssay Description:In vitro binding affinity against melatonin receptor using 2-[125I]iodomelatonin (0.05 nM) and chicken brain membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280933(8-Methoxy-5-methyl-1,2,3,4-tetrahydro-naphthalen-2...)
Affinity DataKi:  436nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280936((8-Methoxy-5-methyl-1,2,3,4-tetrahydro-naphthalen-...)
Affinity DataKi:  575nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in rat striatal membranes using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50016733(8-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-ylamine ...)
Affinity DataKi:  902nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in rat striatal membranes using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280937(2-Dipropylamino-1,2,3,4-tetrahydro-anthracen-9-ol ...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in rat striatal membranes using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280935(10-Methoxy-1,2,3,4-tetrahydro-phenanthren-2-ylamin...)
Affinity DataKi:  1.06E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280938((10-Methoxy-1,2,3,4-tetrahydro-phenanthren-2-yl)-d...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1C(Gallus gallus)
Cnrs-Biocis

Curated by ChEMBL
LigandPNGBDBM29612(CHEMBL33103 | CVD-0001578 | JOH-MSK-a63bdd1d-4 | N...)
Affinity DataKi:  1.64E+3nMAssay Description:In vitro binding affinity against melatonin receptor using 2-[125I]iodomelatonin (0.05 nM) and chicken brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280937(2-Dipropylamino-1,2,3,4-tetrahydro-anthracen-9-ol ...)
Affinity DataKi:  2.52E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280932(9-Methoxy-1,2,3,4-tetrahydro-anthracen-2-ylamine |...)
Affinity DataKi:  2.52E+3nMAssay Description:Displacement of [3H]-8-OH-DPAT from rat hippocampal 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50016737((8-Methoxy-1,2,3,4-tetrahydro-naphthalen-2-yl)-dip...)
Affinity DataKi:  3.97E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in rat striatal membranes using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280938((10-Methoxy-1,2,3,4-tetrahydro-phenanthren-2-yl)-d...)
Affinity DataKi:  6.34E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in rat striatal membranes using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in rat striatal membranes using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280931(7-Dipropylamino-4-methyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in rat striatal membranes using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
Target5-hydroxytryptamine receptor 1B(Rattus norvegicus (Rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50280933(8-Methoxy-5-methyl-1,2,3,4-tetrahydro-naphthalen-2...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity against 5-hydroxytryptamine 1B receptor in rat striatal membranes using [3H]-5-HT as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article