Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 6nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 11nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 22nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 28nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 39nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 210nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 300nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 420nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 430nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 480nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 520nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT1AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 610nMAssay Description:Displacement of [3H]-5Carboxyamidotryptamine from human 5-HT7R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.09E+3nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 1.76E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 1.83E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT2AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.95E+3nMAssay Description:Displacement of [3H]-Raclopride from human dopamine D2 receptor expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 2.29E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT1AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 4.54E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT1AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 4.76E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT1AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 5.20E+3nMAssay Description:Displacement of [3H]-5Carboxyamidotryptamine from human 5-HT7R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 5.71E+3nMAssay Description:Displacement of [3H]-5Carboxyamidotryptamine from human 5-HT7R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 9.45E+3nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT1AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 1.20E+4nMAssay Description:Displacement of [3H]-5Carboxyamidotryptamine from human 5-HT7R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 1.25E+4nMAssay Description:Displacement of [3H]-Raclopride from human 5-HT1AR expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 1.68E+4nMAssay Description:Displacement of [3H]-5Carboxyamidotryptamine from human 5-HT7R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataKi: 3.87E+4nMAssay Description:Displacement of [3H]-5Carboxyamidotryptamine from human 5-HT7R expressed in HEK293 cells by radioligand binding assayMore data for this Ligand-Target Pair
Target1-acyl-sn-glycerol-3-phosphate acyltransferase beta(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataIC50: 8.40nMAssay Description:Inhibition of LPAAT-beta (unknown origin) expressed in Xenopus laevis oocytes incubated for 3 minsMore data for this Ligand-Target Pair
Target1-acyl-sn-glycerol-3-phosphate acyltransferase beta(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataIC50: 15nMAssay Description:Inhibition of LPAAT-beta (unknown origin) expressed in Xenopus laevis oocytes incubated for 3 minsMore data for this Ligand-Target Pair
TargetInosine-5'-monophosphate dehydrogenase 2(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataIC50: 54nMAssay Description:Inhibition of IMPDH2 (unknown origin)More data for this Ligand-Target Pair
Target1-acyl-sn-glycerol-3-phosphate acyltransferase beta(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataIC50: 60nMAssay Description:Inhibition of human LPAAT-beta by cell-free colorimetric assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington
University Of Washington
Affinity DataIC50: 65nMpH: 7.5Assay Description:Inhibitors (initial concentration 10 or 60 μM, three-fold serial dilutions) were incubated with IRE1α* in cleavage buffer (20 mM HEPES at p...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington
University Of Washington
Affinity DataIC50: 66nMpH: 7.5Assay Description:Inhibitors (initial concentration 10 or 60 μM, three-fold serial dilutions) were incubated with IRE1α* in cleavage buffer (20 mM HEPES at p...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington
University Of Washington
Affinity DataIC50: 90nMAssay Description:5′-Carboxyfluorescein (FAM)- and 3′-Black Hole Quencher (BHQ)-labeled XBP1 single stemloop mini-substrate (5′FAM-CUGAGUCCGCAGCACUCA...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington
University Of Washington
Affinity DataIC50: 110nMpH: 7.5Assay Description:Inhibitors (initial concentration 10 or 60 μM, three-fold serial dilutions) were incubated with IRE1α* in cleavage buffer (20 mM HEPES at p...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington
University Of Washington
Affinity DataIC50: 110nMpH: 7.5Assay Description:Inhibitors (initial concentration 10 or 60 μM, three-fold serial dilutions) were incubated with IRE1α* in cleavage buffer (20 mM HEPES at p...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington
University Of Washington
Affinity DataIC50: 120nMAssay Description:5′-Carboxyfluorescein (FAM)- and 3′-Black Hole Quencher (BHQ)-labeled XBP1 single stemloop mini-substrate (5′FAM-CUGAGUCCGCAGCACUCA...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington
University Of Washington
Affinity DataIC50: 140nMpH: 7.5Assay Description:Inhibitors (initial concentration 10 or 60 μM, three-fold serial dilutions) were incubated with IRE1α* in cleavage buffer (20 mM HEPES at p...More data for this Ligand-Target Pair
Target1-acyl-sn-glycerol-3-phosphate acyltransferase beta(Homo sapiens (Human))
Monash University Malaysia
Curated by ChEMBL
Monash University Malaysia
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Inhibition of human LPAAT-beta by cell-free colorimetric assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington
University Of Washington
Affinity DataIC50: 140nMAssay Description:5′-Carboxyfluorescein (FAM)- and 3′-Black Hole Quencher (BHQ)-labeled XBP1 single stemloop mini-substrate (5′FAM-CUGAGUCCGCAGCACUCA...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington
University Of Washington
Affinity DataIC50: 170nMpH: 7.5Assay Description:Inhibitors (initial concentration 10 or 60 μM, three-fold serial dilutions) were incubated with IRE1α* in cleavage buffer (20 mM HEPES at p...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington
University Of Washington
Affinity DataIC50: 170nMpH: 7.5Assay Description:Inhibitors (initial concentration 10 or 60 μM, three-fold serial dilutions) were incubated with IRE1α* in cleavage buffer (20 mM HEPES at p...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington
University Of Washington
Affinity DataIC50: 180nMAssay Description:5′-Carboxyfluorescein (FAM)- and 3′-Black Hole Quencher (BHQ)-labeled XBP1 single stemloop mini-substrate (5′FAM-CUGAGUCCGCAGCACUCA...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington
University Of Washington
Affinity DataIC50: 190nMAssay Description:5′-Carboxyfluorescein (FAM)- and 3′-Black Hole Quencher (BHQ)-labeled XBP1 single stemloop mini-substrate (5′FAM-CUGAGUCCGCAGCACUCA...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington
University Of Washington
Affinity DataIC50: 190nMAssay Description:5′-Carboxyfluorescein (FAM)- and 3′-Black Hole Quencher (BHQ)-labeled XBP1 single stemloop mini-substrate (5′FAM-CUGAGUCCGCAGCACUCA...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase/endoribonuclease IRE1 [547-977](Homo sapiens (Human))
University Of Washington
University Of Washington
Affinity DataIC50: 220nMAssay Description:5′-Carboxyfluorescein (FAM)- and 3′-Black Hole Quencher (BHQ)-labeled XBP1 single stemloop mini-substrate (5′FAM-CUGAGUCCGCAGCACUCA...More data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibition of cGAS (unknown origin)More data for this Ligand-Target Pair