Affinity DataKi: 0.830nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 181nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 207nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 252nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 342nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 432nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 733nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.01E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.04E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.06E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.23E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.25E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.41E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.62E+3nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.78E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.94E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.00E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.18E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.27E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.41E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.71E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.76E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A3 receptor in stably transfected HEK cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.10E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 4.57E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.45E+3nMAssay Description:Displacement of [3H]-CCPA from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.66E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 7.75E+3nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.08E+4nMAssay Description:Displacement of [3H]-NECA from human adenosine A2A receptor in stably transfected CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMpH: 8.0 T: 2°CAssay Description:The potency of inhibition on purified PARP enzyme was determined for selected compounds, and the potency was compared with that of 3-aminobenzamide (...More data for this Ligand-Target Pair
Affinity DataIC50: 10nMpH: 8.0 T: 2°CAssay Description:The potency of inhibition on purified PARP enzyme was determined for selected compounds, and the potency was compared with that of 3-aminobenzamide (...More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMpH: 8.0 T: 2°CAssay Description:The potency of inhibition on purified PARP enzyme was determined for selected compounds, and the potency was compared with that of 3-aminobenzamide (...More data for this Ligand-Target Pair
Affinity DataIC50: 98nMpH: 8.0 T: 2°CAssay Description:The potency of inhibition on purified PARP enzyme was determined for selected compounds, and the potency was compared with that of 3-aminobenzamide (...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMpH: 8.0 T: 2°CAssay Description:The potency of inhibition on purified PARP enzyme was determined for selected compounds, and the potency was compared with that of 3-aminobenzamide (...More data for this Ligand-Target Pair
Affinity DataIC50: 105nMpH: 8.0 T: 2°CAssay Description:The potency of inhibition on purified PARP enzyme was determined for selected compounds, and the potency was compared with that of 3-aminobenzamide (...More data for this Ligand-Target Pair
Affinity DataIC50: 107nMpH: 8.0 T: 2°CAssay Description:The potency of inhibition on purified PARP enzyme was determined for selected compounds, and the potency was compared with that of 3-aminobenzamide (...More data for this Ligand-Target Pair
Affinity DataIC50: 110nMpH: 8.0 T: 2°CAssay Description:The potency of inhibition on purified PARP enzyme was determined for selected compounds, and the potency was compared with that of 3-aminobenzamide (...More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMpH: 8.0 T: 2°CAssay Description:The potency of inhibition on purified PARP enzyme was determined for selected compounds, and the potency was compared with that of 3-aminobenzamide (...More data for this Ligand-Target Pair
Affinity DataIC50: 300nMpH: 8.0 T: 2°CAssay Description:The potency of inhibition on purified PARP enzyme was determined for selected compounds, and the potency was compared with that of 3-aminobenzamide (...More data for this Ligand-Target Pair
Affinity DataIC50: 394nMpH: 8.0 T: 2°CAssay Description:The potency of inhibition on purified PARP enzyme was determined for selected compounds, and the potency was compared with that of 3-aminobenzamide (...More data for this Ligand-Target Pair
Affinity DataIC50: 400nMpH: 8.0 T: 2°CAssay Description:The potency of inhibition on purified PARP enzyme was determined for selected compounds, and the potency was compared with that of 3-aminobenzamide (...More data for this Ligand-Target Pair
Affinity DataIC50: 450nMAssay Description:Tested for inhibition of poly(ADP-ribose) polymerase-1 (PARP-1) in mouse using Cell protection assayMore data for this Ligand-Target Pair
Affinity DataIC50: 450nMpH: 8.0 T: 2°CAssay Description:The potency of inhibition on purified PARP enzyme was determined for selected compounds, and the potency was compared with that of 3-aminobenzamide (...More data for this Ligand-Target Pair