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Found 10 with Last Name = 'hayakawa' and Initial = 'h'
TargetUDP-glucuronosyltransferase 1A1(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50044561(CHEMBL3222137)
Affinity DataKi:  1.54E+3nMAssay Description:Substrate inhibition of human UGT1A1-mediated T-5224 acyl O-glucuronide formation after 10 to 60 mins in presence of UDP-glucuronic acid by HPLC meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-glucuronosyltransferase 1A3(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50044561(CHEMBL3222137)
Affinity DataKi:  2.55E+3nMAssay Description:Substrate inhibition of human UGT1A3-mediated T-5224 hydroxyl O-glucuronide formation after 10 to 60 mins in presence of UDP-glucuronic acid by HPLC ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-glucuronosyltransferase 1A8(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50044561(CHEMBL3222137)
Affinity DataKi:  3.64E+3nMAssay Description:Substrate inhibition of human UGT1A8-mediated T-5224 hydroxyl O-glucuronide formation after 10 to 60 mins in presence of UDP-glucuronic acid by HPLC ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-glucuronosyltransferase 1A1(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50044561(CHEMBL3222137)
Affinity DataKi:  4.67E+3nMAssay Description:Substrate inhibition of human UGT1A1-mediated T-5224 hydroxyl O-glucuronide formation after 10 to 60 mins in presence of UDP-glucuronic acid by HPLC ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUDP-glucuronosyltransferase 1A3(Homo sapiens (Human))
Toyama Chemical

Curated by ChEMBL
LigandPNGBDBM50044561(CHEMBL3222137)
Affinity DataKi:  1.35E+4nMAssay Description:Substrate inhibition of human UGT1A3-mediated T-5224 acyl O-glucuronide formation after 10 to 60 mins in presence of UDP-glucuronic acid by HPLC meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Showa University

Curated by ChEMBL
LigandPNGBDBM50016534(1-(4-azido-5-{[(1,2,3,3-tetrahydroxy-1,2,3-trioxid...)
Affinity DataIC50:  34nMAssay Description:Inhibitory effect of the compound on HIV-1 reverse transcriptase activity using poly(rA)-oligo(dT) template primerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Showa University

Curated by ChEMBL
LigandPNGBDBM50004152((HEPT) 1-(2-Hydroxy-ethoxymethyl)-5-methyl-6-pheny...)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibitory effect of the compound on HIV-1 reverse transcriptase activity using poly(rC)-oligo(dG) template primerMore data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Showa University

Curated by ChEMBL
LigandPNGBDBM50016535(5-methyl-6-(phenylthio)-1-({2-[(1,2,3,3-tetrahydro...)
Affinity DataIC50:  2.80E+5nMAssay Description:Inhibitory effect of the compound on HIV-1 reverse transcriptase activity using poly(rA)-oligo(dT) template primerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Showa University

Curated by ChEMBL
LigandPNGBDBM50016535(5-methyl-6-(phenylthio)-1-({2-[(1,2,3,3-tetrahydro...)
Affinity DataIC50:  2.80E+5nMAssay Description:Inhibitory effect of the compound on HIV-1 reverse transcriptase activity using poly(rC)-oligo(dG) template primerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Showa University

Curated by ChEMBL
LigandPNGBDBM50004152((HEPT) 1-(2-Hydroxy-ethoxymethyl)-5-methyl-6-pheny...)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibitory effect of the compound on HIV-1 reverse transcriptase activity using poly(rA)-oligo(dT) template primerMore data for this Ligand-Target Pair