Compile Data Set for Download or QSAR
maximum 50k data
Found 69 with Last Name = 'ju' and Initial = 'hk'
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50029593(CHEMBL7162 | N-(2-(cyclohexyloxy)-4-nitrophenyl)me...)
Affinity DataIC50: <2nMAssay Description:Inhibitory activity against murine Prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50006811(2-(12-Hydroxy-5,10-dodecadiynyl)-3,5,6-trimethyl-p...)
Affinity DataIC50:  32nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145514((E)-1-Furan-2-yl-3-pyridin-2-yl-propenone | CHEMBL...)
Affinity DataIC50:  370nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50029593(CHEMBL7162 | N-(2-(cyclohexyloxy)-4-nitrophenyl)me...)
Affinity DataIC50:  1.67E+3nMAssay Description:Inhibitory activity against murine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145514((E)-1-Furan-2-yl-3-pyridin-2-yl-propenone | CHEMBL...)
Affinity DataIC50:  1.89E+3nMAssay Description:Inhibitory activity against murine Prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase I/type IB small subunit(Leishmania donovani)
Karunya University

LigandPNGBDBM246595(Camptothecin (CPT))
Affinity DataIC50:  2.80E+3nMpH: 7.5Assay Description:In the preincubation assay, CPT concentrations were 50 and 100 μM, whereas various concentrations of compounds were 25, 50 and 100 μM. LdTOP1LS...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145509((E)-1,3-Di-thiophen-2-yl-propenone | CHEMBL88104)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibitory activity against murine Prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase I/type IB small subunit(Leishmania donovani)
Karunya University

LigandPNGBDBM246595(Camptothecin (CPT))
Affinity DataIC50:  4.20E+3nMpH: 7.5Assay Description:In simultaneous relaxation assay, CPT concentrations were 50 and 100 μM, whereas concentration of compounds were 50, 100 and 200 μM. Relaxation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145509((E)-1,3-Di-thiophen-2-yl-propenone | CHEMBL88104)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145507((E)-1-Pyridin-2-yl-3-thiophen-3-yl-propenone | CHE...)
Affinity DataIC50:  5.22E+3nMAssay Description:Inhibitory activity against murine Prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145518((E)-3-Thiophen-3-yl-1-thiophen-2-yl-propenone | CH...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145515((E)-3-(3-Methyl-thiophen-2-yl)-1-pyridin-2-yl-prop...)
Affinity DataIC50:  6.51E+3nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145516((E)-3-Furan-2-yl-1-pyridin-2-yl-propenone | CHEMBL...)
Affinity DataIC50:  7.44E+3nMAssay Description:Inhibitory activity against murine Prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145506((E)-1-(5-Chloro-thiophen-2-yl)-3-furan-2-yl-propen...)
Affinity DataIC50:  7.52E+3nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145507((E)-1-Pyridin-2-yl-3-thiophen-3-yl-propenone | CHE...)
Affinity DataIC50:  7.60E+3nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145504((E)-3-Furan-3-yl-1-pyridin-3-yl-propenone | CHEMBL...)
Affinity DataIC50:  7.92E+3nMAssay Description:Inhibitory activity against murine Prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50047342((E)-3-Phenyl-1-pyridin-2-yl-propenone | 3-Phenyl-1...)
Affinity DataIC50:  8.13E+3nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145509((E)-1,3-Di-thiophen-2-yl-propenone | CHEMBL88104)
Affinity DataIC50:  9.01E+3nMAssay Description:Inhibitory activity against murine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145505((E)-1-Pyridin-2-yl-3-thiophen-2-yl-propenone | CHE...)
Affinity DataIC50:  9.01E+3nMAssay Description:Inhibitory activity against murine Prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145511((E)-1-Phenyl-3-(thiophen-2-yl)prop-2-en-1-one | (E...)
Affinity DataIC50:  9.02E+3nMAssay Description:Inhibitory activity against murine Prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145511((E)-1-Phenyl-3-(thiophen-2-yl)prop-2-en-1-one | (E...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145505((E)-1-Pyridin-2-yl-3-thiophen-2-yl-propenone | CHE...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145510((E)-1-Pyridin-3-yl-3-thiophen-3-yl-propenone | CHE...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against lipoxygenase-2 in micceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145505((E)-1-Pyridin-2-yl-3-thiophen-2-yl-propenone | CHE...)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibitory activity against murine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM29143(CHEMBL7976 | Chalcone 1 | Chalcone, 13 | cid_63776...)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibitory activity against murine Prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145513((E)-3-Furan-3-yl-1-pyridin-2-yl-propenone | CHEMBL...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory activity against cyclooxygenase-2 in miccMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145512((E)-3-Furan-2-yl-1-pyridin-3-yl-propenone | CHEMBL...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory activity against murine Prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145512((E)-3-Furan-2-yl-1-pyridin-3-yl-propenone | CHEMBL...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM29143(CHEMBL7976 | Chalcone 1 | Chalcone, 13 | cid_63776...)
Affinity DataIC50:  1.22E+4nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145519((E)-1,3-Di-furan-2-yl-propenone | CHEMBL315017)
Affinity DataIC50:  1.28E+4nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145507((E)-1-Pyridin-2-yl-3-thiophen-3-yl-propenone | CHE...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibitory activity against murine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase I/type IB small subunit(Leishmania donovani)
Karunya University

LigandPNGBDBM246594(Bi-lawsone analog, 3d)
Affinity DataIC50:  1.30E+4nMpH: 7.5Assay Description:In the preincubation assay, CPT concentrations were 50 and 100 μM, whereas various concentrations of compounds were 25, 50 and 100 μM. LdTOP1LS...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145510((E)-1-Pyridin-3-yl-3-thiophen-3-yl-propenone | CHE...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibitory activity against murine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145504((E)-3-Furan-3-yl-1-pyridin-3-yl-propenone | CHEMBL...)
Affinity DataIC50:  1.34E+4nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145516((E)-3-Furan-2-yl-1-pyridin-2-yl-propenone | CHEMBL...)
Affinity DataIC50:  1.35E+4nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145517((E)-3-Furan-2-yl-1-thiophen-2-yl-propenone | CHEMB...)
Affinity DataIC50:  1.37E+4nMAssay Description:Inhibitory activity against murine Prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145513((E)-3-Furan-3-yl-1-pyridin-2-yl-propenone | CHEMBL...)
Affinity DataIC50:  1.38E+4nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase I/type IB small subunit(Leishmania donovani)
Karunya University

LigandPNGBDBM246593(Bi-lawsone analog, 3c)
Affinity DataIC50:  1.40E+4nMpH: 7.5Assay Description:In the preincubation assay, CPT concentrations were 50 and 100 μM, whereas various concentrations of compounds were 25, 50 and 100 μM. LdTOP1LS...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyunsaturated fatty acid 5-lipoxygenase(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145517((E)-3-Furan-2-yl-1-thiophen-2-yl-propenone | CHEMB...)
Affinity DataIC50:  1.40E+4nMAssay Description:Inhibitory activity against murine lipoxygenase-2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145506((E)-1-(5-Chloro-thiophen-2-yl)-3-furan-2-yl-propen...)
Affinity DataIC50:  1.41E+4nMAssay Description:Inhibitory activity against murine Prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase I/type IB small subunit(Leishmania donovani)
Karunya University

LigandPNGBDBM246591(Bi-lawsone analog, 3a)
Affinity DataIC50:  1.60E+4nMpH: 7.5Assay Description:In the preincubation assay, CPT concentrations were 50 and 100 μM, whereas various concentrations of compounds were 25, 50 and 100 μM. LdTOP1LS...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase I/type IB small subunit(Leishmania donovani)
Karunya University

LigandPNGBDBM246592(Bi-lawsone analog, 3b)
Affinity DataIC50:  1.70E+4nMpH: 7.5Assay Description:In the preincubation assay, CPT concentrations were 50 and 100 μM, whereas various concentrations of compounds were 25, 50 and 100 μM. LdTOP1LS...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145510((E)-1-Pyridin-3-yl-3-thiophen-3-yl-propenone | CHE...)
Affinity DataIC50:  1.84E+4nMAssay Description:Inhibitory activity against murine Prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
University Of Madras

Curated by ChEMBL
LigandPNGBDBM50555459(CHEMBL4800560)
Affinity DataIC50:  1.91E+4nMAssay Description:Inhibition of recombinant human topoisomerase 2 assessed as decrease in relaxation of supercoiled pBlue-Script KS(+) plasmid DNA incubated for 30 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145504((E)-3-Furan-3-yl-1-pyridin-3-yl-propenone | CHEMBL...)
Affinity DataIC50:  2.10E+4nMAssay Description:Inhibitory activity against murine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM29143(CHEMBL7976 | Chalcone 1 | Chalcone, 13 | cid_63776...)
Affinity DataIC50:  2.21E+4nMAssay Description:Inhibitory activity against murine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
University Of Madras

Curated by ChEMBL
LigandPNGBDBM50555458(CHEMBL4753823)
Affinity DataIC50:  2.34E+4nMAssay Description:Inhibition of recombinant human topoisomerase 2 assessed as decrease in relaxation of supercoiled pBlue-Script KS(+) plasmid DNA incubated for 30 min...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Mus musculus (Mouse))
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145515((E)-3-(3-Methyl-thiophen-2-yl)-1-pyridin-2-yl-prop...)
Affinity DataIC50:  2.34E+4nMAssay Description:Inhibitory activity against murine Prostaglandin G/H synthase 2.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145516((E)-3-Furan-2-yl-1-pyridin-2-yl-propenone | CHEMBL...)
Affinity DataIC50:  2.36E+4nMAssay Description:Inhibitory activity against murine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Mus musculus)
Yeungnam University

Curated by ChEMBL
LigandPNGBDBM50145513((E)-3-Furan-3-yl-1-pyridin-2-yl-propenone | CHEMBL...)
Affinity DataIC50:  2.36E+4nMAssay Description:Inhibitory activity against murine prostaglandin G/H synthase 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 69 total ) | Next | Last >>
Jump to: