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Found 53 with Last Name = 'janiczek-dolphin' and Initial = 'n'
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093310(3-{4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-3-ox...)
Affinity DataIC50:  3nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093310(3-{4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-3-ox...)
Affinity DataIC50:  4nMAssay Description:Compound was tested for in vitro inhibitory activity against ProthrombinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093302(3-{4-[4-(2,6-Dimethyl-piperidin-1-yl)-butyl]-3-oxo...)
Affinity DataIC50:  12nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093306(3-{4-[5-(2,5-Dimethyl-pyrrolidin-1-yl)-pentyl]-3-o...)
Affinity DataIC50:  48nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093313(3-[3-Oxo-4-(5-piperidin-1-yl-pentyl)-3,4-dihydro-2...)
Affinity DataIC50:  53nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093312(3-{4-[6-(2,6-Dimethyl-piperidin-1-yl)-hexyl]-3-oxo...)
Affinity DataIC50:  68nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093309(3-[4-(5-Diisopropylamino-pentyl)-3-oxo-3,4-dihydro...)
Affinity DataIC50:  120nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093299(3-[4-(5-Morpholin-4-yl-pentyl)-3-oxo-3,4-dihydro-2...)
Affinity DataIC50:  240nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093302(3-{4-[4-(2,6-Dimethyl-piperidin-1-yl)-butyl]-3-oxo...)
Affinity DataIC50:  300nMAssay Description:In vitro inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093310(3-{4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-3-ox...)
Affinity DataIC50:  330nMAssay Description:In vitro inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093306(3-{4-[5-(2,5-Dimethyl-pyrrolidin-1-yl)-pentyl]-3-o...)
Affinity DataIC50:  760nMAssay Description:In vitro inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093308(2-(3-Aminomethyl-phenyl)-4-[5-(2,6-dimethyl-piperi...)
Affinity DataIC50:  840nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093310(3-{4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-3-ox...)
Affinity DataIC50:  890nMAssay Description:Compound was tested for in vitro inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093306(3-{4-[5-(2,5-Dimethyl-pyrrolidin-1-yl)-pentyl]-3-o...)
Affinity DataIC50:  910nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093313(3-[3-Oxo-4-(5-piperidin-1-yl-pentyl)-3,4-dihydro-2...)
Affinity DataIC50:  990nMAssay Description:In vitro inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093302(3-{4-[4-(2,6-Dimethyl-piperidin-1-yl)-butyl]-3-oxo...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093299(3-[4-(5-Morpholin-4-yl-pentyl)-3-oxo-3,4-dihydro-2...)
Affinity DataIC50:  1.10E+3nMAssay Description:In vitro inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093309(3-[4-(5-Diisopropylamino-pentyl)-3-oxo-3,4-dihydro...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093309(3-[4-(5-Diisopropylamino-pentyl)-3-oxo-3,4-dihydro...)
Affinity DataIC50:  1.20E+3nMAssay Description:In vitro inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093320(3-{4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-3-ox...)
Affinity DataIC50:  1.50E+3nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093301(3-[4-(5-Dihexylamino-pentyl)-3-oxo-3,4-dihydro-2H-...)
Affinity DataIC50:  1.60E+3nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093318(4-{4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-3-ox...)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093301(3-[4-(5-Dihexylamino-pentyl)-3-oxo-3,4-dihydro-2H-...)
Affinity DataIC50:  1.90E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093312(3-{4-[6-(2,6-Dimethyl-piperidin-1-yl)-hexyl]-3-oxo...)
Affinity DataIC50:  2.10E+3nMAssay Description:In vitro inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093299(3-[4-(5-Morpholin-4-yl-pentyl)-3-oxo-3,4-dihydro-2...)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093301(3-[4-(5-Dihexylamino-pentyl)-3-oxo-3,4-dihydro-2H-...)
Affinity DataIC50:  2.20E+3nMAssay Description:Compound was tested for in vitro inhibitory activity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093301(3-[4-(5-Dihexylamino-pentyl)-3-oxo-3,4-dihydro-2H-...)
Affinity DataIC50:  2.50E+3nMAssay Description:In vitro inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093311(3-{4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-3-ox...)
Affinity DataIC50:  2.80E+3nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093313(3-[3-Oxo-4-(5-piperidin-1-yl-pentyl)-3,4-dihydro-2...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093317(3-[4-(5-Amino-pentyl)-3-oxo-3,4-dihydro-2H-benzo[1...)
Affinity DataIC50:  4.30E+3nMAssay Description:In vitro inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093314(4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-2-(4-me...)
Affinity DataIC50:  4.90E+3nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093312(3-{4-[6-(2,6-Dimethyl-piperidin-1-yl)-hexyl]-3-oxo...)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093319(3-{4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-3-ox...)
Affinity DataIC50:  5.60E+3nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093317(3-[4-(5-Amino-pentyl)-3-oxo-3,4-dihydro-2H-benzo[1...)
Affinity DataIC50:  6.30E+3nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093308(2-(3-Aminomethyl-phenyl)-4-[5-(2,6-dimethyl-piperi...)
Affinity DataIC50:  7.80E+3nMAssay Description:In vitro inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093318(4-{4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-3-ox...)
Affinity DataIC50:  7.90E+3nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093310(3-{4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-3-ox...)
Affinity DataIC50:  8.40E+3nMAssay Description:Compound was tested for in vitro inhibitory activity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093312(3-{4-[6-(2,6-Dimethyl-piperidin-1-yl)-hexyl]-3-oxo...)
Affinity DataIC50:  1.20E+4nMAssay Description:Compound was tested for in vitro inhibitory activity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093318(4-{4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-3-ox...)
Affinity DataIC50:  1.30E+4nMAssay Description:In vitro inhibitory activity against trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093304(2-(2-Chloro-phenyl)-4-[5-(2,6-dimethyl-piperidin-1...)
Affinity DataIC50:  1.60E+4nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093303(3-{4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-3-ox...)
Affinity DataIC50:  1.70E+4nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093313(3-[3-Oxo-4-(5-piperidin-1-yl-pentyl)-3,4-dihydro-2...)
Affinity DataIC50:  2.10E+4nMAssay Description:Compound was tested for in vitro inhibitory activity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin K-dependent protein C(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093310(3-{4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-3-ox...)
Affinity DataIC50:  2.30E+4nMAssay Description:Compound was tested for in vitro inhibitory activity against activated protein CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093305(2-(4-Chloro-phenyl)-4-[5-(2,6-dimethyl-piperidin-1...)
Affinity DataIC50:  2.30E+4nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093308(2-(3-Aminomethyl-phenyl)-4-[5-(2,6-dimethyl-piperi...)
Affinity DataIC50:  2.50E+4nMAssay Description:Compound was tested for in vitro inhibitory activity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093315(2-(3,4-Dichloro-phenyl)-4-[5-(2,6-dimethyl-piperid...)
Affinity DataIC50:  2.60E+4nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093300(4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-2-pheny...)
Affinity DataIC50:  2.70E+4nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093316(4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-2-p-tol...)
Affinity DataIC50:  2.80E+4nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093307(4-{4-[5-(2,6-Dimethyl-piperidin-1-yl)-pentyl]-3-ox...)
Affinity DataIC50:  3.40E+4nMAssay Description:In vitro inhibition of coagulation factor Xa.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50093302(3-{4-[4-(2,6-Dimethyl-piperidin-1-yl)-butyl]-3-oxo...)
Affinity DataIC50:  3.80E+4nMAssay Description:Compound was tested for in vitro inhibitory activity against plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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