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Found 78 with Last Name = 'haigh' and Initial = 'rm'
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246925(1-(4-[3-(2,6-Difluorophenyl)ureidomethyl]-3-methyl...)
Affinity DataKi:  200nMAssay Description:Binding affinity to human vasopressin V2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246575(1-(2-Methyl-4-(2,3,4,5-tetrahydro-1-benzazepin-1-y...)
Affinity DataKi:  2.00E+3nMAssay Description:Binding affinity to human vasopressin V2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246925(1-(4-[3-(2,6-Difluorophenyl)ureidomethyl]-3-methyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to oxytocin receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246575(1-(2-Methyl-4-(2,3,4,5-tetrahydro-1-benzazepin-1-y...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to oxytocin receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246890(1-(4-[3-(2,6-Difluorophenyl)ureidomethyl]benzoyl)-...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity to oxytocin receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152972((2S,4R)-4-Methoxy-2-(4-methyl-[1,4]diazepane-1-car...)
Affinity DataEC50:  430nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152973((S)-2-(4-Methyl-[1,4]diazepane-1-carbothioyl)-pyrr...)
Affinity DataEC50:  810nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152972((2S,4R)-4-Methoxy-2-(4-methyl-[1,4]diazepane-1-car...)
Affinity DataEC50:  230nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152974((2S)-N-{2-Methyl-4-[(1-methyl-4,10-dihydropyrazolo...)
Affinity DataEC50:  850nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152975((2S,4R)-4-Methoxy-2-(2-pyridin-2-yl-ethylthiocarba...)
Affinity DataEC50:  200nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152976((3S,5R)-4-Methoxy-pyrrolidine-1,2-dicarboxylic aci...)
Affinity DataEC50:  1.50E+3nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152977((3S,5R)-4-Methoxy-2-(4-pyrrolidin-1-yl-piperidine-...)
Affinity DataEC50:  1.10E+3nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152978((3S,5R)-4-Methoxy-2-(4-methyl-[1,4]diazepane-1-car...)
Affinity DataEC50:  1.30E+3nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152979((S)-2-(4-Methyl-[1,4]diazepane-1-carbothioyl)-pyrr...)
Affinity DataEC50:  890nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152980((3S,5R)-2-([1,4'']Bipiperidinyl-1''-carbonyl)-4-me...)
Affinity DataEC50:  2.20E+3nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152981((2S,4R)-4-Methoxy-2-(4-pyrrolidin-1-yl-piperidine-...)
Affinity DataEC50:  100nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152974((2S)-N-{2-Methyl-4-[(1-methyl-4,10-dihydropyrazolo...)
Affinity DataEC50:  33nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152973((S)-2-(4-Methyl-[1,4]diazepane-1-carbothioyl)-pyrr...)
Affinity DataEC50:  1.80E+3nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152977((3S,5R)-4-Methoxy-2-(4-pyrrolidin-1-yl-piperidine-...)
Affinity DataEC50:  2.30E+3nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152980((3S,5R)-2-([1,4'']Bipiperidinyl-1''-carbonyl)-4-me...)
Affinity DataEC50:  1.20E+3nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152979((S)-2-(4-Methyl-[1,4]diazepane-1-carbothioyl)-pyrr...)
Affinity DataEC50:  640nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152982((2S,4R)-4-Methoxy-pyrrolidine-1,2-dicarboxylic aci...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152976((3S,5R)-4-Methoxy-pyrrolidine-1,2-dicarboxylic aci...)
Affinity DataEC50:  570nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152975((2S,4R)-4-Methoxy-2-(2-pyridin-2-yl-ethylthiocarba...)
Affinity DataEC50:  470nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152982((2S,4R)-4-Methoxy-pyrrolidine-1,2-dicarboxylic aci...)
Affinity DataEC50:  1.80E+3nMAssay Description:Effective concentration for human Vassopressin V2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152978((3S,5R)-4-Methoxy-2-(4-methyl-[1,4]diazepane-1-car...)
Affinity DataEC50:  2.80E+3nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50152981((2S,4R)-4-Methoxy-2-(4-pyrrolidin-1-yl-piperidine-...)
Affinity DataEC50:  480nMAssay Description:Effective concentration for human Oxytocin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246608((4R)-4-Methoxy-1-(2-methyl-4-(2,3,4,5-tetrahydro-1...)
Affinity DataEC50:  4.70nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246609((4R)-4-Ethoxy-1-(2-methyl-4-(2,3,4,5-tetrahydro-1-...)
Affinity DataEC50:  4.30nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246610((4R)-4-tert-Butoxyoxy-1-(2-methyl-4-(2,3,4,5-tetra...)
Affinity DataEC50:  46nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246611((4R)-4-Benzyloxy-1-(2-methyl-4-(2,3,4,5-tetrahydro...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246612(1-(2-Methyl-4-(2,3,4,5-tetrahydro-1-benzazepin-1-y...)
Affinity DataEC50:  27nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246642(4,4-Difluoro-1-(2-methyl-4-(2,3,4,5-tetrahydro-1-b...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246643(4,4-Dimethoxy-1-(2-methyl-4-(2,3,4,5-tetrahydro-1-...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246644(1-(4-(5-Hydroxy-2,3,4,5-tetrahydro-1-benzazepin-1-...)
Affinity DataEC50:  230nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246645(1-(2-Methyl-4-(5-methyl-2,3,4,5-tetrahydro-1-benza...)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246719(1-(4-(5,5-Difluoro-2,3,4,5-tetrahydro-1-benzazepin...)
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246720(1-(2-Methyl-4-(2,3,4,5-tetrahydro-1,5-benzoxazepin...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246721(1-(4-(10,11-Dihydro-5H-pyrrolo[2,1-c][1,4]benzodia...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246722(1-(4-(6,7-Dihydro-5H-dibenzo[b,d]azepin-5-ylcarbon...)
Affinity DataEC50:  84nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246765(1-(4-(6,7-Dihydro-5H-pyrrolo[1,2-a][1,5]benzodiaze...)
Affinity DataEC50:  140nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246925(1-(4-[3-(2,6-Difluorophenyl)ureidomethyl]-3-methyl...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at rat vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246609((4R)-4-Ethoxy-1-(2-methyl-4-(2,3,4,5-tetrahydro-1-...)
Affinity DataEC50:  15nMAssay Description:Agonist activity at rat vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246608((4R)-4-Methoxy-1-(2-methyl-4-(2,3,4,5-tetrahydro-1...)
Affinity DataEC50:  65nMAssay Description:Agonist activity at rat vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246596((4R)-4-Hydroxy-1-(2-methyl-4-(2,3,4,5-tetrahydro-1...)
Affinity DataEC50:  41nMAssay Description:Agonist activity at rat vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246575(1-(2-Methyl-4-(2,3,4,5-tetrahydro-1-benzazepin-1-y...)
Affinity DataEC50:  150nMAssay Description:Agonist activity at rat vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Rattus norvegicus (Rat))
Vantia

Curated by ChEMBL
LigandPNGBDBM50240946(1-(4-[N-(2-dimethylamino-2-oxoethylcarbamoyl)amino...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at rat vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246958(1-(4-[3-(2,6-Difluorophenyl)ureidomethyl]-3-ethylb...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246959(1-(4-[3-(2,6-Difluorophenyl)ureidomethyl]-3,5-dime...)
Affinity DataEC50:  82nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
Vantia

Curated by ChEMBL
LigandPNGBDBM50246889(1-(4-[3-(2-Fluorophenyl)ureidomethyl]-3-methylbenz...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human vasopressin V2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP level by CRE-luciferase report...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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