Compile Data Set for Download or QSAR
maximum 50k data
Found 50 with Last Name = 'harries' and Initial = 'mh'
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331382(CHEMBL1289063 | N-((3R,4R)-4-(4-(6-fluoropyridin-3...)
Affinity DataIC50:  80nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331371(CHEMBL1290275 | N-((3R,4R)-4-(4'-cyanobiphenyl-4-y...)
Affinity DataIC50:  400nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331373(CHEMBL1290391 | N-((3R,4R)-4-(4'-cyanobiphenyl-4-y...)
Affinity DataIC50:  800nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331381(CHEMBL1289062 | N-((3R,4R)-4-(4-(6-fluoropyridin-3...)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331369(CHEMBL1290165 | N-((3R,4R)-4-(3'-(methylsulfonamid...)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331370(CHEMBL1290166 | N-((3R,4R)-4-(4'-cyanobiphenyl-4-y...)
Affinity DataIC50:  2.00E+3nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331367(CHEMBL1290058 | N-((3R,4R)-1-ethyl-4-(3'-(methylsu...)
Affinity DataIC50:  2.50E+3nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331377(CHEMBL1290612 | N-((3R,4R)-1-methyl-4-(3'-(trifluo...)
Affinity DataIC50:  4.00E+3nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331384(CHEMBL1289180 | N-((3R,4R)-1-methyl-4-(4-(thiophen...)
Affinity DataIC50:  4.00E+3nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331368(CHEMBL1290059 | N-((3R,4R)-1-isopropyl-4-(3'-(meth...)
Affinity DataIC50:  6.30E+3nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331380(CHEMBL1290732 | N-((3R,4R)-4-(4-(2-fluoropyridin-3...)
Affinity DataIC50:  6.30E+3nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331376(CHEMBL1290504 | N-((3R,4R)-4-(3'-acetylbiphenyl-4-...)
Affinity DataIC50:  7.90E+3nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331387(CHEMBL1289294 | N-((3S,4S)-4-(4-(6-fluoropyridin-3...)
Affinity DataIC50:  1.26E+4nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331375(CHEMBL1290503 | N-(4'-((3R,4R)-1-methyl-4-(1-methy...)
Affinity DataIC50:  1.26E+4nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331385(CHEMBL1289181 | N-((3S,4S)-4-(4'-cyanobiphenyl-4-y...)
Affinity DataIC50:  1.26E+4nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331379(CHEMBL1290731 | N-((3R,4R)-1-methyl-4-(4-(pyridin-...)
Affinity DataIC50:  3.16E+4nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331366(CHEMBL1289960 | N-((3R,4R)-1-methyl-4-(3'-(methyls...)
Affinity DataIC50:  3.16E+4nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331386(CHEMBL1289293 | N-((3S,4S)-4-(3'-acetylbiphenyl-4-...)
Affinity DataIC50: >6.30E+4nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331390(CHEMBL1289410 | N-((3S,4S)-4-(4-(thiophen-2-yl)phe...)
Affinity DataIC50: >6.30E+4nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331391(CHEMBL1289523 | N-((3S,4S)-4-(4-(thiophen-3-yl)phe...)
Affinity DataIC50: >6.30E+4nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331383(CHEMBL1289179 | N-((3R,4R)-1-methyl-4-(4-(thiophen...)
Affinity DataIC50: >6.30E+4nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331389(CHEMBL1289409 | N-((3S,4S)-4-(4-(5-fluoropyridin-2...)
Affinity DataIC50: >6.30E+4nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331374(CHEMBL1290392 | N-((3R,4R)-1-methyl-4-(3'-(methyls...)
Affinity DataIC50: >6.30E+4nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331388(CHEMBL1289408 | N-((3S,4S)-4-(4-(5-fluoropyridin-3...)
Affinity DataIC50: >6.30E+4nMAssay Description:Displacement of [3H]-dofetilide from human hERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331377(CHEMBL1290612 | N-((3R,4R)-1-methyl-4-(3'-(trifluo...)
Affinity DataEC50:  7.94E+4nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331376(CHEMBL1290504 | N-((3R,4R)-4-(3'-acetylbiphenyl-4-...)
Affinity DataEC50:  6.30E+3nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331375(CHEMBL1290503 | N-(4'-((3R,4R)-1-methyl-4-(1-methy...)
Affinity DataEC50:  4.00E+3nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331374(CHEMBL1290392 | N-((3R,4R)-1-methyl-4-(3'-(methyls...)
Affinity DataEC50:  5.00E+3nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331373(CHEMBL1290391 | N-((3R,4R)-4-(4'-cyanobiphenyl-4-y...)
Affinity DataEC50:  6.20E+3nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331372(CHEMBL1290276 | N-((3R,4R)-4-(4'-cyanobiphenyl-4-y...)
Affinity DataEC50:  2.00E+4nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331371(CHEMBL1290275 | N-((3R,4R)-4-(4'-cyanobiphenyl-4-y...)
Affinity DataEC50:  7.90E+3nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331370(CHEMBL1290166 | N-((3R,4R)-4-(4'-cyanobiphenyl-4-y...)
Affinity DataEC50:  5.00E+3nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331369(CHEMBL1290165 | N-((3R,4R)-4-(3'-(methylsulfonamid...)
Affinity DataEC50:  5.00E+3nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331368(CHEMBL1290059 | N-((3R,4R)-1-isopropyl-4-(3'-(meth...)
Affinity DataEC50:  6.30E+3nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331367(CHEMBL1290058 | N-((3R,4R)-1-ethyl-4-(3'-(methylsu...)
Affinity DataEC50:  1.60E+3nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331366(CHEMBL1289960 | N-((3R,4R)-1-methyl-4-(3'-(methyls...)
Affinity DataEC50:  300nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331391(CHEMBL1289523 | N-((3S,4S)-4-(4-(thiophen-3-yl)phe...)
Affinity DataEC50:  400nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331390(CHEMBL1289410 | N-((3S,4S)-4-(4-(thiophen-2-yl)phe...)
Affinity DataEC50:  300nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331389(CHEMBL1289409 | N-((3S,4S)-4-(4-(5-fluoropyridin-2...)
Affinity DataEC50:  300nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331388(CHEMBL1289408 | N-((3S,4S)-4-(4-(5-fluoropyridin-3...)
Affinity DataEC50:  300nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331387(CHEMBL1289294 | N-((3S,4S)-4-(4-(6-fluoropyridin-3...)
Affinity DataEC50:  300nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331386(CHEMBL1289293 | N-((3S,4S)-4-(3'-acetylbiphenyl-4-...)
Affinity DataEC50:  100nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331385(CHEMBL1289181 | N-((3S,4S)-4-(4'-cyanobiphenyl-4-y...)
Affinity DataEC50:  500nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331384(CHEMBL1289180 | N-((3R,4R)-1-methyl-4-(4-(thiophen...)
Affinity DataEC50:  3.20E+3nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331383(CHEMBL1289179 | N-((3R,4R)-1-methyl-4-(4-(thiophen...)
Affinity DataEC50:  2.00E+4nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331382(CHEMBL1289063 | N-((3R,4R)-4-(4-(6-fluoropyridin-3...)
Affinity DataEC50:  4.00E+3nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331381(CHEMBL1289062 | N-((3R,4R)-4-(4-(6-fluoropyridin-3...)
Affinity DataEC50:  5.00E+3nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331378(CHEMBL1290613 | N-((3R,4R)-4-(2'-fluorobiphenyl-4-...)
Affinity DataEC50:  2.50E+3nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331379(CHEMBL1290731 | N-((3R,4R)-1-methyl-4-(4-(pyridin-...)
Affinity DataEC50:  4.00E+3nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutamate receptor 2(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50331380(CHEMBL1290732 | N-((3R,4R)-4-(4-(2-fluoropyridin-3...)
Affinity DataEC50:  2.50E+3nMAssay Description:Positive modulation of human GluA2 flip receptor by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed