TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: 2.17E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: 7.88E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: 1.04E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: 2.25E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: 1.43E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: 3.65E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: 2.08E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: 120nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: 6.27E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: 420nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: 6.91E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: 3.32E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: 3.11E+3nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.70E+3nMAssay Description:Agonist activity at human FXR expressed in COS1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite Louis Pasteur
Curated by ChEMBL
Universite Louis Pasteur
Curated by ChEMBL
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at TGR5 expressed in CHO cells by CRE-driven luciferase reporter gene assayMore data for this Ligand-Target Pair