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Found 15 with Last Name = 'gidlöf' and Initial = 'r'
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333162(2-(4-Methylphenyl)-9-[2-(3-thienyl)ethyl]-2,6-dihy...)
Affinity DataKi:  0.140nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha1beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
Target InfoGoogleScholar
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333160(9-Methyl-2-phenyl-2,6-dihydro[1,2,4]triazolo[4,3-c...)
Affinity DataKi:  0.430nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha1beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
Target InfoGoogleScholar
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333163(2-(4-Methylphenyl)-9-[2-(3-pyridyl)ethyl]-2,6-dihy...)
Affinity DataKi:  0.680nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha1beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
Target InfoGoogleScholar
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333162(2-(4-Methylphenyl)-9-[2-(3-thienyl)ethyl]-2,6-dihy...)
Affinity DataKi:  0.710nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha3beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333160(9-Methyl-2-phenyl-2,6-dihydro[1,2,4]triazolo[4,3-c...)
Affinity DataKi:  1nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha2beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333160(9-Methyl-2-phenyl-2,6-dihydro[1,2,4]triazolo[4,3-c...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha3beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333162(2-(4-Methylphenyl)-9-[2-(3-thienyl)ethyl]-2,6-dihy...)
Affinity DataKi:  1.70nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha2beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333163(2-(4-Methylphenyl)-9-[2-(3-pyridyl)ethyl]-2,6-dihy...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha3beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333161(2-(4-Methylphenyl)-9-(2-phenylethyl)-2,6-dihydro[1...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha1beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
Target InfoGoogleScholar
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333162(2-(4-Methylphenyl)-9-[2-(3-thienyl)ethyl]-2,6-dihy...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha5beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333163(2-(4-Methylphenyl)-9-[2-(3-pyridyl)ethyl]-2,6-dihy...)
Affinity DataKi:  4.40nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha2beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333163(2-(4-Methylphenyl)-9-[2-(3-pyridyl)ethyl]-2,6-dihy...)
Affinity DataKi:  9.10nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha5beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333161(2-(4-Methylphenyl)-9-(2-phenylethyl)-2,6-dihydro[1...)
Affinity DataKi:  9.70nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha3beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333161(2-(4-Methylphenyl)-9-(2-phenylethyl)-2,6-dihydro[1...)
Affinity DataKi:  65nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha2beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
Lund University

Curated by ChEMBL
LigandPNGBDBM50333161(2-(4-Methylphenyl)-9-(2-phenylethyl)-2,6-dihydro[1...)
Affinity DataKi:  66nMAssay Description:Displacement of [3H]flumazenil human recombinant alpha5beta3gamma2 GABA(A) receptor expressed in HEK293 cells after 30 mins by glass fiber filtration...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed