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Found 13 with Last Name = 'höltje' and Initial = 'm'
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50120404(Acetic acid 2-(8-hydroxy-6,11-dimethyl-1,2,5,6-tet...)
Affinity DataKi:  228nMAssay Description:Inhibition of [3H]-U-69,593 binding towards Opioid receptor kappa 1 in guinea pig brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Catania

Curated by ChEMBL
LigandPNGBDBM50120406(2-(8-Hydroxy-6,11-dimethyl-1,2,5,6-tetrahydro-4H-2...)
Affinity DataKi:  2.36E+3nMAssay Description:Inhibition of [3H]-U-69,593 binding towards Opioid receptor kappa 1 in guinea pig brain homogenates.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Università

Curated by ChEMBL
LigandPNGBDBM50101397(2-(2,6-Dichloro-phenyl)-3-(6-methyl-pyridin-2-yl)-...)
Affinity DataIC50:  2.24E+3nMAssay Description:HIV-1 reverse transcriptase (RT) activity using Poly (rC)/oligo (dG) as template/primer and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Università

Curated by ChEMBL
LigandPNGBDBM50101407(2-(2,6-Difluoro-phenyl)-3-(4-methyl-pyridin-2-yl)-...)
Affinity DataIC50:  2.84E+3nMAssay Description:HIV-1 reverse transcriptase (RT) activity using Poly (rC)/oligo (dG) as template/primer and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Università

Curated by ChEMBL
LigandPNGBDBM50121354(2-(2-Fluoro-6-methyl-phenyl)-3-(6-methyl-pyridin-2...)
Affinity DataIC50:  2.85E+3nMAssay Description:HIV-1 reverse transcriptase (RT) activity using Poly (rC)/oligo (dG) as template/primer and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Università

Curated by ChEMBL
LigandPNGBDBM50101404(2-(2,6-Difluoro-phenyl)-3-(6-methyl-pyridin-2-yl)-...)
Affinity DataIC50:  2.90E+3nMAssay Description:HIV-1 reverse transcriptase (RT) activity using Poly (rC)/oligo (dG) as template/primer and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Università

Curated by ChEMBL
LigandPNGBDBM50121357(2-(2,6-Difluoro-phenyl)-3-(4,6-dimethyl-pyridin-2-...)
Affinity DataIC50:  4.12E+3nMAssay Description:HIV-1 reverse transcriptase (RT) activity using Poly (rC)/oligo (dG) as template/primer and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Università

Curated by ChEMBL
LigandPNGBDBM50121350(2-(2-Chloro-6-fluoro-phenyl)-3-(4-methyl-pyridin-2...)
Affinity DataIC50:  4.12E+3nMAssay Description:HIV-1 reverse transcriptase (RT) activity using Poly (rC)/oligo (dG) as template/primer and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Università

Curated by ChEMBL
LigandPNGBDBM50121347(CHEMBL625 | THIABENDAZOLE)
Affinity DataIC50:  1.46E+4nMAssay Description:HIV-1 reverse transcriptase (RT) activity using Poly (rC)/oligo (dG) as template/primer and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Università

Curated by ChEMBL
LigandPNGBDBM50121352(2-(2-Chloro-6-methyl-phenyl)-3-(5-methyl-pyridin-2...)
Affinity DataIC50:  4.24E+4nMAssay Description:HIV-1 reverse transcriptase (RT) activity using Poly (rC)/oligo (dG) as template/primer and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Università

Curated by ChEMBL
LigandPNGBDBM50121351(3-(5-Bromo-pyridin-2-yl)-2-(2,6-dichloro-phenyl)-t...)
Affinity DataIC50:  5.66E+4nMAssay Description:HIV-1 reverse transcriptase (RT) activity using Poly (rC)/oligo (dG) as template/primer and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Università

Curated by ChEMBL
LigandPNGBDBM50121356(3-(5-Bromo-pyridin-2-yl)-2-(2,6-difluoro-phenyl)-t...)
Affinity DataIC50:  6.14E+4nMAssay Description:HIV-1 reverse transcriptase (RT) activity using Poly (rC)/oligo (dG) as template/primer and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Università

Curated by ChEMBL
LigandPNGBDBM50121353(3-(5-Chloro-pyridin-2-yl)-2-(2,6-difluoro-phenyl)-...)
Affinity DataIC50:  6.70E+4nMAssay Description:HIV-1 reverse transcriptase (RT) activity using Poly (rC)/oligo (dG) as template/primer and [3H]dGTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed