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Found 18 with Last Name = 'goodsell' and Initial = 'ds'
TargetGag-Pol polyprotein [489-587,G537V,H558K,V571A](Human immunodeficiency virus)
The Scripps Research Institute

LigandPNGBDBM84460(HIV-1 PR Inhibitor, compound 6)
Affinity DataKi:  1.70nM IC50:  6nMAssay Description:The inhibition activity against HIV-1 PR and three mutants (G48V, V82F, V82A)were done in 96 well microtiter plate and were assayed. Wells that show...More data for this Ligand-Target Pair
Ligand InfoMMDBPC cidPC sid
In DepthDetails ArticlePubMedMMDB

TargetGag-Pol polyprotein [489-587,G537V,H558K,V571A](Human immunodeficiency virus)
The Scripps Research Institute

LigandPNGBDBM84461(HIV-1 PR Inhibitor, compound 8)
Affinity DataKi:  4nM IC50:  13nMAssay Description:The inhibition activity against HIV-1 PR and three mutants (G48V, V82F, V82A)were done in 96 well microtiter plate and were assayed. Wells that show...More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587,G537V,H558K,V571A](Human immunodeficiency virus)
The Scripps Research Institute

LigandPNGBDBM84461(HIV-1 PR Inhibitor, compound 8)
Affinity DataKi:  9.70nM IC50:  17nMAssay Description:The inhibition activity against HIV-1 PR and three mutants (G48V, V82F, V82A)were done in 96 well microtiter plate and were assayed. Wells that show...More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587,G537V,H558K,V571A](Human immunodeficiency virus)
The Scripps Research Institute

LigandPNGBDBM84460(HIV-1 PR Inhibitor, compound 6)
Affinity DataKi:  10nM IC50:  19nMAssay Description:The inhibition activity against HIV-1 PR and three mutants (G48V, V82F, V82A)were done in 96 well microtiter plate and were assayed. Wells that show...More data for this Ligand-Target Pair
Ligand InfoMMDBPC cidPC sid
In DepthDetails ArticlePubMedMMDB

TargetGag-Pol polyprotein [489-587,G537V,H558K,V571A](Human immunodeficiency virus)
The Scripps Research Institute

LigandPNGBDBM84461(HIV-1 PR Inhibitor, compound 8)
Affinity DataKi:  13nM IC50:  24nMAssay Description:The inhibition activity against HIV-1 PR and three mutants (G48V, V82F, V82A)were done in 96 well microtiter plate and were assayed. Wells that show...More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [489-587,G537V,H558K,V571A](Human immunodeficiency virus)
The Scripps Research Institute

LigandPNGBDBM84460(HIV-1 PR Inhibitor, compound 6)
Affinity DataKi:  22nM IC50:  39nMAssay Description:The inhibition activity against HIV-1 PR and three mutants (G48V, V82F, V82A)were done in 96 well microtiter plate and were assayed. Wells that show...More data for this Ligand-Target Pair
Ligand InfoMMDBPC cidPC sid
In DepthDetails ArticlePubMedMMDB

TargetGag-Pol polyprotein [489-587,G537V,H558K,V571A](Human immunodeficiency virus)
The Scripps Research Institute

LigandPNGBDBM84460(HIV-1 PR Inhibitor, compound 6)
Affinity DataKi:  27nM IC50:  46nMAssay Description:The inhibition activity against HIV-1 PR and three mutants (G48V, V82F, V82A)were done in 96 well microtiter plate and were assayed. Wells that show...More data for this Ligand-Target Pair
Ligand InfoMMDBPC cidPC sid
In DepthDetails ArticlePubMedMMDB

TargetGag-Pol polyprotein [489-587,G537V,H558K,V571A](Human immunodeficiency virus)
The Scripps Research Institute

LigandPNGBDBM84461(HIV-1 PR Inhibitor, compound 8)
Affinity DataKi:  30nM IC50:  52nMAssay Description:The inhibition activity against HIV-1 PR and three mutants (G48V, V82F, V82A)were done in 96 well microtiter plate and were assayed. Wells that show...More data for this Ligand-Target Pair
TargetAdenosine 5'-phosphosulfate reductase(Mycobacterium tuberculosis)
The Scripps Research Institute

LigandPNGBDBM25469(2-[(7-nitro-2,1,3-benzoxadiazol-4-yl)sulfanyl]-1-o...)
Affinity DataKd:  1.95E+4nMpH: 7.5 T: 2°CAssay Description:Values of Ki were determined from the dependence of the observed rate constant (kobs) on inhibitor concentration. With subsaturing APS, the inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine 5'-phosphosulfate reductase(Mycobacterium tuberculosis)
The Scripps Research Institute

LigandPNGBDBM22858(1,2-Dione-Based Compound, 15 | 2-nitro-9,10-dihydr...)
Affinity DataKd:  6.81E+3nMpH: 7.5 T: 2°CAssay Description:Values of Ki were determined from the dependence of the observed rate constant (kobs) on inhibitor concentration. With subsaturing APS, the inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine 5'-phosphosulfate reductase(Mycobacterium tuberculosis)
The Scripps Research Institute

LigandPNGBDBM25468(3,7-difluoro-2-nitro-9H-fluoren-9-one | NSC57476)
Affinity DataKd:  4.46E+4nMpH: 7.5 T: 2°CAssay Description:Values of Ki were determined from the dependence of the observed rate constant (kobs) on inhibitor concentration. With subsaturing APS, the inhibit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine 5'-phosphosulfate reductase(Mycobacterium tuberculosis)
The Scripps Research Institute

LigandPNGBDBM25467(2,4-dinitro-9H-fluoren-9-one | NSC55545)
Affinity DataKd:  4.81E+4nMpH: 7.5 T: 2°CAssay Description:Values of Ki were determined from the dependence of the observed rate constant (kobs) on inhibitor concentration. With subsaturing APS, the inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine 5'-phosphosulfate reductase(Mycobacterium tuberculosis)
The Scripps Research Institute

LigandPNGBDBM25466(N-(3-nitro-9-oxo-9H-fluoren-2-yl)acetamide | NSC60...)
Affinity DataKd:  3.18E+4nMpH: 7.5 T: 2°CAssay Description:Values of Ki were determined from the dependence of the observed rate constant (kobs) on inhibitor concentration. With subsaturing APS, the inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine 5'-phosphosulfate reductase(Mycobacterium tuberculosis)
The Scripps Research Institute

LigandPNGBDBM25465((1R,2R,5S,6S,10S,13S,15R)-5-acetyl-13-hydroxy-6,10...)
Affinity DataKd:  1.27E+5nMpH: 7.5 T: 2°CAssay Description:Values of Ki were determined from the dependence of the observed rate constant (kobs) on inhibitor concentration. With subsaturing APS, the inhibit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine 5'-phosphosulfate reductase(Mycobacterium tuberculosis)
The Scripps Research Institute

LigandPNGBDBM25464(6-[(7-nitro-2,1,3-benzoxadiazol-4-yl)sulfanyl]-9H-...)
Affinity DataKd:  1.52E+4nMpH: 7.5 T: 2°CAssay Description:Values of Ki were determined from the dependence of the observed rate constant (kobs) on inhibitor concentration. With subsaturing APS, the inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine 5'-phosphosulfate reductase(Mycobacterium tuberculosis)
The Scripps Research Institute

LigandPNGBDBM25463(2-(1,2,4-triazatriphenylen-3-ylsulfanyl)acetic aci...)
Affinity DataKd:  4.69E+4nMpH: 7.5 T: 2°CAssay Description:Values of Ki were determined from the dependence of the observed rate constant (kobs) on inhibitor concentration. With subsaturing APS, the inhibit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine 5'-phosphosulfate reductase(Mycobacterium tuberculosis)
The Scripps Research Institute

LigandPNGBDBM25460(2-[(4-oxo-4H-triphenylene-11-)sulfinyl]acetic acid...)
Affinity DataKd:  1.80E+5nMpH: 7.5 T: 2°CAssay Description:Values of Ki were determined from the dependence of the observed rate constant (kobs) on inhibitor concentration. With subsaturing APS, the inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine 5'-phosphosulfate reductase(Mycobacterium tuberculosis)
The Scripps Research Institute

LigandPNGBDBM25462(2,3-dinitro-9H-fluoren-9-one | NSC133896)
Affinity DataKd:  3.71E+4nMpH: 7.5 T: 2°CAssay Description:Values of Ki were determined from the dependence of the observed rate constant (kobs) on inhibitor concentration. With subsaturing APS, the inhibit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed