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Found 31 with Last Name = 'giusti' and Initial = 'l'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50166018(2-[(R)-1-Amino-2-((S)-4-hydroxy-phenyl)-ethyl]-thi...)
Affinity DataKi:  3.10E+3nMAssay Description:Inhibition of [3H]-DAMGO binding to rat whole brain Opioid receptor muMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50589443(CHEMBL5193820)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of CYP1A2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50589443(CHEMBL5193820)
Affinity DataIC50: >1.50E+4nMAssay Description:Inhibition of CYP2D6 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50589443(CHEMBL5193820)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of hERGMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Promidis

Curated by ChEMBL
LigandPNGBDBM50589443(CHEMBL5193820)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of CYP3A4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589438(CHEMBL5179943)
Affinity DataEC50:  130nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589439(CHEMBL5189176)
Affinity DataEC50:  80nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589440(CHEMBL5171378)
Affinity DataEC50:  1.31E+3nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589441(CHEMBL5205223)
Affinity DataEC50:  160nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589442(CHEMBL5206952)
Affinity DataEC50:  640nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589443(CHEMBL5193820)
Affinity DataEC50:  28nMAssay Description:Modulation of capsid assembly in HBV genotype E infected in human HepG2.2.15 cells assessed as inhibition of viral DNA replicationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589444(CHEMBL5208835)
Affinity DataEC50:  440nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589445(CHEMBL5201534)
Affinity DataEC50:  360nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589446(CHEMBL5201042)
Affinity DataEC50:  900nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589447(CHEMBL5169424)
Affinity DataEC50:  630nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589448(CHEMBL5182899)
Affinity DataEC50:  240nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589449(CHEMBL5177883)
Affinity DataEC50:  50nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589450(CHEMBL5207945)
Affinity DataEC50:  530nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589451(CHEMBL5191124)
Affinity DataEC50:  70nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589443(CHEMBL5193820)
Affinity DataEC50:  60nMAssay Description:Modulation of capsid assembly in HBV infected in human HepG2.2.15 cells assessed as inhibition of viral DNA replicationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589443(CHEMBL5193820)
Affinity DataEC50:  1.05E+3nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication in presence of 40% normal human ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589443(CHEMBL5193820)
Affinity DataEC50:  28nMAssay Description:Modulation of capsid assembly in HBV genotype A infected in human HepG2.2.15 cells assessed as inhibition of viral DNA replicationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589443(CHEMBL5193820)
Affinity DataEC50:  28nMAssay Description:Modulation of capsid assembly in HBV genotype B infected in human HepG2.2.15 cells assessed as inhibition of viral DNA replicationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589443(CHEMBL5193820)
Affinity DataEC50:  28nMAssay Description:Modulation of capsid assembly in HBV genotype C infected in human HepG2.2.15 cells assessed as inhibition of viral DNA replicationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589443(CHEMBL5193820)
Affinity DataEC50:  39nMAssay Description:Modulation of capsid assembly in HBV genotype D infected in human HepG2.2.15 cells assessed as inhibition of viral DNA replicationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589437(CHEMBL5188350)
Affinity DataEC50:  500nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589436(CHEMBL5175001)
Affinity DataEC50:  6.68E+3nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589435(CHEMBL5180875)
Affinity DataEC50:  130nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589434(CHEMBL5198985)
Affinity DataEC50:  2.40E+3nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50535698(CHEMBL4533071)
Affinity DataEC50:  260nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
TargetCapsid protein(Hepatitis B virus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50589443(CHEMBL5193820)
Affinity DataEC50:  62nMAssay Description:Modulation of capsid assembly in HBV infected in human HePAD38 cells assessed as inhibition of viral DNA replication measured after 96 hrs by qPCR an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed