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Found 56 with Last Name = 'hauck newman' and Initial = 'a'
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM86701(3-(bis(4-fluorophenyl)methoxy)-8-methyl-8-aza-bicy...)
Affinity DataKi:  4.10nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50147595((S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50147594((S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM86701(3-(bis(4-fluorophenyl)methoxy)-8-methyl-8-aza-bicy...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]pirenzepine from muscarinic acetylcholine receptor M1 of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50147593((R)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]pirenzepine from muscarinic acetylcholine receptor M1 of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50147593((R)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50147595((S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]pirenzepine from muscarinic acetylcholine receptor M1 of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50147594((S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  48nMAssay Description:Displacement of [3H]pirenzepine from muscarinic acetylcholine receptor M1 of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451947(CHEMBL2112508)
Affinity DataKi:  57nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM22418(Cocaine | Cocaine (-) | methyl (1R,2R,3S,5S)-3-(be...)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451943(CHEMBL2112509)
Affinity DataKi:  75nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451945(CHEMBL2112515)
Affinity DataKi:  81nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451942(CHEMBL2112513)
Affinity DataKi:  107nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451940(CHEMBL2112511)
Affinity DataKi:  119nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451943(CHEMBL2112509)
Affinity DataKi:  142nMAssay Description:Displacement of [3H]pirenzepine from muscarinic acetylcholine receptor M1 of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451941(CHEMBL2112512)
Affinity DataKi:  148nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451939(CHEMBL2112510)
Affinity DataKi:  151nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451944(CHEMBL2112514)
Affinity DataKi:  171nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451946(CHEMBL2112516)
Affinity DataKi:  175nMAssay Description:Displacement of [3H]WIN-35428 from dopamine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM22418(Cocaine | Cocaine (-) | methyl (1R,2R,3S,5S)-3-(be...)
Affinity DataKi:  293nMAssay Description:Displacement of [3H]-citalopram from serotonin transporter of rat brain membraneMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451947(CHEMBL2112508)
Affinity DataKi:  432nMAssay Description:Displacement of [3H]pirenzepine from muscarinic acetylcholine receptor M1 of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451942(CHEMBL2112513)
Affinity DataKi:  552nMAssay Description:Displacement of [3H]pirenzepine from muscarinic acetylcholine receptor M1 of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451945(CHEMBL2112515)
Affinity DataKi:  617nMAssay Description:Displacement of [3H]pirenzepine from muscarinic acetylcholine receptor M1 of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451941(CHEMBL2112512)
Affinity DataKi:  723nMAssay Description:Displacement of [3H]pirenzepine from muscarinic acetylcholine receptor M1 of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451939(CHEMBL2112510)
Affinity DataKi:  784nMAssay Description:Displacement of [3H]pirenzepine from muscarinic acetylcholine receptor M1 of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM86701(3-(bis(4-fluorophenyl)methoxy)-8-methyl-8-aza-bicy...)
Affinity DataKi:  844nMAssay Description:Displacement of [3H]-nisoxatine from norepinephrine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50147594((S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]-nisoxatine from norepinephrine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451942(CHEMBL2112513)
Affinity DataKi:  1.37E+3nMAssay Description:Displacement of [3H]-nisoxatine from norepinephrine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50147595((S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  1.38E+3nMAssay Description:Displacement of [3H]-nisoxatine from norepinephrine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451940(CHEMBL2112511)
Affinity DataKi:  2.27E+3nMAssay Description:Displacement of [3H]pirenzepine from muscarinic acetylcholine receptor M1 of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451946(CHEMBL2112516)
Affinity DataKi:  3.17E+3nMAssay Description:Displacement of [3H]-nisoxatine from norepinephrine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM86701(3-(bis(4-fluorophenyl)methoxy)-8-methyl-8-aza-bicy...)
Affinity DataKi:  3.26E+3nMAssay Description:Displacement of [3H]-citalopram from serotonin transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM22418(Cocaine | Cocaine (-) | methyl (1R,2R,3S,5S)-3-(be...)
Affinity DataKi:  3.30E+3nMAssay Description:Displacement of [3H]-nisoxatine from norepinephrine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451944(CHEMBL2112514)
Affinity DataKi:  3.48E+3nMAssay Description:Displacement of [3H]pirenzepine from muscarinic acetylcholine receptor M1 of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451943(CHEMBL2112509)
Affinity DataKi:  3.72E+3nMAssay Description:Displacement of [3H]-nisoxatine from norepinephrine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451942(CHEMBL2112513)
Affinity DataKi:  3.73E+3nMAssay Description:Displacement of [3H]-citalopram from serotonin transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451946(CHEMBL2112516)
Affinity DataKi:  4.44E+3nMAssay Description:Displacement of [3H]-citalopram from serotonin transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451944(CHEMBL2112514)
Affinity DataKi:  5.69E+3nMAssay Description:Displacement of [3H]-nisoxatine from norepinephrine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451940(CHEMBL2112511)
Affinity DataKi:  5.85E+3nMAssay Description:Displacement of [3H]-citalopram from serotonin transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451940(CHEMBL2112511)
Affinity DataKi:  6.21E+3nMAssay Description:Displacement of [3H]-nisoxatine from norepinephrine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50147593((R)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  6.39E+3nMAssay Description:Displacement of [3H]-nisoxatine from norepinephrine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451941(CHEMBL2112512)
Affinity DataKi:  6.61E+3nMAssay Description:Displacement of [3H]-nisoxatine from norepinephrine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451945(CHEMBL2112515)
Affinity DataKi:  6.88E+3nMAssay Description:Displacement of [3H]-nisoxatine from norepinephrine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451947(CHEMBL2112508)
Affinity DataKi:  6.91E+3nMAssay Description:Displacement of [3H]-nisoxatine from norepinephrine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451944(CHEMBL2112514)
Affinity DataKi:  7.96E+3nMAssay Description:Displacement of [3H]-citalopram from serotonin transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451941(CHEMBL2112512)
Affinity DataKi:  7.96E+3nMAssay Description:Displacement of [3H]-citalopram from serotonin transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50147595((S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  8.29E+3nMAssay Description:Displacement of [3H]-citalopram from serotonin transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451946(CHEMBL2112516)
Affinity DataKi:  8.43E+3nMAssay Description:Displacement of [3H]pirenzepine from muscarinic acetylcholine receptor M1 of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50147594((S)-3-[Bis-(4-fluoro-phenyl)-methoxy]-8-methyl-8-a...)
Affinity DataKi:  9.09E+3nMAssay Description:Displacement of [3H]citalopram from serotonin transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus)
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL
LigandPNGBDBM50451939(CHEMBL2112510)
Affinity DataKi:  1.02E+4nMAssay Description:Displacement of [3H]-nisoxatine from norepinephrine transporter of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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