Compile Data Set for Download or QSAR
maximum 50k data
Found 12 with Last Name = 'ichikawa' and Initial = 'a'
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Waseda University

Curated by ChEMBL
LigandPNGBDBM50004907(2-Amino-3-(4-phosphonomethyl-phenyl)-propionic aci...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibitory activity against Syk C-terminal SH2 domain in in-silico screeningMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Waseda University

Curated by ChEMBL
LigandPNGBDBM50107899(2-[4-(4-{2-[(5-Carboxy-pentyl)-(3-cyclohexyl-propy...)
Affinity DataIC50:  3.80E+4nMAssay Description:Inhibitory activity against Syk C-terminal SH2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Waseda University

Curated by ChEMBL
LigandPNGBDBM50107897(2-[4-(4-{2-[(5-Carboxy-pentyl)-(3-cyclohexyl-propy...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibitory activity against Syk C-terminal SH2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Waseda University

Curated by ChEMBL
LigandPNGBDBM50107901(2-[4-(4-{2-[(5-Carboxy-pentyl)-(3-cyclohexyl-propy...)
Affinity DataIC50:  4.10E+4nMAssay Description:Inhibitory activity against Syk C-terminal SH2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Waseda University

Curated by ChEMBL
LigandPNGBDBM50107900(2-[4-(4-{2-[(5-Carboxy-pentyl)-(5-methyl-hexyl)-su...)
Affinity DataIC50:  6.30E+4nMAssay Description:Inhibitory activity against Syk C-terminal SH2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Waseda University

Curated by ChEMBL
LigandPNGBDBM50107902(2-[4-(4-{2-[(5-Carboxy-pentyl)-(5-methyl-hexyl)-su...)
Affinity DataIC50:  6.90E+4nMAssay Description:Inhibitory activity against Syk C-terminal SH2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Waseda University

Curated by ChEMBL
LigandPNGBDBM50107898(2-[4-(4-{2-[(5-Carboxy-pentyl)-(5-methyl-hexyl)-su...)
Affinity DataIC50:  7.10E+4nMAssay Description:Inhibitory activity against Syk C-terminal SH2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Waseda University

Curated by ChEMBL
LigandPNGBDBM50107895(2-(4-{4-[2-(5-Carboxy-pentylsulfamoyl)-vinyl]-phen...)
Affinity DataIC50:  3.50E+5nMAssay Description:Inhibitory activity against Syk C-terminal SH2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Waseda University

Curated by ChEMBL
LigandPNGBDBM50107903(2-Cyclohexyl-malonic acid | CHEMBL142870)
Affinity DataIC50:  5.90E+6nMAssay Description:Inhibitory activity against Syk C-terminal SH2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Waseda University

Curated by ChEMBL
LigandPNGBDBM50107894(2-Cyclooct-4-enyl-malonic acid | CHEMBL357125)
Affinity DataIC50:  7.70E+6nMAssay Description:Inhibitory activity against Syk C-terminal SH2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Waseda University

Curated by ChEMBL
LigandPNGBDBM50107896(6-(2-Phenyl-ethenesulfonylamino)-hexanoic acid | C...)
Affinity DataIC50:  8.00E+6nMAssay Description:Inhibitory activity against Syk C-terminal SH2 (at 10 mM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase SYK(Homo sapiens (Human))
Waseda University

Curated by ChEMBL
LigandPNGBDBM14676(2-phenylpropanedioic acid | CHEMBL78794 | Fragment...)
Affinity DataIC50:  1.20E+7nMAssay Description:Inhibitory activity against Syk C-terminal SH2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed