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Found 145 with Last Name = 'hernández' and Initial = 'e'
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163035(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Instituto PolitéCnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM17292((1S,10R,11S,14S,15S)-15-methyltetracyclo[8.7.0.0^{...)
Affinity DataKi:  0.160nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34143(CHEMBL175835 | E-6837)
Affinity DataKi:  0.200nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163094(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataKi:  0.300nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163067(Biphenyl-4-sulfonic acid [3-(2-dimethylamino-ethyl...)
Affinity DataKi:  0.400nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34145(pyrrolidinylindole, (R)-5b)
Affinity DataKi:  0.400nM ΔG°:  -55.8kJ/mole EC50:  4.5nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163061(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34143(CHEMBL175835 | E-6837)
Affinity DataKi:  0.700nM ΔG°:  -54.4kJ/mole EC50:  0.290nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM28583(5-chloro-N-[4-methoxy-3-(piperazin-1-yl)phenyl]-3-...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163053(CHEMBL368390 | Naphthalene-1-sulfonic acid [3-(2-d...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163077(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataKi:  1nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34147(CHEMBL425196 | pyrrolidinylindole, 6)
Affinity DataKi:  1nM ΔG°:  -53.4kJ/mole EC50:  53.3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34144((R)-5a | WAY-466)
Affinity DataKi:  1nM ΔG°:  -53.4kJ/mole EC50:  0.400nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163071(Biphenyl-4-sulfonic acid [3-(2-diethylamino-ethyl)...)
Affinity DataKi:  1nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163052(6-Chloro-imidazo[2,1-b]thiazole-5-sulfonic acid [1...)
Affinity DataKi:  1.90nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM21358(2-[1-({6-chloroimidazo[2,1-b][1,3]thiazole-5-}sulf...)
Affinity DataKi:  2nM ΔG°:  -51.6kJ/mole EC50:  6.5nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34141(CHEMBL76237 | MS-245)
Affinity DataKi:  2nM ΔG°:  -51.6kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34148(CHEMBL371292 | piperidinylindole, 7)
Affinity DataKi:  2nM ΔG°:  -51.6kJ/mole EC50:  24nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34152(CHEMBL362628 | E-6801)
Affinity DataKi:  2.20nM ΔG°:  -51.4kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34152(CHEMBL362628 | E-6801)
Affinity DataKi:  2.20nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34156(indenylsulfonamide, 28)
Affinity DataKi:  3nM ΔG°:  -50.6kJ/mole IC50:  1.60E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34149(CHEMBL94422 | N-benzenesulfonylgramine antagonist,...)
Affinity DataKi:  3nM ΔG°:  -50.6kJ/mole EC50:  880nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163102(5-Chloro-naphthalene-1-sulfonic acid [3-(2-diethyl...)
Affinity DataKi:  3.30nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163097(CHEMBL180425 | Naphthalene-1-sulfonic acid [3-(2-d...)
Affinity DataKi:  3.5nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163080(CHEMBL176292 | Naphthalene-2-sulfonic acid [3-(2-d...)
Affinity DataKi:  3.90nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163059(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataKi:  4nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163086(CHEMBL427134 | Naphthalene-2-sulfonic acid [3-(2-p...)
Affinity DataKi:  4.30nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163098(CHEMBL367867 | Naphthalene-1-sulfonic acid [3-(2-p...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34153(CHEMBL476006 | indenylsulfonamide, 14)
Affinity DataKi:  4.5nM ΔG°:  -49.6kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163040(CHEMBL361230 | Naphthalene-1-sulfonic acid [3-(1-m...)
Affinity DataKi:  4.70nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163055(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163034(CHEMBL175471 | Naphthalene-2-sulfonic acid [3-(2-d...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163034(CHEMBL175471 | Naphthalene-2-sulfonic acid [3-(2-d...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163073(Biphenyl-4-sulfonic acid [3-(1-methyl-piperidin-4-...)
Affinity DataKi:  6.80nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163064(CHEMBL175529 | Naphthalene-1-sulfonic acid [3-(2-d...)
Affinity DataKi:  7.20nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163038(3,5-Dichloro-N-[3-(2-diethylamino-ethyl)-1H-indol-...)
Affinity DataKi:  9.30nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163079(5-Chloro-naphthalene-1-sulfonic acid [3-(1-methyl-...)
Affinity DataKi:  9.60nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163091(6-Chloro-imidazo[2,1-b]thiazole-5-sulfonic acid [1...)
Affinity DataKi:  9.80nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34146(pyrrolidinylindole, (S)-5b)
Affinity DataKi:  10nM ΔG°:  -47.5kJ/mole EC50:  21.6nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34154(CHEMBL515307 | indenylsulfonamide, 15)
Affinity DataKi:  10nM ΔG°:  -47.5kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34151(CHEMBL372109 | N-arenesulfonylindole antagonist, 1...)
Affinity DataKi:  10nM ΔG°:  -47.5kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34150(4-(3-methyl-1H-indole-1-sulfonyl)aniline, 8 | CHEM...)
Affinity DataKi:  12nM ΔG°:  -47.0kJ/mole EC50:  320nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Instituto PolitéCnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM50323914(CHEMBL1213786 | Tamoxifen butyl bromide)
Affinity DataKi:  13.0nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Instituto PolitéCnico Nacional 2508

Curated by ChEMBL
LigandPNGBDBM50323912(CHEMBL1213784 | Tamoxifen ethyl bromide)
Affinity DataKi:  13.7nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50090524(4-Amino-N-(2,6-bis-methylamino-pyridin-4-yl)-benze...)
Affinity DataKi:  14.8nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163060(CHEMBL176117 | Naphthalene-2-sulfonic acid [1-(2-d...)
Affinity DataKi:  14.9nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163090(5-Chloro-3-methyl-benzo[b]thiophene-2-sulfonic aci...)
Affinity DataKi:  15.1nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34142(2-ethyl-5-methoxy-N,N-dimethyltryptamine | CHEMBL2...)
Affinity DataKi:  16nM ΔG°:  -46.3kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM34158(indenylsulfonamide, 30)
Affinity DataKi:  18nM ΔG°:  -46.0kJ/molepH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed using membranes from HEK-293 transfected with human 5-HT6 receptor. In these membranes the receptor concent...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Laboratorios Dr. Esteve

Curated by ChEMBL
LigandPNGBDBM50163099(2-[5-(6-Chloro-imidazo[2,1-b]thiazole-5-sulfonylam...)
Affinity DataKi:  18.4nMAssay Description:Inhibition of [3H]-LSD binding to human 5-hydroxytryptamine 6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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