TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Parke-Davis Pharmaceutical Research
Parke-Davis Pharmaceutical Research
Affinity DataKi: 0.0300nM ΔG°: -62.5kJ/molepH: 6.2 T: 2°CAssay Description:For determination of IC50 values, HIV-1 protease was added to assay buffer containing inhibitor and the substrate (H-His-Lys-Ala-Arg-Val-Leu- (p-NO2)...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Parke-Davis Pharmaceutical Research
Parke-Davis Pharmaceutical Research
Affinity DataKi: 0.0900nMAssay Description:For determination of IC50 values, HIV-1 protease was added to assay buffer containing inhibitor and the substrate (H-His-Lys-Ala-Arg-Val-Leu- (p-NO2)...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Parke-Davis Pharmaceutical Research
Parke-Davis Pharmaceutical Research
Affinity DataKi: 0.0900nMAssay Description:For determination of IC50 values, HIV-1 protease was added to assay buffer containing inhibitor and the substrate (H-His-Lys-Ala-Arg-Val-Leu- (p-NO2)...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Parke-Davis Pharmaceutical Research
Parke-Davis Pharmaceutical Research
Affinity DataKi: 0.110nMAssay Description:For determination of IC50 values, HIV-1 protease was added to assay buffer containing inhibitor and the substrate (H-His-Lys-Ala-Arg-Val-Leu- (p-NO2)...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Parke-Davis Pharmaceutical Research
Parke-Davis Pharmaceutical Research
Affinity DataKi: 0.170nM ΔG°: -58.0kJ/molepH: 6.2 T: 2°CAssay Description:For determination of IC50 values, HIV-1 protease was added to assay buffer containing inhibitor and the substrate (H-His-Lys-Ala-Arg-Val-Leu- (p-NO2)...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Parke-Davis Pharmaceutical Research
Parke-Davis Pharmaceutical Research
Affinity DataKi: 0.430nMAssay Description:For determination of IC50 values, HIV-1 protease was added to assay buffer containing inhibitor and the substrate (H-His-Lys-Ala-Arg-Val-Leu- (p-NO2)...More data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Parke-Davis Pharmaceutical Research
Parke-Davis Pharmaceutical Research
Affinity DataKi: 1.10nMAssay Description:For determination of IC50 values, HIV-1 protease was added to assay buffer containing inhibitor and the substrate (H-His-Lys-Ala-Arg-Val-Leu- (p-NO2)...More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity for adenosine A1 receptor in rat brain membranes using [3H]CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity for adenosine A1 receptor in rat brain membranes using [3H]CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.20nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.40nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Binding affinity towards adenosine A2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 12.1nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Parke-Davis Pharmaceutical Research
Parke-Davis Pharmaceutical Research
Affinity DataKi: 18.4nM ΔG°: -45.9kJ/molepH: 6.2 T: 2°CAssay Description:For determination of IC50 values, HIV-1 protease was added to assay buffer containing inhibitor and the substrate (H-His-Lys-Ala-Arg-Val-Leu- (p-NO2)...More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity for adenosine A1 receptor in rat brain membranes using [3H]CHA as radioligandMore data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Parke-Davis Pharmaceutical Research
Parke-Davis Pharmaceutical Research
Affinity DataKi: 25nMAssay Description:For determination of IC50 values, HIV-1 protease was added to assay buffer containing inhibitor and the substrate (H-His-Lys-Ala-Arg-Val-Leu- (p-NO2)...More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding affinity for adenosine A1 receptor in rat brain membranes using [3H]CHA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Binding affinity for adenosine A1 receptor in rat brain membranes using [3H]CHA as radioligandMore data for this Ligand-Target Pair
TargetDimer of Gag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Parke-Davis Pharmaceutical Research
Parke-Davis Pharmaceutical Research
Affinity DataKi: 31nMAssay Description:For determination of IC50 values, HIV-1 protease was added to assay buffer containing inhibitor and the substrate (H-His-Lys-Ala-Arg-Val-Leu- (p-NO2)...More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 41nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 41.7nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Binding affinity towards adenosine A2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 46nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Binding affinity towards adenosine A1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Binding affinity towards adenosine A2 receptorMore data for this Ligand-Target Pair