Affinity DataIC50: 20nMAssay Description:Inhibition of PAC3 homodimer (unknown origin) protein-protein interactionMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of PAC3 homodimerization by protein fragment complementation assayMore data for this Ligand-Target Pair
TargetTyrosyl-DNA phosphodiesterase 1(Homo sapiens (Human))
Biomedicinal Information Research Center (Birc)
Curated by ChEMBL
Biomedicinal Information Research Center (Birc)
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Inhibition of human Tdp1 using 3'-phosphate-(4-methylumbelliferone)-thymidine as substrate after 180 mins by spectrophotometryMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of PAC3 homodimer (unknown origin) protein-protein interactionMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of PAC1/PAC2 heterodimer (unknown origin) protein-protein interactionMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of PAC3 homodimer (unknown origin) protein-protein interactionMore data for this Ligand-Target Pair