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Found 89 with Last Name = 'ingkaninan' and Initial = 'k'
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden University

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataKi:  1.55E+3nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in rat brain cortex membrane in presence of 0.5 mM GTPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden University

Curated by ChEMBL
LigandPNGBDBM7459(2-(3,4-dihydroxyphenyl)-5,7-dihydroxy-4H-chromen-4...)
Affinity DataKi:  1.66E+3nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM10847(1,3-dimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-dion...)
Affinity DataKi:  8.50E+3nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAdenosine receptor A1(Homo sapiens (Human))
Leiden University

Curated by ChEMBL
LigandPNGBDBM10849(1,3,7-trimethyl-2,3,6,7-tetrahydro-1H-purine-2,6-d...)
Affinity DataKi:  2.90E+4nMAssay Description:Binding affinity to adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50259668(4-(cis)-acetyl-3,6,8-trihydroxy-3-methyldihydronap...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50244182(5-acetonyl-7-hydroxy-2-methyl chromone | 5-acetony...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50259665(5-acetonyl-7-hydroxy-2-hydroxymethylchromone | CHE...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Leiden University

Curated by ChEMBL
LigandPNGBDBM50259667(4-(trans)-acetyl-3,6,8-trihydroxy-3-methyldihydron...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in rat brain cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
King Mongkut'S Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM14390(5-[2-ethoxy-5-(4-methyl-1-piperazinylsulfonyl)phen...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of human PDE5 using [3H]cGMP as substrate incubated for 10 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM14390(5-[2-ethoxy-5-(4-methyl-1-piperazinylsulfonyl)phen...)
Affinity DataIC50:  2nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
King Mongkut'S Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50033312(Benzyl-(6-chloro-2-imidazol-1-yl-quinazolin-4-yl)-...)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of human platelet PDE5More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
King Mongkut'S Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50518237(CHEMBL4552529)
Affinity DataIC50:  3.90nMAssay Description:Inhibition of PDE5 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Naresuan University

Curated by ChEMBL
LigandPNGBDBM50380808(CHEMBL2018162)
Affinity DataIC50:  71nMAssay Description:Inhibition of AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518228(CHEMBL4445920)
Affinity DataIC50:  72nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518224(CHEMBL4570769)
Affinity DataIC50:  89nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Mahidol University

Curated by ChEMBL
LigandPNGBDBM50377954(CHEMBL557422)
Affinity DataIC50:  91nMAssay Description:Inhibition of Torpedo californica AchE activity by Ellman's assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
King Mongkut'S Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50518228(CHEMBL4445920)
Affinity DataIC50:  100nMAssay Description:Inhibition of human PDE5 using [3H]cGMP as substrate incubated for 10 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518223(CHEMBL4529354)
Affinity DataIC50:  116nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
King Mongkut'S Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50602260(CHEMBL5175706)
Affinity DataIC50:  150nMAssay Description:Inhibition of human PDE5 using [3H]cGMP as substrate incubated for 10 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518225(CHEMBL4434898)
Affinity DataIC50:  177nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518217(CHEMBL4544782)
Affinity DataIC50:  218nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
King Mongkut'S Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50602263(CHEMBL5178863)
Affinity DataIC50:  220nMAssay Description:Inhibition of human PDE5 using [3H]cGMP as substrate incubated for 10 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518232(CHEMBL4460740)
Affinity DataIC50:  224nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Naresuan University

Curated by ChEMBL
LigandPNGBDBM50380807(CHEMBL376478)
Affinity DataIC50:  227nMAssay Description:Inhibition of AChE by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518220(CHEMBL4540726)
Affinity DataIC50:  284nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
King Mongkut'S Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50602240(CHEMBL5194921)
Affinity DataIC50:  290nMAssay Description:Inhibition of human PDE5 using [3H]cGMP as substrate incubated for 10 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518234(CHEMBL4516390)
Affinity DataIC50:  290nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Naresuan University

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  300nMAssay Description:Inhibition of human AChE by Ellman's methodMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518227(CHEMBL4452377)
Affinity DataIC50:  350nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
King Mongkut'S Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50602247(CHEMBL5187496)
Affinity DataIC50:  360nMAssay Description:Inhibition of human PDE5 using [3H]cGMP as substrate incubated for 10 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
King Mongkut'S Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50602245(CHEMBL5194783)
Affinity DataIC50:  410nMAssay Description:Inhibition of human PDE5 using [3H]cGMP as substrate incubated for 10 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
King Mongkut'S Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50602246(CHEMBL5184989)
Affinity DataIC50:  430nMAssay Description:Inhibition of human PDE5 using [3H]cGMP as substrate incubated for 10 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518233(CHEMBL4526365)
Affinity DataIC50:  443nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
King Mongkut'S Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50602243(CHEMBL5203939)
Affinity DataIC50:  490nMAssay Description:Inhibition of human PDE5 using [3H]cGMP as substrate incubated for 10 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
King Mongkut'S Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50602241(CHEMBL5186856)
Affinity DataIC50:  500nMAssay Description:Inhibition of human PDE5 using [3H]cGMP as substrate incubated for 10 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518226(CHEMBL4534674)
Affinity DataIC50:  514nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
King Mongkut'S Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50602242(CHEMBL5195499)
Affinity DataIC50:  520nMAssay Description:Inhibition of human PDE5 using [3H]cGMP as substrate incubated for 10 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518230(CHEMBL4453311)
Affinity DataIC50:  525nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518221(CHEMBL4450878)
Affinity DataIC50:  555nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Tetronarce californica (Pacific electric ray) (Tor...)
Mahidol University

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  590nMAssay Description:Inhibition of Torpedo californica AchE activity by Ellman's assayMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
Naresuan University

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  590nMAssay Description:Inhibition of AChE activityMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
Naresuan University

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  600nMAssay Description:Inhibition of electric eel AChE using acetylcholine iodide as substrate measured every 5 sec for 2 mins by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
King Mongkut'S Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50602244(CHEMBL5191104)
Affinity DataIC50:  600nMAssay Description:Inhibition of human PDE5 using [3H]cGMP as substrate incubated for 10 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518218(CHEMBL4567109)
Affinity DataIC50:  775nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518229(CHEMBL4558761)
Affinity DataIC50:  946nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Homo sapiens (Human))
Naresuan University

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataIC50:  980nMAssay Description:Inhibition of AChE (unknown origin) by microplate assayMore data for this Ligand-Target Pair
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
King Mongkut'S Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM50602259(CHEMBL5200202)
Affinity DataIC50:  1.03E+3nMAssay Description:Inhibition of human PDE5 using [3H]cGMP as substrate incubated for 10 mins by liquid scintillation counter analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518236(CHEMBL4469064)
Affinity DataIC50:  1.26E+3nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518231(CHEMBL597248 | GNF-Pf-4180 | MMV006169)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetcGMP-specific 3',5'-cyclic phosphodiesterase(Rattus norvegicus)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50518235(CHEMBL4525521)
Affinity DataIC50:  1.44E+3nMAssay Description:Inhibition of rat lung PDE5 using [3H]cGMP as substrate measured after 10 mins by scintillation counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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