TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Affinity DataKi: 0.0600nMAssay Description:Inhibition of human recombinant matrix metalloprotease 9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Affinity DataKi: 0.0600nMAssay Description:Inhibition of recombinant human matrix metalloproteinase-9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Affinity DataKi: 0.0800nMAssay Description:Inhibitory activity against matrix metalloprotease-9 (MMP-9)(gelatinase-B).More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Affinity DataKi: 0.0970nMAssay Description:Inhibition of human recombinant matrix metalloprotease 9More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Affinity DataKi: 0.100nMAssay Description:Inhibitory activity against matrix metalloprotease-9 (MMP-9)(gelatinase-B).More data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Affinity DataKi: 0.310nMAssay Description:Inhibitory activity against matrix metalloprotease-9 (MMP-9)(gelatinase-B).More data for this Ligand-Target Pair
Affinity DataKi: 0.350nMAssay Description:Inhibition of human recombinant matrix metalloprotease 3More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Hokkaido Collaboration Center
Curated by ChEMBL
Hokkaido Collaboration Center
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Inhibition of recombinant human TNF-alpha converting enzyme (TACE)More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Hokkaido Collaboration Center
Curated by ChEMBL
Hokkaido Collaboration Center
Curated by ChEMBL
Affinity DataKi: 0.400nMAssay Description:Inhibition of recombinant human tumor necrosis factor-alpha converting enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Inhibition of recombinant human matrix metalloproteinase-3More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Inhibitory activity against matrix metalloprotease-3 (MMP-3)(stromelysin-1).More data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Inhibition of human recombinant matrix metalloprotease 3More data for this Ligand-Target Pair
Affinity DataKi: 0.510nMAssay Description:Inhibition of recombinant human matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Hokkaido Collaboration Center
Curated by ChEMBL
Hokkaido Collaboration Center
Curated by ChEMBL
Affinity DataKi: 0.530nMAssay Description:Inhibition of human tumor necrosis factor alpha converting enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 0.530nMAssay Description:Inhibitory activity against matrix metalloprotease-3 (MMP-3)(stromelysin-1).More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Hokkaido Collaboration Center
Curated by ChEMBL
Hokkaido Collaboration Center
Curated by ChEMBL
Affinity DataKi: 0.530nMAssay Description:Inhibition of recombinant human TNF-alpha converting enzymeMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Hokkaido Collaboration Center
Curated by ChEMBL
Hokkaido Collaboration Center
Curated by ChEMBL
Affinity DataKi: 0.570nMAssay Description:Inhibition of recombinant human TNF-alpha converting enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 0.590nMAssay Description:Inhibition of aurora AMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibition of aurora AMore data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Affinity DataKi: 0.600nMAssay Description:Inhibitory activity against matrix metalloprotease-9 (MMP-9)(gelatinase-B).More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Hokkaido Collaboration Center
Curated by ChEMBL
Hokkaido Collaboration Center
Curated by ChEMBL
Affinity DataKi: 0.840nMAssay Description:Inhibition of recombinant human TNF-alpha converting enzymeMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.880nMAssay Description:Inhibition of [3H]-NMS binding to human muscarinic acetylcholine receptor M1 expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Affinity DataKi: 0.930nMAssay Description:Inhibition of recombinant human matrix metalloproteinase-9More data for this Ligand-Target Pair
Affinity DataKi: 0.970nMAssay Description:Inhibitory activity against matrix metalloprotease-1 (MMP-1)(recombinant human collagenase-1).More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.980nMAssay Description:Binding affinity against human Muscarinic acetylcholine receptor M1 in transfected CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1nMAssay Description:Binding affinity against human Muscarinic acetylcholine receptor M1 in transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of recombinant human matrix metalloproteinase-1More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of Recombinant human matrix metalloproteinase-1More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Binding affinity against human muscarinic acetylcholine receptor M3 in transfected CHO cellsMore data for this Ligand-Target Pair
TargetMatrix metalloproteinase-9(Homo sapiens (Human))
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Hokkaido Collaboration Center N-21
Curated by ChEMBL
Affinity DataKi: 1.13nMAssay Description:Inhibitory activity against matrix metalloprotease-9 (MMP-9)(gelatinase-B).More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Binding affinity against human muscarinic acetylcholine receptor M3 in transfected CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.20nMAssay Description:Inhibition of [3H]-NMS binding to human muscarinic acetylcholine receptor M1 expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibition of aurora AMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity against human Muscarinic acetylcholine receptor M1 in transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Compound was evaluated for inhibitory activity against human heart chymase (HHC)More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Inhibition of [3H]-NMS binding to human muscarinic acetylcholine receptor M1 expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.40nMAssay Description:Binding affinity against human muscarinic acetylcholine receptor M3 in transfected CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Inhibition of [3H]-NMS binding to human muscarinic acetylcholine receptor M1 expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Binding affinity against human Muscarinic acetylcholine receptor M1 in transfected CHO cellsMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.5nMAssay Description:Binding affinity against human Muscarinic acetylcholine receptor M1 in transfected CHO cellsMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Hokkaido Collaboration Center
Curated by ChEMBL
Hokkaido Collaboration Center
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Inhibition of recombinant human TNF-alpha converting enzyme (TACE)More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of recombinant human matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Binding affinity against human muscarinic acetylcholine receptor M3 in transfected CHO cellsMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Hokkaido Collaboration Center
Curated by ChEMBL
Hokkaido Collaboration Center
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Inhibition of human tumor necrosis factor alpha converting enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Inhibition of recombinant human matrix metalloproteinase-3More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Binding affinity against human Muscarinic acetylcholine receptor M1 in transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.81nMAssay Description:Inhibitory activity against matrix metalloprotease-1 (MMP-1)(recombinant human collagenase-1).More data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Hokkaido Collaboration Center
Curated by ChEMBL
Hokkaido Collaboration Center
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Inhibition of recombinant human TNF-alpha converting enzymeMore data for this Ligand-Target Pair
TargetDisintegrin and metalloproteinase domain-containing protein 17(Homo sapiens (Human))
Hokkaido Collaboration Center
Curated by ChEMBL
Hokkaido Collaboration Center
Curated by ChEMBL
Affinity DataKi: 1.90nMAssay Description:Inhibition of recombinant human TNF-alpha converting enzymeMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Banyu Tsukuba Research Institute In Collaboration With Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Ability to inhibit binding of [3H]-NMS was determined by receptor binding assay using membranes from chinese hamster ovary (CHO) cells expressing clo...More data for this Ligand-Target Pair