Compile Data Set for Download or QSAR
maximum 50k data
Found 28 with Last Name = 'gavenonis' and Initial = 'j'
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50008059(CHEBI:5292 | GELDANAMYCIN)
Affinity DataIC50: <10nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
TargetHeat shock protein HSP 90(Oryctolagus cuniculus)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50008059(CHEBI:5292 | GELDANAMYCIN)
Affinity DataIC50:  282nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048520(CHEMBL3360777)
Affinity DataIC50:  730nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90(Oryctolagus cuniculus)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048520(CHEMBL3360777)
Affinity DataIC50:  4.11E+3nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90(Oryctolagus cuniculus)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048519(CHEMBL3360776)
Affinity DataIC50:  8.43E+3nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048498(CHEMBL3360774)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90(Oryctolagus cuniculus)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048494(CHEMBL3360770)
Affinity DataIC50:  1.44E+4nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048490(Coumermycin A1)
Affinity DataIC50:  1.53E+4nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048494(CHEMBL3360770)
Affinity DataIC50:  1.58E+4nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048499(CHEMBL3360775)
Affinity DataIC50:  1.68E+4nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048492(CHEMBL3360767)
Affinity DataIC50:  1.86E+4nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048493(CHEMBL3360769)
Affinity DataIC50:  1.88E+4nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048519(CHEMBL3360776)
Affinity DataIC50: >2.70E+4nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90(Oryctolagus cuniculus)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048490(Coumermycin A1)
Affinity DataIC50:  2.81E+4nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90(Oryctolagus cuniculus)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048499(CHEMBL3360775)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90(Oryctolagus cuniculus)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048497(CHEMBL3360773)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90(Oryctolagus cuniculus)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048493(CHEMBL3360769)
Affinity DataIC50:  3.79E+4nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90(Oryctolagus cuniculus)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048498(CHEMBL3360774)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048496(CHEMBL3360772)
Affinity DataIC50: >6.70E+4nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90(Oryctolagus cuniculus)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048492(CHEMBL3360767)
Affinity DataIC50:  9.45E+4nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048495(CHEMBL3360771)
Affinity DataIC50: >1.20E+5nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048497(CHEMBL3360773)
Affinity DataIC50:  1.21E+5nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90(Oryctolagus cuniculus)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048496(CHEMBL3360772)
Affinity DataIC50:  1.37E+5nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048491(CHEMBL3360762)
Affinity DataIC50: >1.60E+5nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90(Oryctolagus cuniculus)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048495(CHEMBL3360771)
Affinity DataIC50:  1.68E+5nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50423645(Albamycin | Cathomycin | NOVOBIOCIN)
Affinity DataIC50:  2.31E+5nMAssay Description:Inhibition of HSP90 in human MDA-kb2 cells assessed as reduction in glucocorticoid receptor-dependent luciferase expression after 18 hrs by firefly l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90(Oryctolagus cuniculus)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50048491(CHEMBL3360762)
Affinity DataIC50:  2.33E+5nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeat shock protein HSP 90(Oryctolagus cuniculus)
Tufts University

Curated by ChEMBL
LigandPNGBDBM50423645(Albamycin | Cathomycin | NOVOBIOCIN)
Affinity DataIC50:  4.14E+5nMAssay Description:Inhibition of HSP90 in rabbit reticulocyte lysate after 90 mins by luciferase renaturation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed