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Found 199 with Last Name = 'itoh' and Initial = 'n'
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50580223(CHEMBL5079957)
Affinity DataIC50:  3nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50580222(CHEMBL5076078)
Affinity DataIC50:  3.10nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50580225(CHEMBL5084053)
Affinity DataIC50:  3.80nMAssay Description:Antagonist activity at rat P2X3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Shionogi

Curated by ChEMBL
LigandPNGBDBM271626(US10065941, Compound I-127 | US9732060, Compound I...)
Affinity DataIC50:  4nMAssay Description:Antagonist activity at rat P2X3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM271626(US10065941, Compound I-127 | US9732060, Compound I...)
Affinity DataIC50:  4.20nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM271569(US10065941, Compound I-070 | US9732060, Compound I...)
Affinity DataIC50:  4.90nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM271893(US10065941, Compound R-208 | US9732060, Compound R...)
Affinity DataIC50:  5.20nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50580225(CHEMBL5084053)
Affinity DataIC50:  5.40nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50580221(CHEMBL5073093)
Affinity DataIC50:  5.60nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50580224(CHEMBL5090841)
Affinity DataIC50:  5.60nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM265772(US9718790, I-0616)
Affinity DataIC50:  5.70nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM271685(US10065941, Compound R-019 | US9732060, Compound R...)
Affinity DataIC50:  5.80nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563052(CHEMBL4748113)
Affinity DataIC50:  6.10nMAssay Description:Antagonist activity at rat P2X3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50580220(CHEMBL5086991)
Affinity DataIC50:  6.30nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183231(US9150546, I-401 | US9688643, I-401 | US9718790, I...)
Affinity DataIC50:  6.70nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183205(US9150546, I-369 | US9688643, I-369 | US9718790, I...)
Affinity DataIC50:  6.70nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183198(US9150546, I-362 | US9688643, I-362 | US9718790, I...)
Affinity DataIC50:  6.90nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183344(US9150546, I-518 | US9688643, I-518 | US9718790, I...)
Affinity DataIC50:  7nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM271805(US10065941, Compound R-120 | US9732060, Compound R...)
Affinity DataIC50:  7.70nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Shionogi

Curated by ChEMBL
LigandPNGBDBM50580221(CHEMBL5073093)
Affinity DataIC50:  7.70nMAssay Description:Antagonist activity at rat P2X3 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183287(US9150546, I-456 | US9688643, I-456 | US9718790, I...)
Affinity DataIC50:  7.80nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM271892(US10065941, Compound R-207 | US9732060, Compound R...)
Affinity DataIC50:  8.60nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183292(US9150546, I-461 | US9688643, I-461 | US9718790, I...)
Affinity DataIC50:  9nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183238(US9150546, I-408 | US9688643, I-408 | US9718790, I...)
Affinity DataIC50:  9.80nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM271767(US10065941, Compound R-078 | US9732060, Compound R...)
Affinity DataIC50:  9.90nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM265838(US9718790, I-0638)
Affinity DataIC50:  10nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183345(US9150546, I-519 | US9688643, I-519 | US9718790, I...)
Affinity DataIC50:  12nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183330(US9150546, I-500 | US9688643, I-500 | US9718790, I...)
Affinity DataIC50:  13nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183187(US9150546, I-351 | US9688643, I-351 | US9718790, I...)
Affinity DataIC50:  15nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM265821(US9718790, I-1284)
Affinity DataIC50:  15nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183291(US9150546, I-460 | US9688643, I-460 | US9718790, I...)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183364(US9150546, I-538 | US9688643, I-538 | US9718790, I...)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50563052(CHEMBL4748113)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM266400(US9718790, I-0837)
Affinity DataIC50:  17nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50580219(CHEMBL5074869)
Affinity DataIC50:  17nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183363(US9150546, I-537 | US9688643, I-537 | US9718790, I...)
Affinity DataIC50:  19nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM183191(US9150546, I-355 | US9688643, I-355 | US9718790, I...)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM265000(US9718790, I-0991)
Affinity DataIC50:  22nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM266159(US9718790, I-0750)
Affinity DataIC50:  22nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38224(US8546380, 1043 | US8633188, 1043)
Affinity DataIC50:  27nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38224(US8546380, 1043 | US8633188, 1043)
Affinity DataIC50:  27nMpH: 5.0 T: 2°CAssay Description:Zero point five μL of the test compounds (dissolved in N,N′-dimethylsulfoxide) were incubated with 48.5 μL of the fluorescence-quench...More data for this Ligand-Target Pair
TargetP2X purinoceptor 3(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50580218(CHEMBL5088459)
Affinity DataIC50:  31nMAssay Description:Antagonist activity at P2X3 receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38226(US8546380, 1199 | US8633188, 1199)
Affinity DataIC50:  32nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38226(US8546380, 1199 | US8633188, 1199)
Affinity DataIC50:  32nMpH: 5.0 T: 2°CAssay Description:Zero point five μL of the test compounds (dissolved in N,N′-dimethylsulfoxide) were incubated with 48.5 μL of the fluorescence-quench...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38220(US8546380, 1100 | US8633188, 1100)
Affinity DataIC50:  37nMpH: 5.0 T: 2°CAssay Description:Zero point five μL of the test compounds (dissolved in N,N′-dimethylsulfoxide) were incubated with 48.5 μL of the fluorescence-quench...More data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38220(US8546380, 1100 | US8633188, 1100)
Affinity DataIC50:  37nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103377(US8546380, 165 | US8633188, 165)
Affinity DataIC50:  39.4nMpH: 5.0 T: 2°CAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM103377(US8546380, 165 | US8633188, 165)
Affinity DataIC50:  39.4nMpH: 5.0 T: 2°CAssay Description:Zero point five μL of the test compounds (dissolved in N,N′-dimethylsulfoxide) were incubated with 48.5 μL of the fluorescence-quench...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38216(US8546380, 739 | US8633188, 739)
Affinity DataIC50:  49nMAssay Description:Inhibition assay using beta-Secretase activity.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Shionogi

US Patent
LigandPNGBDBM38216(US8546380, 739 | US8633188, 739)
Affinity DataIC50:  49nMpH: 5.0 T: 2°CAssay Description:Zero point five μL of the test compounds (dissolved in N,N′-dimethylsulfoxide) were incubated with 48.5 μL of the fluorescence-quench...More data for this Ligand-Target Pair
In DepthDetails US Patent
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