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Found 45 with Last Name = 'gillen' and Initial = 'ml'
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.0800nMAssay Description:Inhibition of the 2-[125I]- iodomelatonin binding to Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)
Affinity DataKi:  0.0800nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50035202(CHEMBL291857 | N-[2-(2,7-Dimethoxy-naphthalen-1-yl...)
Affinity DataKi:  0.0990nMAssay Description:Inhibition of the 2-[125I]- iodomelatonin binding to Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50035202(CHEMBL291857 | N-[2-(2,7-Dimethoxy-naphthalen-1-yl...)
Affinity DataKi:  0.0990nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.120nMAssay Description:Inhibition of the 2-[125I]- iodomelatonin binding to Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.130nMAssay Description:Binding affinity of the compound against human Melatonin receptor type 1A by displacement of [125I]-iodomelatonin stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticleDrugBank

TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM29611(2-Iodomelatonin | CHEMBL289233 | Melatonin,2-Iodo)
Affinity DataKi:  0.150nMAssay Description:Compound was tested for binding affinity against human Melatonin receptor type 1B in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.200nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticleDrugBank

TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.230nMAssay Description:Binding affinity of the compound against human Melatonin receptor type 1B by displacement of [125I]-iodomelatonin stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticleDrugBank

TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.290nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticleDrugBank

TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50035202(CHEMBL291857 | N-[2-(2,7-Dimethoxy-naphthalen-1-yl...)
Affinity DataKi:  0.380nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50035202(CHEMBL291857 | N-[2-(2,7-Dimethoxy-naphthalen-1-yl...)
Affinity DataKi:  0.380nMAssay Description:Inhibition of the 2-[125I]- iodomelatonin binding to Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290238(CHEMBL80736 | N-[2-(2-Ethoxy-7-methoxy-naphthalen-...)
Affinity DataKi:  0.390nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290000(CHEMBL68864 | N-[2-(6-Methoxy-quinolin-4-yl)-ethyl...)
Affinity DataKi:  0.410nMAssay Description:Binding affinity of the compound against human Melatonin receptor type 1B by displacement of [125I]-iodomelatonin stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290003(CHEMBL306468 | N-[2-(6-Methoxy-quinolin-4-yl)-ethy...)
Affinity DataKi:  0.960nMAssay Description:Binding affinity of the compound against human Melatonin receptor type 1B by displacement of [125I]-iodomelatonin stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290238(CHEMBL80736 | N-[2-(2-Ethoxy-7-methoxy-naphthalen-...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290234(CHEMBL440692 | N-[2-(2-Hydroxy-7-methoxy-naphthale...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290239(CHEMBL78751 | N-{2-[2-(2-Hydroxy-ethoxy)-7-methoxy...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50061570(Bromo-acetic acid 7-methoxy-1-(2-propionylamino-et...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of the 2-[125I]- iodomelatonin binding to Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290002(CHEMBL69521 | N-[2-(6-Methoxy-quinolin-4-yl)-ethyl...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity of the compound against human Melatonin receptor type 1B by displacement of [125I]-iodomelatonin stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50061569(CHEMBL131919 | Chloro-acetic acid 7-methoxy-1-(2-p...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of the 2-[125I]- iodomelatonin binding to Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290234(CHEMBL440692 | N-[2-(2-Hydroxy-7-methoxy-naphthale...)
Affinity DataKi:  2.20nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290000(CHEMBL68864 | N-[2-(6-Methoxy-quinolin-4-yl)-ethyl...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity of the compound against human Melatonin receptor type 1A by displacement of [125I]-iodomelatonin stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290239(CHEMBL78751 | N-{2-[2-(2-Hydroxy-ethoxy)-7-methoxy...)
Affinity DataKi:  4.30nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290002(CHEMBL69521 | N-[2-(6-Methoxy-quinolin-4-yl)-ethyl...)
Affinity DataKi:  5.90nMAssay Description:Binding affinity of the compound against human Melatonin receptor type 1A by displacement of [125I]-iodomelatonin stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290237(CHEMBL82135 | N-[2-(2-Butoxy-7-methoxy-naphthalen-...)
Affinity DataKi:  6.70nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290003(CHEMBL306468 | N-[2-(6-Methoxy-quinolin-4-yl)-ethy...)
Affinity DataKi:  6.90nMAssay Description:Binding affinity of the compound against human Melatonin receptor type 1A by displacement of [125I]-iodomelatonin stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290237(CHEMBL82135 | N-[2-(2-Butoxy-7-methoxy-naphthalen-...)
Affinity DataKi:  7.70nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290241(CHEMBL311106 | N-[2-(7-Methoxy-2-propoxy-naphthale...)
Affinity DataKi:  8.10nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290236(CHEMBL80792 | N-{2-[2-(2-Dimethylamino-ethoxy)-7-m...)
Affinity DataKi:  10nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50061569(CHEMBL131919 | Chloro-acetic acid 7-methoxy-1-(2-p...)
Affinity DataKi:  11nMAssay Description:Inhibition of the 2-[125I]- iodomelatonin binding to Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290241(CHEMBL311106 | N-[2-(7-Methoxy-2-propoxy-naphthale...)
Affinity DataKi:  16nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290235(CHEMBL78338 | {2-[7-Methoxy-1-(2-propionylamino-et...)
Affinity DataKi:  23nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290236(CHEMBL80792 | N-{2-[2-(2-Dimethylamino-ethoxy)-7-m...)
Affinity DataKi:  42nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290240(CHEMBL79224 | N-{2-[2-(2-Iodo-ethoxy)-7-methoxy-na...)
Affinity DataKi:  73nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290235(CHEMBL78338 | {2-[7-Methoxy-1-(2-propionylamino-et...)
Affinity DataKi:  93nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290240(CHEMBL79224 | N-{2-[2-(2-Iodo-ethoxy)-7-methoxy-na...)
Affinity DataKi:  100nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290004(4-(2-Acetylamino-ethyl)-6-methoxy-1-methyl-quinoli...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity of the compound against human Melatonin receptor type 1B by displacement of [125I]-iodomelatonin stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290001(6-Methoxy-1-methyl-4-(2-propionylamino-ethyl)-quin...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity of the compound against human Melatonin receptor type 1A by displacement of [125I]-iodomelatonin stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290001(6-Methoxy-1-methyl-4-(2-propionylamino-ethyl)-quin...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity of the compound against human Melatonin receptor type 1B by displacement of [125I]-iodomelatonin stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM50290004(4-(2-Acetylamino-ethyl)-6-methoxy-1-methyl-quinoli...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity of the compound against human Melatonin receptor type 1A by displacement of [125I]-iodomelatonin stably expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataKi:  7.10E+3nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM55121(3-HYDROXYTYRAMINE HYDROCHLORIDE | 4-(2-aminoethyl)...)
Affinity DataKi:  9.10E+3nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1B(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of 2-[125I]-Iodomelatonin binding to human Melatonin receptor type 1B expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMelatonin receptor type 1A(Homo sapiens (Human))
Duquesne University

Curated by ChEMBL
LigandPNGBDBM10755(14C-5-hydroxy tryptamine creatinine disulfate | 2-...)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of 2-[125I]-Iodomelatonin from human Melatonin receptor type 1A expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails Article