TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.140nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.180nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.630nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 0.700nMAssay Description:Inhibition Constant for 4-[125I]-IPBS binding to sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.32nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.46nMAssay Description:Inhibition Constant for 4-[125I]-IPBS binding to sigma 1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.54nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.64nMAssay Description:Binding affinity against sigma-1 receptor in guinea pig brain using [3H]-(+)-pentazocine as radioligand.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Binding affinity against sigma-1 receptor in guinea pig brain using [3H]-(+)-pentazocine as radioligand.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 3.02nMAssay Description:Binding affinity against sigma-1 receptor in guinea pig brain using [3H]-(+)-pentazocine as radioligandMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 3.11nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 3.70nMAssay Description:Compound was evaluated for its invitro competition binding studies using sigma-ligand (0.05-10000 nM) - [3H]-(+)-pentazocine (sigma1 receptor) in gui...More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 4.30nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 4.60nMAssay Description:Binding affinity against sigma receptor of MCF cellsMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 4.97nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 6.65nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 10.1nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 24.8nMAssay Description:Binding affinity against D-2 dopamine receptor in rat brain membranes using [3H]-(-)-sulpiride as radioligand.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 27.7nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 41.8nMAssay Description:Inhibition of [3H]-(+)-pentazocine binding to sigma-1 receptor in guinea pig brain membranesMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 60nMAssay Description:Binding affinity against sigma receptor of MCF cellsMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 63.4nMAssay Description:Binding affinity against D-2 dopamine receptor in rat brain membranes using [3H]-(-)-sulpiride as radioligand.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 152nMAssay Description:Compound was evaluated for its inhibition constant from the competition binding assays for sigma-1 receptor in guinea pig membranes.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 152nMAssay Description:Compound was evaluated for its inhibition constant from the competition binding assays for sigma-1 receptor in guinea pig membranes.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
George Washington University Medical Center
Curated by ChEMBL
George Washington University Medical Center
Curated by ChEMBL
Affinity DataKi: 382nMAssay Description:Binding affinity against D-2 dopamine receptor in rat brain membranes using [3H]-(-)-sulpiride as radioligand.More data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
The George Washington University Medical Center
Curated by ChEMBL
The George Washington University Medical Center
Curated by ChEMBL
Affinity DataKd: 38.2nMAssay Description:Binding affinity against MCF cells in the membrane preparation using radioligand binding assay.More data for this Ligand-Target Pair