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Found 698 with Last Name = 'josien' and Initial = 'h'
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50095105(4-{2-[4-(Benzo[1,3]dioxole-5-sulfonyl)-phenyl]-[1,...)
Affinity DataKi:  0.0100nMAssay Description:Antagonistic activity of the compound against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103771((4-{2-[4-(4-Methoxy-benzenesulfonyl)-phenyl]-[1,3]...)
Affinity DataKi:  0.140nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103774((5-Fluoro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy-ben...)
Affinity DataKi:  0.200nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103772((5,7-Difluoro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy...)
Affinity DataKi:  0.230nMAssay Description:Antagonistic activity of the compound against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103767((5,8-Difluoro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy...)
Affinity DataKi:  0.290nMAssay Description:Antagonistic activity of the compound against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103768((5-Bromo-naphthalen-1-yl)-(4-{2-[4-(4-methoxy-benz...)
Affinity DataKi:  0.510nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103773((4-Fluoro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy-ben...)
Affinity DataKi:  0.510nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50065428(CHEMBL3401350)
Affinity DataKi:  0.600nMAssay Description:Inhibition of renin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103775((6-Fluoro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy-ben...)
Affinity DataKi:  0.810nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103769((8-Fluoro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy-ben...)
Affinity DataKi:  0.990nMAssay Description:Antagonistic activity of the compound against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104933(CHEMBL105821 | {4-[(4-Bromo-phenyl)-ethoxyimino-me...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104940(CHEMBL323172 | {4-[(4-Bromo-phenyl)-methoxyimino-m...)
Affinity DataKi:  1.10nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103770((7-Fluoro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy-ben...)
Affinity DataKi:  1.20nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104942((4-Fluoro-naphthalen-1-yl)-{4-[4-(4-methoxy-benzen...)
Affinity DataKi:  1.30nMAssay Description:Inhibitory activity against Muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50103776((6-Chloro-naphthalen-1-yl)-(4-{2-[4-(4-methoxy-ben...)
Affinity DataKi:  1.40nMAssay Description:Antagonistic activity of the compound against muscarinic acetylcholine receptor M2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115512(CHEMBL324671 | {4-[(4-Bromo-phenyl)-methoxyimino-m...)
Affinity DataKi:  2nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115528((Z)-(4-((4-bromophenyl)(ethoxyimino)methyl)-4'-met...)
Affinity DataKi:  2nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50065395(CHEMBL3401345)
Affinity DataKi:  2nMAssay Description:Inhibition of renin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104931((4-{(4-Bromo-phenyl)-[(E)-ethoxyimino]-methyl}-4''...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50065426(CHEMBL3401348)
Affinity DataKi:  2.20nMAssay Description:Inhibition of renin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115511(CHEMBL321413 | {4-[(4-Bromo-phenyl)-ethoxyimino-me...)
Affinity DataKi:  3nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104936((2-Amino-6-chloro-phenyl)-{4-[(4-bromo-phenyl)-met...)
Affinity DataKi:  3.40nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115549((2,4-Dimethyl-1-oxy-pyridin-3-yl)-{4-[ethoxyimino-...)
Affinity DataKi:  3.80nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115550(CHEMBL109008 | {4-[(4-Bromo-phenyl)-isopropoxyimin...)
Affinity DataKi:  4nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115527((2,4-Dimethyl-1-oxy-pyridin-3-yl)-{4-[ethoxyimino-...)
Affinity DataKi:  4.40nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104938((2-Amino-6-methyl-phenyl)-{4-[(4-bromo-phenyl)-met...)
Affinity DataKi:  4.5nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115531((2,4-Dimethyl-1-oxy-pyridin-3-yl)-{4-[methoxyimino...)
Affinity DataKi:  5.30nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115548(CHEMBL343826 | CHEMBL419735 | {4-[(4-Chloro-phenyl...)
Affinity DataKi:  5.60nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50065424(CHEMBL3401346)
Affinity DataKi:  6nMAssay Description:Inhibition of renin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115517(CHEMBL110757 | {4-[(4-Bromo-phenyl)-ethoxyimino-me...)
Affinity DataKi:  7nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115522((2,4-Dimethyl-1-oxy-pyridin-3-yl)-{4-[methoxyimino...)
Affinity DataKi:  7.60nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115542(CHEMBL107154 | {4-[1-(4-Bromo-phenyl)-vinyl]-4'-me...)
Affinity DataKi:  8nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115529(CHEMBL418997 | {4-[(4-Bromo-phenyl)-tert-butoxyimi...)
Affinity DataKi:  9nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115526(CHEMBL107363 | {4-[(4-Bromo-phenyl)-(2-methoxy-eth...)
Affinity DataKi:  12nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50065425(CHEMBL3401347)
Affinity DataKi:  15nMAssay Description:Inhibition of renin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115538(4-[(Z)-(4-Bromophenyl)(ethoxyimino)methyl]-4'-meth...)
Affinity DataKi:  16nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104937(1'-(2-Hydroxy-6-methylbenzoyl)-4-[(Z)-(4-bromophen...)
Affinity DataKi:  18nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRenin(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50065393(CHEMBL3401344)
Affinity DataKi:  19nMAssay Description:Inhibition of renin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104941(CHEMBL106098 | CHEMBL138198 | {4-[(4-Bromo-phenyl)...)
Affinity DataKi:  19nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115537((2,4-Dimethyl-1-oxy-pyridin-3-yl)-{4-[ethoxyimino-...)
Affinity DataKi:  20nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115518(CHEMBL106099 | CHEMBL138143 | {4-[(4-Chloro-phenyl...)
Affinity DataKi:  24nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104929((4-{(4-Bromo-phenyl)-[(E)-methoxyimino]-methyl}-4'...)
Affinity DataKi:  25nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115543((2,6-Dimethyl-phenyl)-[4'-methyl-4-(4-trifluoromet...)
Affinity DataKi:  25nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115519(4-[(Z)-(4-Bromophenyl)(ethoxyimino)methyl]-4'-meth...)
Affinity DataKi:  26nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50104932(CHEMBL108569 | [4-(4-Bromo-phenoxy)-4'-methyl-[1,4...)
Affinity DataKi:  29nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115552(CHEMBL107018 | CHEMBL140922 | {4-[(4-Bromo-phenyl)...)
Affinity DataKi: >30nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115515(CHEMBL322267 | {4-[(4-Bromo-phenyl)-ethoxyimino-me...)
Affinity DataKi: >30nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115536((2,4-Dimethyl-1-oxy-pyridin-3-yl)-{4-[ethoxyimino-...)
Affinity DataKi:  30nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115551(CHEMBL108959 | {4-[(4-Bromo-phenyl)-ethoxyimino-me...)
Affinity DataKi: >30nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Mus musculus)
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50115525(CHEMBL106573 | {4-[(4-Bromo-phenyl)-phenoxyimino-m...)
Affinity DataKi: >30nMAssay Description:Inhibition of RANTES binding to Chemokine receptor type 5 receptor from NIH 3T3 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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