Compile Data Set for Download or QSAR
maximum 50k data
Found 134 with Last Name = 'hari' and Initial = 'sb'
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50569820(CHEMBL4860275)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50569815(CHEMBL4873623)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50606915(CHEMBL5219240)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50516529(CHEMBL4520796)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50252344(CHEMBL4086515)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50516522(CHEMBL4447416)
Affinity DataKi:  28nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50606915(CHEMBL5219240)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50569815(CHEMBL4873623)
Affinity DataKi:  210nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50606915(CHEMBL5219240)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50569820(CHEMBL4860275)
Affinity DataKi:  320nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50569815(CHEMBL4873623)
Affinity DataKi:  420nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50516529(CHEMBL4520796)
Affinity DataKi:  430nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50569820(CHEMBL4860275)
Affinity DataKi:  480nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50569815(CHEMBL4873623)
Affinity DataKi:  520nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT1AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50606915(CHEMBL5219240)
Affinity DataKi:  610nMAssay Description:Displacement of [3H]-5Carboxyamidotryptamine from human 5-HT7R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50516522(CHEMBL4447416)
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50516529(CHEMBL4520796)
Affinity DataKi:  1.09E+3nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50252344(CHEMBL4086515)
Affinity DataKi:  1.76E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50516522(CHEMBL4447416)
Affinity DataKi:  1.83E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50252344(CHEMBL4086515)
Affinity DataKi:  1.95E+3nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50606915(CHEMBL5219240)
Affinity DataKi:  2.29E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT1AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50516522(CHEMBL4447416)
Affinity DataKi:  4.54E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT1AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50569820(CHEMBL4860275)
Affinity DataKi:  4.76E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT1AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50569815(CHEMBL4873623)
Affinity DataKi:  5.20E+3nMAssay Description:Displacement of [3H]-5Carboxyamidotryptamine from human 5-HT7R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50569820(CHEMBL4860275)
Affinity DataKi:  5.71E+3nMAssay Description:Displacement of [3H]-5Carboxyamidotryptamine from human 5-HT7R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50252344(CHEMBL4086515)
Affinity DataKi:  9.45E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT1AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50516529(CHEMBL4520796)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [3H]-5Carboxyamidotryptamine from human 5-HT7R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50516529(CHEMBL4520796)
Affinity DataKi:  1.25E+4nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT1AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50252344(CHEMBL4086515)
Affinity DataKi:  1.68E+4nMAssay Description:Displacement of [3H]-5Carboxyamidotryptamine from human 5-HT7R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50516522(CHEMBL4447416)
Affinity DataKi:  3.87E+4nMAssay Description:Displacement of [3H]-5Carboxyamidotryptamine from human 5-HT7R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target1-acyl-sn-glycerol-3-phosphate acyltransferase beta(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50606913(CHEMBL5219455)
Affinity DataIC50:  8.40nMAssay Description:Inhibition of LPAAT-beta (unknown origin) expressed in Xenopus laevis oocytes incubated for 3 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Target1-acyl-sn-glycerol-3-phosphate acyltransferase beta(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50606912(CHEMBL5219496)
Affinity DataIC50:  15nMAssay Description:Inhibition of LPAAT-beta (unknown origin) expressed in Xenopus laevis oocytes incubated for 3 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50116131(CHEMBL66782 | N-(3-Methoxy-4-oxazol-5-yl-phenyl)-6...)
Affinity DataIC50:  54nMAssay Description:Inhibition of IMPDH2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
Target1-acyl-sn-glycerol-3-phosphate acyltransferase beta(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50141287(5TT4A4MBLR | CHEMBL36501 | CT 32228 | CT-32228 | H...)
Affinity DataIC50:  60nMAssay Description:Inhibition of human LPAAT-beta by cell-free colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington

LigandPNGBDBM482158(BDBM50242742 | TAE684)
Affinity DataIC50:  65nMpH: 7.5Assay Description:Inhibitors (initial concentration 10 or 60 μM, three-fold serial dilutions) were incubated with IRE1α* in cleavage buffer (20 mM HEPES at p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington

LigandPNGBDBM50062357(AP26113 | CHEMBL3397300)
Affinity DataIC50:  66nMpH: 7.5Assay Description:Inhibitors (initial concentration 10 or 60 μM, three-fold serial dilutions) were incubated with IRE1α* in cleavage buffer (20 mM HEPES at p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington

LigandPNGBDBM192721(KIRA analog, 3)
Affinity DataIC50:  90nMAssay Description:5′-Carboxyfluorescein (FAM)- and 3′-Black Hole Quencher (BHQ)-labeled XBP1 single stemloop mini-substrate (5′FAM-CUGAGUCCGCAGCACUCA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington

LigandPNGBDBM192751(AT9283)
Affinity DataIC50:  110nMpH: 7.5Assay Description:Inhibitors (initial concentration 10 or 60 μM, three-fold serial dilutions) were incubated with IRE1α* in cleavage buffer (20 mM HEPES at p...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington

LigandPNGBDBM192731(KIRA analog, 13)
Affinity DataIC50:  110nMpH: 7.5Assay Description:Inhibitors (initial concentration 10 or 60 μM, three-fold serial dilutions) were incubated with IRE1α* in cleavage buffer (20 mM HEPES at p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington

LigandPNGBDBM192720(KIRA analog, 2)
Affinity DataIC50:  120nMAssay Description:5′-Carboxyfluorescein (FAM)- and 3′-Black Hole Quencher (BHQ)-labeled XBP1 single stemloop mini-substrate (5′FAM-CUGAGUCCGCAGCACUCA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington

LigandPNGBDBM192721(KIRA analog, 3)
Affinity DataIC50:  140nMpH: 7.5Assay Description:Inhibitors (initial concentration 10 or 60 μM, three-fold serial dilutions) were incubated with IRE1α* in cleavage buffer (20 mM HEPES at p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target1-acyl-sn-glycerol-3-phosphate acyltransferase beta(Homo sapiens (Human))
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50172949(6-(5-Chloro-2-ethoxy-phenyl)-N-(4-chloro-phenyl)-[...)
Affinity DataIC50:  140nMAssay Description:Inhibition of human LPAAT-beta by cell-free colorimetric assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington

LigandPNGBDBM192734(KIRA analog, 16)
Affinity DataIC50:  140nMAssay Description:5′-Carboxyfluorescein (FAM)- and 3′-Black Hole Quencher (BHQ)-labeled XBP1 single stemloop mini-substrate (5′FAM-CUGAGUCCGCAGCACUCA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington

LigandPNGBDBM192739(KIRA analog, 21)
Affinity DataIC50:  170nMpH: 7.5Assay Description:Inhibitors (initial concentration 10 or 60 μM, three-fold serial dilutions) were incubated with IRE1α* in cleavage buffer (20 mM HEPES at p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington

LigandPNGBDBM192720(KIRA analog, 2)
Affinity DataIC50:  170nMpH: 7.5Assay Description:Inhibitors (initial concentration 10 or 60 μM, three-fold serial dilutions) were incubated with IRE1α* in cleavage buffer (20 mM HEPES at p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington

LigandPNGBDBM192722(KIRA analog, 4)
Affinity DataIC50:  180nMAssay Description:5′-Carboxyfluorescein (FAM)- and 3′-Black Hole Quencher (BHQ)-labeled XBP1 single stemloop mini-substrate (5′FAM-CUGAGUCCGCAGCACUCA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington

LigandPNGBDBM192738(KIRA analog, 20)
Affinity DataIC50:  190nMAssay Description:5′-Carboxyfluorescein (FAM)- and 3′-Black Hole Quencher (BHQ)-labeled XBP1 single stemloop mini-substrate (5′FAM-CUGAGUCCGCAGCACUCA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington

LigandPNGBDBM192730(KIRA analog, 12)
Affinity DataIC50:  190nMAssay Description:5′-Carboxyfluorescein (FAM)- and 3′-Black Hole Quencher (BHQ)-labeled XBP1 single stemloop mini-substrate (5′FAM-CUGAGUCCGCAGCACUCA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington

LigandPNGBDBM192731(KIRA analog, 13)
Affinity DataIC50:  220nMAssay Description:5′-Carboxyfluorescein (FAM)- and 3′-Black Hole Quencher (BHQ)-labeled XBP1 single stemloop mini-substrate (5′FAM-CUGAGUCCGCAGCACUCA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclic GMP-AMP synthase(Homo sapiens)
Monash University Malaysia

Curated by ChEMBL
LigandPNGBDBM50582696(CHEMBL5076595)
Affinity DataIC50:  240nMAssay Description:Inhibition of cGAS (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
Displayed 1 to 50 (of 134 total ) | Next | Last >>
Jump to: