Affinity DataKi: 0.0170nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataKi: 0.0200nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataKi: 0.0230nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0230nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0280nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataKi: 0.0290nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0330nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0330nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataKi: 0.0350nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0360nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0360nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataKi: 0.0380nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataKi: 0.0390nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0430nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0470nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.0570nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.0580nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0620nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0630nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0630nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.0670nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.0690nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 0.0700nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataKi: 0.0870nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.0960nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
Affinity DataKi: 0.118nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.119nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:In vitro binding affinity on D3 receptor is inhibition of binding of [125I]- NCQ 298 to Sf9 cells infected with recombinant baculovirusMore data for this Ligand-Target Pair
Affinity DataKi: 0.210nMAssay Description:In vitro binding affinity on D3 receptor is inhibition of binding of [125I]- NCQ 298 to Sf9 cells infected with recombinant baculovirusMore data for this Ligand-Target Pair
Affinity DataKi: 0.213nMAssay Description:Binding affinity towards Dopamine receptor D2 by displacing [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity for mouse opioid receptor muMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of human recombinant Aurora A after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Affinity DataKi: 0.450nMAssay Description:Affinity to opioid receptor kappa 1 using [3H]U-69593 as radioligand in homogenates of guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:In vitro binding affinity on D3 receptor is inhibition of binding of [125I]- NCQ 298 to Sf9 cells infected with recombinant baculovirusMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Pharmazeutisches Institut Der Universit£T Freiburg
Curated by ChEMBL
Affinity DataKi: 0.490nMAssay Description:Affinity to opioid receptor kappa 1 using [3H]U-69593 as radioligand in homogenates of guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataKi: 0.520nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
Affinity DataKi: 0.550nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.560nMAssay Description:Kinase assay using cyclin-dependant kinases (CDK).More data for this Ligand-Target Pair
Affinity DataKi: 0.630nMAssay Description:Inhibition of [125I]- NCQ 298 binding to D2 receptor of rat striatal tissueMore data for this Ligand-Target Pair
Affinity DataKi: 0.680nMAssay Description:The compound was tested in vitro for binding affinity towards 5-hydroxytryptamine 2 receptor by displacing [125]I-LSD radioligandMore data for this Ligand-Target Pair