TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of California Berkeley
Curated by ChEMBL
University Of California Berkeley
Curated by ChEMBL
Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of California Berkeley
Curated by ChEMBL
University Of California Berkeley
Curated by ChEMBL
Affinity DataKi: 8.80nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 375nMAssay Description:Irreversible inhibition of human 20S proteasome beta5 subunit using suc-LLVY-AMC as substrate after 4 hrs at 30 mins time interval by fluorescence as...More data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of California Berkeley
Curated by ChEMBL
University Of California Berkeley
Curated by ChEMBL
Affinity DataKi: 410nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of California Berkeley
Curated by ChEMBL
University Of California Berkeley
Curated by ChEMBL
Affinity DataKi: 470nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
University Of California Berkeley
Curated by ChEMBL
University Of California Berkeley
Curated by ChEMBL
Affinity DataKi: 590nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB1 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of California Berkeley
Curated by ChEMBL
University Of California Berkeley
Curated by ChEMBL
Affinity DataKi: 860nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
TargetCannabinoid receptor 2(Homo sapiens (Human))
University Of California Berkeley
Curated by ChEMBL
University Of California Berkeley
Curated by ChEMBL
Affinity DataKi: 1.03E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant CB2 receptor expressed in HEK293 cells after 90 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.74E+3nMAssay Description:Irreversible inhibition of human 20S proteasome beta5 subunit using suc-LLVY-AMC as substrate after 4 hrs at 30 mins time interval by fluorescence as...More data for this Ligand-Target Pair
Affinity DataKi: 3.92E+4nMAssay Description:Irreversible inhibition of human 20S proteasome beta5 subunit using suc-LLVY-AMC as substrate after 4 hrs at 30 mins time interval by fluorescence as...More data for this Ligand-Target Pair
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of C-terminal his6-tagged recombinant SARS-CoV-2 3CL protease expressed in Escherichia coli BL21 (DE3) using Dabcyl-KNSTLQSGLRKE-Edans as ...More data for this Ligand-Target Pair
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of SARS-CoV-2 3CL proteaseMore data for this Ligand-Target Pair
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of SARS-CoV-2 3CL protease expressed in Escherichia coli BL21 (DE3) using DABCYLKTSAVLQSGFRKME-EDANS as substrate preincubated for 1 hr fo...More data for this Ligand-Target Pair
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of SARS-CoV-2 3CL protease expressed in Escherichia coli BL21 (DE3) using DABCYLKTSAVLQSGFRKME-EDANS as substrate preincubated for 1 hr fo...More data for this Ligand-Target Pair
Affinity DataIC50: 3.80E+4nMAssay Description:Inhibition of SARS-CoV-2 3CL protease expressed in Escherichia coli BL21 (DE3) using DABCYLKTSAVLQSGFRKME-EDANS as substrate preincubated for 1 hr fo...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+5nMAssay Description:Inhibition of SARS-CoV 2 spike glycoproteinMore data for this Ligand-Target Pair