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Found 532 with Last Name = 'jensen' and Initial = 'kg'
TargetAlpha-1A adrenergic receptor(CALF)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50426619(CHEMBL2326175)
Affinity DataKi:  0.160nMAssay Description:Displacement of [3H]prazosine from bovine alpha1A adrenoceptor expressed in BHK cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50122815(1-(2-{4-[1-(4-Fluoro-phenyl)-5-(2-methyl-2H-tetraz...)
Affinity DataKi:  0.230nMAssay Description:Displacement of [3H]prazosine from bovine alpha1A adrenoceptor expressed in BHK cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50426621(CHEMBL2325935)
Affinity DataKi:  0.280nMAssay Description:Displacement of [3H]prazosine from bovine alpha1A adrenoceptor expressed in BHK cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50426630(CHEMBL2325926)
Affinity DataKi:  0.320nMAssay Description:Displacement of [3H]prazosine from bovine alpha1A adrenoceptor expressed in BHK cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001786(1-(2-{4-[5-chloro-1-(4-fluorophenyl)-1H-indol-3-yl...)
Affinity DataKi:  0.330nMAssay Description:Displacement of [3H]prazosine from hamster alpha1B adrenoceptor expressed in Rat1 cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001786(1-(2-{4-[5-chloro-1-(4-fluorophenyl)-1H-indol-3-yl...)
Affinity DataKi:  0.370nMAssay Description:Displacement of [3H]prazosine from bovine alpha1A adrenoceptor expressed in BHK cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001786(1-(2-{4-[5-chloro-1-(4-fluorophenyl)-1H-indol-3-yl...)
Affinity DataKi:  0.450nMAssay Description:Displacement of [3H]spiperone from human dopamine D2 receptor expressed in CHO cells after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-1A adrenergic receptor(CALF)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50328477(1-(8-chloro-10,11-dihydrodibenzo[b,f]thiepin-10-yl...)
Affinity DataKi:  0.520nMAssay Description:Displacement of [3H]prazosine from bovine alpha1A adrenoceptor expressed in BHK cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50426620(CHEMBL2326176)
Affinity DataKi:  0.540nMAssay Description:Displacement of [3H]prazosine from bovine alpha1A adrenoceptor expressed in BHK cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50001786(1-(2-{4-[5-chloro-1-(4-fluorophenyl)-1H-indol-3-yl...)
Affinity DataKi:  0.660nMAssay Description:Displacement of [3H]prazosine from rat alpha1D adrenoceptor expressed in CHO cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50122815(1-(2-{4-[1-(4-Fluoro-phenyl)-5-(2-methyl-2H-tetraz...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]prazosine from hamster alpha1B adrenoceptor expressed in Rat1 cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337403(CHEMBL1682668 | methyl 1-(((1R,2S)-2-(benzyl(methy...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50400902(1-(2-(2,4-dimethylphenylsulfanyl)phenyl)piperazine...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity to human SERTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337411((1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50328477(1-(8-chloro-10,11-dihydrodibenzo[b,f]thiepin-10-yl...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]prazosine from hamster alpha1B adrenoceptor expressed in Rat1 cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337418((1S,2R)-1-(3,4-dichlorophenyl)-2-((3-(4-(N,N-dimet...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50122815(1-(2-{4-[1-(4-Fluoro-phenyl)-5-(2-methyl-2H-tetraz...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]prazosine from rat alpha1D adrenoceptor expressed in CHO cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50426624(CHEMBL2325932)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]prazosine from bovine alpha1A adrenoceptor expressed in BHK cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50328477(1-(8-chloro-10,11-dihydrodibenzo[b,f]thiepin-10-yl...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]prazosine from rat alpha1D adrenoceptor expressed in CHO cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50388667(CHEMBL2059323)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]raclopride from human D2L receptor expressed in CHO cells after 60 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(CALF)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50426628(CHEMBL2325928)
Affinity DataKi:  2.70nMAssay Description:Displacement of [3H]prazosine from bovine alpha1A adrenoceptor expressed in BHK cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM85330(CAS_68647 | NSC_68647 | ONDANSETRON | Ondansetron ...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]granisetron from human 5HT3A receptor expressed in HEK293 cells by filter binding assayMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337404((1S,2R)-N-benzyl-1-(3,4-dichlorophenyl)-2-((4-(3,3...)
Affinity DataKi:  2.80nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]raclopride from human D2L receptor expressed in CHO cells after 60 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAlpha-1A adrenergic receptor(CALF)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50122807(1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-[1,2,3...)
Affinity DataKi:  3nMAssay Description:Displacement of [3H]prazosine from bovine alpha1A adrenoceptor expressed in BHK cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337409((1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-...)
Affinity DataKi:  3.30nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337407(CHEMBL1682672 | N1-(1-(((1R,2S)-2-(benzyl(methyl)c...)
Affinity DataKi:  3.60nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50400902(1-(2-(2,4-dimethylphenylsulfanyl)phenyl)piperazine...)
Affinity DataKi:  3.70nMAssay Description:Binding affinity to human 5HT3A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337410((1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337401((1S,2R)-N-benzyl-1-(3,4-dichlorophenyl)-N-methyl-2...)
Affinity DataKi:  4.20nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337435(CHEMBL1682637 | rac-2-((4-acetamido-4-phenylpiperi...)
Affinity DataKi:  4.60nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337425(CHEMBL1682628 | rac-2-((4-acetamido-4-phenylpiperi...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50388674(OXIPEROMIDE)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]raclopride from human D2L receptor expressed in CHO cells after 60 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337405((1S,2R)-N-benzyl-1-(3,4-dichlorophenyl)-N-methyl-2...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337431((1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)met...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337416((1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-...)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337441(CHEMBL1682643 | rac-2-((4-acetamido-4-phenylpiperi...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337421((1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)met...)
Affinity DataKi:  5.90nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50122807(1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-[1,2,3...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]prazosine from hamster alpha1B adrenoceptor expressed in Rat1 cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337402((1S,2R)-N-benzyl-1-(3,4-dichlorophenyl)-N-methyl-2...)
Affinity DataKi:  6.10nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1B adrenergic receptor(C.H.O.)
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50426619(CHEMBL2326175)
Affinity DataKi:  6.40nMAssay Description:Displacement of [3H]prazosine from hamster alpha1B adrenoceptor expressed in Rat1 cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50388682(CHEMBL2059318)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]raclopride from human D2L receptor expressed in CHO cells after 60 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337397((1S,2R)-2-((4-acetamido-4-phenylpiperidin-1-yl)met...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50400899(CHEMBL2204363)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]granisetron from human 5HT3A receptor expressed in HEK293 cells by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337413((1S,2R)-1-(3,4-dichlorophenyl)-N-(4-fluorobenzyl)-...)
Affinity DataKi:  7.30nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337433(CHEMBL1681797 | rac-2-((4-acetamido-4-phenylpiperi...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337415((1S,2R)-1-(3,4-dichlorophenyl)-2-((4-(N,N-dimethyl...)
Affinity DataKi:  7.60nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337408((1S,2R)-N-benzyl-1-(3,4-dichlorophenyl)-N-methyl-2...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Rattus norvegicus (Rat))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50122807(1-(2-{4-[1-(4-Fluoro-phenyl)-5-(1-methyl-1H-[1,2,3...)
Affinity DataKi:  8.60nMAssay Description:Displacement of [3H]prazosine from rat alpha1D adrenoceptor expressed in CHO cells after 20 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Homo sapiens (Human))
H. Lundbeck

Curated by ChEMBL
LigandPNGBDBM50337417((1S,2R)-2-((4-(2-(azepan-1-yl)acetyl)piperazin-1-y...)
Affinity DataKi:  8.70nMAssay Description:Displacement of [3H]Lu AE93103 from human NK3 receptor expressed in BHK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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