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Found 53 with Last Name = 'juan' and Initial = 'm'
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014005(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  15nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014007(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  69nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014009(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  505nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014013(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  603nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014012(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  913nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014004(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  1.00E+3nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014011(4-Ethyl-2,6-dimethyl-1,4-dihydro-pyridine-3,5-dica...)
Affinity DataKi:  1.01E+3nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014008(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  1.05E+3nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014010(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  2.09E+3nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50014006(2,4,6-Trimethyl-1,4-dihydro-pyridine-3,5-dicarboxy...)
Affinity DataKi:  4.41E+3nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlatelet-activating factor receptor(Cavia porcellus)
Alter

Curated by ChEMBL
LigandPNGBDBM50318494(3-ethyl 5-methyl 2,6-dimethyl-4-(3-nitrophenyl)-1,...)
Affinity DataKi:  7.33E+4nMAssay Description:Tested for inhibition of [3H]PAF binding to rabbit platelet Platelet activating factor receptor More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter

Curated by ChEMBL
LigandPNGBDBM50002644(2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataIC50:  1.40nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter

Curated by ChEMBL
LigandPNGBDBM50002628(4-(2,3-Dichloro-phenyl)-2,6-dimethyl-1,4-dihydro-p...)
Affinity DataIC50:  2.90nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter

Curated by ChEMBL
LigandPNGBDBM50336640((nifedipine) 2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-d...)
Affinity DataIC50:  2.90nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter

Curated by ChEMBL
LigandPNGBDBM50002603(2,6-Dimethyl-4-(3-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataIC50:  3.30nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter

Curated by ChEMBL
LigandPNGBDBM50002613(2,6-Dimethyl-4-(2-trifluoromethyl-phenyl)-1,4-dihy...)
Affinity DataIC50:  3.60nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter

Curated by ChEMBL
LigandPNGBDBM50002607(4-(2,3-Dichloro-phenyl)-2,6-dimethyl-1,4-dihydro-p...)
Affinity DataIC50:  5.10nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter

Curated by ChEMBL
LigandPNGBDBM50002626(2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataIC50:  5.10nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter

Curated by ChEMBL
LigandPNGBDBM50002600(2,6-Dimethyl-4-(3-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataIC50:  7.80nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter

Curated by ChEMBL
LigandPNGBDBM50002643(4-(2-Chloro-phenyl)-2,6-dimethyl-1,4-dihydro-pyrid...)
Affinity DataIC50:  10nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter

Curated by ChEMBL
LigandPNGBDBM50002635(2,6-Dimethyl-4-(3-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataIC50:  13nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter

Curated by ChEMBL
LigandPNGBDBM50002621(2,6-Dimethyl-4-(3-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataIC50:  15nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter

Curated by ChEMBL
LigandPNGBDBM50002580(2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataIC50:  25nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter

Curated by ChEMBL
LigandPNGBDBM50002631(2,6-Dimethyl-4-(3-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataIC50:  25nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter

Curated by ChEMBL
LigandPNGBDBM50002589(2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataIC50:  31nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333483(1-[5-tert-Butyl-3-(1,1-dioxo-1lambda*6*-thiomorpho...)
Affinity DataIC50:  34nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter

Curated by ChEMBL
LigandPNGBDBM50002604(2,6-Dimethyl-4-(2-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataIC50:  38nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
Alter

Curated by ChEMBL
LigandPNGBDBM50002637(2,6-Dimethyl-4-(3-nitro-phenyl)-1,4-dihydro-pyridi...)
Affinity DataIC50:  65nMAssay Description:Blockade of calcium-evoked contractions in depolarized aortic stripsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333468(1-(5-tert-butyl-3-((2-(dimethylamino)ethyl)carbamo...)
Affinity DataIC50:  521nMAssay Description:Inhibition of S6K1 in ribosomal protein S6 by whole cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333467(2-(3-1H-indazol-5-ylureido)-5-tert-butyl-N-cyclopr...)
Affinity DataIC50:  685nMAssay Description:Inhibition of S6K1 in ribosomal protein S6 by whole cell assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333484(1-[5-tert-Butyl-3-(1,1-dioxo-1lambda*6*-thiomorpho...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333473(2-(3-1H-indazol-5-ylureido)-5-tert-butyl-N-(2-meth...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333489(1-[5-tert-Butyl-3-(1,1-dioxo-1lambda*6*-thiomorpho...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333467(2-(3-1H-indazol-5-ylureido)-5-tert-butyl-N-cyclopr...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333468(1-(5-tert-butyl-3-((2-(dimethylamino)ethyl)carbamo...)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333472(2-(3-1H-indazol-5-ylureido)-5-tert-butyl-N-(2-hydr...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333475(1-(5-tert-butylthiophen-2-yl)-3-(1H-indazol-5-yl)u...)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333488(1-Benzo[4,5]furo[3,2-b]pyridin-8-yl-3-[5-tert-buty...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333487(1-[5-tert-Butyl-3-(1,1-dioxo-1lambda*6*-thiomorpho...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333486(1-[5-tert-Butyl-3-(1,1-dioxo-1lambda*6*-thiomorpho...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333485(1-[5-tert-Butyl-3-(1,1-dioxo-1lambda*6*-thiomorpho...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333490(1-[5-tert-Butyl-3-(1,1-dioxo-1lambda*6*-thiomorpho...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333482(2-(3-1H-indazol-5-ylureido)-N-(2-(dimethylamino)et...)
Affinity DataIC50:  2.90E+4nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333474(2-(3-1H-indazol-5-ylureido)-5-tert-butylthiophene-...)
Affinity DataIC50:  5.20E+4nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333481(2-(3-1H-indazol-5-ylureido)-N-(2-(dimethylamino)et...)
Affinity DataIC50:  6.20E+4nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333480(2-(3-1H-indazol-5-ylureido)-5-cyclopropyl-N-(2-(di...)
Affinity DataIC50:  7.00E+4nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333469(2-(3-1H-indazol-5-ylureido)-5-tert-butyl-N-(2-fluo...)
Affinity DataIC50:  1.91E+5nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333477((R)-2-(3-1H-indazol-5-ylureido)-N-(2-(dimethylamin...)
Affinity DataIC50:  1.96E+5nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333470(2-(3-1H-indazol-5-ylureido)-N-benzyl-5-tert-butylt...)
Affinity DataIC50:  2.01E+5nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRibosomal protein S6 kinase beta-1(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50333471(1-(5-tert-butyl-3-(morpholine-4-carbonyl)thiophen-...)
Affinity DataIC50:  2.07E+5nMAssay Description:Inhibition of S6K1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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