Compile Data Set for Download or QSAR
maximum 50k data
Found 21 with Last Name = 'jessup' and Initial = 'r'
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280074((Z)-6-{(2S,4S,5R)-2-[1-Methyl-1-(4-methyl-2-nitro-...)
Affinity DataIC50:  18nMAssay Description:Inhibition of human Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280066((Z)-6-{(2S,4S,5R)-2-[1-Methyl-1-(4-methyl-2-nitro-...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280723(CHEMBL175801 | {6-Fluoro-9-[3-(6-pyridin-3-yl-hex-...)
Affinity DataIC50:  40nMAssay Description:Human microsomal Thromboxane synthase inhibition was determined by inhibiting TXB2 formation from [14C]- labelled arachidonic acidMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280073((Z)-6-{(2S,4S,5R)-4-(3-Methyl-3H-imidazol-4-yl)-2-...)
Affinity DataIC50:  50nMAssay Description:Inhibition of human Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280719(CHEMBL175538 | {6-Fluoro-9-[3-(5-pyridin-3-yl-pent...)
Affinity DataIC50:  50nMAssay Description:Human microsomal Thromboxane synthase inhibition was determined by inhibiting TXB2 formation from [14C]- labelled arachidonic acidMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280072((Z)-6-[(4S,5R)-2,2-Dimethyl-4-(3-methyl-3H-imidazo...)
Affinity DataIC50:  70nMAssay Description:Inhibition of human Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280063((Z)-6-((4S,5R)-2,2-Dimethyl-4-thiazol-5-yl-[1,3]di...)
Affinity DataIC50:  80nMAssay Description:Inhibition of human Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280720(CHEMBL425325 | {6-Fluoro-9-[3-(4-pyridin-3-yl-buto...)
Affinity DataIC50:  100nMAssay Description:Human microsomal Thromboxane synthase inhibition was determined by inhibiting TXB2 formation from [14C]- labelled arachidonic acidMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280070((Z)-6-((4S,5R)-2,2-Dimethyl-4-pyridin-3-yl-[1,3]di...)
Affinity DataIC50:  120nMAssay Description:Inhibition of human Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280724(CHEMBL362418 | {6-Fluoro-9-[3-((Z)-5-pyridin-3-yl-...)
Affinity DataIC50:  200nMAssay Description:Human microsomal Thromboxane synthase inhibition was determined by inhibiting TXB2 formation from [14C]- labelled arachidonic acidMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280721(CHEMBL174388 | {6-Fluoro-9-[3-(5-pyridin-3-yl-pent...)
Affinity DataIC50:  300nMAssay Description:Human microsomal Thromboxane synthase inhibition was determined by inhibiting TXB2 formation from [14C]- labelled arachidonic acidMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280722(CHEMBL172198 | {6-Fluoro-9-[4-(6-pyridin-3-yl-hex-...)
Affinity DataIC50:  400nMAssay Description:Human microsomal Thromboxane synthase inhibition was determined by inhibiting TXB2 formation from [14C]- labelled arachidonic acidMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280067((Z)-6-{(2S,4S,5R)-4-(3-Hexyl-3H-imidazol-4-yl)-2-[...)
Affinity DataIC50:  490nMAssay Description:Inhibition of human Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280726(CHEMBL177596 | {6-Fluoro-9-[3-(5-pyridin-3-yl-pent...)
Affinity DataIC50:  500nMAssay Description:Human microsomal Thromboxane synthase inhibition was determined by inhibiting TXB2 formation from [14C]- labelled arachidonic acidMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280725(CHEMBL427300 | {6-Fluoro-9-[4-(5-pyridin-3-yl-pent...)
Affinity DataIC50:  600nMAssay Description:Human microsomal Thromboxane synthase inhibition was determined by inhibiting TXB2 formation from [14C]- labelled arachidonic acidMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280069((Z)-6-[(4S,5R)-4-(3-Hexyl-3H-imidazol-4-yl)-2,2-di...)
Affinity DataIC50:  900nMAssay Description:Inhibition of human Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280071((Z)-6-((4S,5R)-2,2-Dimethyl-4-thiophen-2-yl-[1,3]d...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of human Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280068((Z)-6-((4S,5R)-2,2-Dimethyl-4-pyridazin-4-yl-[1,3]...)
Affinity DataIC50:  7.40E+3nMAssay Description:Inhibition of human Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280065((Z)-6-((4S,5R)-2,2-Dimethyl-4-pyrazin-2-yl-[1,3]di...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280064((Z)-6-((4S,5R)-2,2-Dimethyl-4-oxazol-5-yl-[1,3]dio...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article
TargetThromboxane-A synthase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280075((Z)-6-((4S,5R)-2,2-Dimethyl-4-pyrimidin-5-yl-[1,3]...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human Thromboxane A2 synthaseMore data for this Ligand-Target Pair
In DepthDetails Article