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Found 14 with Last Name = 'gudmundsson' and Initial = 'ks'
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50316633((S)-N-((4-(3-(dimethylamino)propyl)isoquinolin-3-y...)
Affinity DataIC50:  3.40nMAssay Description:Binding affinity to human CXCR4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50314758((S)-N-((1-(((S)-1-isopropylpiperidin-3-yl)methyl)-...)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of human CXCR4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50316634((S)-2-(dimethylamino)-N-((3-((methyl(5,6,7,8-tetra...)
Affinity DataIC50:  16nMAssay Description:Binding affinity to human CXCR4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50315287((R)-N1-((1H-benzo[d]imidazol-2-yl)methyl)-N1-(5,6,...)
Affinity DataIC50:  36nMAssay Description:Binding affinity to human CXCR4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50314756(CHEMBL577268 | N-((1-(3-aminopropyl)-1H-benzo[d]im...)
Affinity DataIC50:  47nMAssay Description:Inhibition of human CXCR4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50314757(CHEMBL1091591 | N-methyl-N-((1-(1-methylpiperidin-...)
Affinity DataIC50:  76nMAssay Description:Inhibition of human CXCR4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50269061((1R)-6-Bromo-N-[(1R)-1-phenylethyl]-2,3,4,9-tetrah...)
Affinity DataIC50:  160nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50269061((1R)-6-Bromo-N-[(1R)-1-phenylethyl]-2,3,4,9-tetrah...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50295257((R)-N-(6-chloro-2,3,4,9-tetrahydro-1H-carbazol-1-y...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50295257((R)-N-(6-chloro-2,3,4,9-tetrahydro-1H-carbazol-1-y...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50295256((R)-N-(6-chloro-2,3,4,9-tetrahydro-1H-carbazol-1-y...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50295256((R)-N-(6-chloro-2,3,4,9-tetrahydro-1H-carbazol-1-y...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50295255(6-bromo-N-phenyl-2,3,4,9-tetrahydro-1H-carbazol-1-...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50295255(6-bromo-N-phenyl-2,3,4,9-tetrahydro-1H-carbazol-1-...)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of CYP2D6More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed